Search Results - "Patel, Champa B."

The discovery of 2-amino-3,5-diarylbenzamide inhibitors of IKK-α and IKK-β kinases by Christopher, John A., Avitabile, Barbara G., Bamborough, Paul, Champigny, Aurelie C., Cutler, Geoffrey J., Dyos, Susan L., Grace, Ken G., Kerns, Jeffrey K., Kitson, Jeremy D., Mellor, Geoffrey W., Morey, James V., Morse, Mary A., O’Malley, Carolyn F., Patel, Champa B., Probst, Nicholas, Rumsey, William, Smith, Clive A., Wilson, Michael J.

“…A potent and selective series of 2-amino-3,5-diarylbenzamide inhibitors of IKK-α and IKK-β is described. The most potent compounds are 8h, 8r and 8v, with…”
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5-(1 H-Benzimidazol-1-yl)-3-alkoxy-2-thiophenecarbonitriles as potent, selective, inhibitors of IKK-ε kinase by Bamborough, Paul, Christopher, John A., Cutler, Geoffrey J., Dickson, Marion C., Mellor, Geoffrey W., Morey, James V., Patel, Champa B., Shewchuk, Lisa M.

“…The identification and hit-to-lead exploration of a novel, potent, and selective series of substituted benzimidazole-thiophene carbonitrile inhibitors of IKK-…”
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