Search Results - "Poissonnet, Guillaume"

Ni-Catalyzed Reductive and Merged Photocatalytic Cross-Coupling Reactions toward sp3/sp2‑Functionalized Isoquinolones: Creating Diversity at C‑6 and C‑7 to Address Bioactive Analogues by Dumas, Adrien, Garsi, Jean-Baptiste, Poissonnet, Guillaume, Hanessian, Stephen

“…Naturally occurring isoquinolones have gained considerable attention over the years for their bioactive properties. While the late-stage introduction of…”
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Binding mode prediction and MD/MMPBSA-based free energy ranking for agonists of REV-ERBα/NCoR by Westermaier, Yvonne, Ruiz-Carmona, Sergio, Theret, Isabelle, Perron-Sierra, Françoise, Poissonnet, Guillaume, Dacquet, Catherine, Boutin, Jean A., Ducrot, Pierre, Barril, Xavier

“…The knowledge of the free energy of binding of small molecules to a macromolecular target is crucial in drug design as is the ability to predict the functional…”
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Ni-Catalyzed Reductive and Merged Photocatalytic Cross-Coupling Reactions toward sp 3 /sp 2 -Functionalized Isoquinolones: Creating Diversity at C-6 and C-7 to Address Bioactive Analogues by Dumas, Adrien, Garsi, Jean-Baptiste, Poissonnet, Guillaume, Hanessian, Stephen

“…Naturally occurring isoquinolones have gained considerable attention over the years for their bioactive properties. While the late-stage introduction of…”
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Practical Syntheses of 5-Trifluoromethyl-1H-indoles by Goldstein, Solo, Parmentier, Jean-Gilles, Poissonnet, Guillaume

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Binding mode prediction and MD/MMPBSA-based free energy ranking for agonists of REV-ERB[alpha]/NCoR by Westermaier, Yvonne, Ruiz-carmona, Sergio, Theret, Isabelle, Perron-sierra, Françoise, Poissonnet, Guillaume, Dacquet, Catherine, Boutin, Jean A, Ducrot, Pierre, Barril, Xavier

“…The knowledge of the free energy of binding of small molecules to a macromolecular target is crucial in drug design as is the ability to predict the functional…”
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Characterization of phospholipase C activity at h5-HT2C compared with h5-HT2B receptors: influence of novel ligands upon membrane-bound levels of [3H]phosphatidylinositols by Cussac, Didier, Newman-Tancredi, Adrian, Quentric, Yann, Carpentier, Nathalie, Poissonnet, Guillaume, Parmentier, Jean-Gilles, Goldstein, Solo, Millan, Mark J

“…Employing a novel, rapid and sensitive method for evaluation of phospholipase C (PLC) activity, the present study characterized the actions of diverse agonists…”
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Preparation and 1,3-Dipolar Cycloaddition Reactions of β-Carboline Azomethine Ylides:  A Direct Entry into C-1- and/or C-2-Functionalized Indolizino[8,7-b]indole Derivatives by Poissonnet, Guillaume, Théret-Bettiol, Marie-Hélène, Dodd, Robert H

“…Treatment of norharman with (trimethylsilyl)methyl triflate in dichloromethane gave 2-N-[(trimethylsilyl)methyl]-β-carboline triflate (10). The latter reacted…”
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A Simple and Convenient Synthesis of 1,2-Benzoxazoles Via Intramolecular Mitsunobu Reaction from Salicylaldoximes and Orthohydroxyarylketoximes by Poissonnet, Guillaume

“…Various substituted 1,2-benzoxazoles were prepared with good yields from salicylaldoximes and orthohydroxyphenylketoximes via intramolecular Mitsunobu reaction…”
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Characterization of phospholipase C activity at h5-HT 2C compared with h5-HT 2B receptors: influence of novel ligands upon membrane-bound levels of [ 3 H]phosphatidylinositols by Cussac, Didier, Newman-Tancredi, Adrian, Quentric, Yann, Carpentier, Nathalie, Poissonnet, Guillaume, Parmentier, Jean-Gilles, Goldstein, Solo, Millan, Mark

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Cytotoxic activities of novel hexahydroindolizino[8,7-b]indole derivatives prepared by 1,3-dipolar cycloaddition reactions of 3,4-dihydro-β-carboline ylides by Bertrand, Martial, Poissonnet, Guillaume, Théret-Bettiol, Marie-Hélène, Gaspard, Christiane, Werner, Georges H., Pfeiffer, Bruno, Renard, Pierre, Léonce, Stéphane, Dodd, Robert H.

“…A series of 1-cyano and 2-cyanohexahydroindolizino[8,7-b]indole derivatives was prepared by 1,3-dipolar cycloaddition of acrylonitrile with ylides derived from…”
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Mild Synthesis of N-Alkyl- and N-Alkyl-b-carboline Anhydoro-bases Using Trifluoromethanesulfonates by H. Dodd, Robert, Poissonnet, Guillaume, Potier, Pierre

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Synthesis of Functionalized Indolizino[8,7-b]indoles via 1,3-Dipolar Cycloaddition Reactions of 3,4-Dihydro-b-carboline Azomethine Ylides with Olefinic Derivatives by H. Dodd, Robert, Poissonnet, Guillaume, Th屍et, Marie-H四ene

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Synthesis of functionalized indolizino[8,7-b]indoles via 1,3-dipolar cycloaddition reactions of 3,4-dihydro-β-carboline azomethine ylides with olefinic derivatives by POISSONNET, G, THERET, M.-H, DODD, R. H

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Mild synthesis of N-alkyl- and N-acyl-β-carboline anhydro-bases using trifluoromethanesulfonates by DODD, R. H, POISSONNET, G, POTIER, P

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Synthesis and benzodiazepine receptor affinities of rigid analogs of 3-carboxy-.beta.-carbolines: demonstration that the benzodiazepine receptor recognizes preferentially the s-cis conformation of the 3-carboxy group by Dorey, Gilbert, Poissonnet, Guillaume, Potier, Marie Claude, De Carvalho, Lia Prado, Venault, Patrice, Chapouthier, Georges, Rossier, Jean, Potier, Pierre, Dodd, Robert H

“…1H-Indolo[3',2':4,5]pyrido[3,2-b]-2-penten-5-olide (6) and 1H,5H-indolo[3',2'-c]-6,7-dihydro-2-pyridone (7), rigid analogues of methyl…”
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