Search Results - "Paolo Lupattelli"

Last Decade of Unconventional Methodologies for the Synthesis of Substituted Benzofurans by Chiummiento, Lucia, D'Orsi, Rosarita, Funicello, Maria, Lupattelli, Paolo

“…This review describes the progress of the last decade on the synthesis of substituted benzofurans, which are useful scaffolds for the synthesis of numerous…”
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Synthesis and Evaluation of the Antioxidant Activity of Lipophilic Phenethyl Trifluoroacetate Esters by In Vitro ABTS, DPPH and in Cell-Culture DCF Assays by Bernini, Roberta, Barontini, Maurizio, Cis, Valentina, Carastro, Isabella, Tofani, Daniela, Chiodo, Rosa Anna, Lupattelli, Paolo, Incerpi, Sandra

“…Polyphenols are natural compounds showing a variety of health-promoting effects. Unfortunately, due to low lipid solubility, their applications in the…”
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PEGylated Liposomes Loaded with Carbamate Inhibitor ANP0903 Trigger Apoptosis by Enhancing ER Stress in HepG2 Cancer Cells by Caddeo, Carla, Miglionico, Rocchina, Rinaldi, Roberta, Nigro, Ilaria, Lamorte, Daniela, Chiummiento, Lucia, Lupattelli, Paolo, Funicello, Maria, D'Orsi, Rosarita, Valenti, Donatella, Santoro, Valentina, Fadda, Anna Maria, Bisaccia, Faustino, Vassallo, Antonio, Armentano, Maria Francesca

“…Liver cancer is one of the most common causes of cancer death worldwide. In recent years, substantial progress has been made in the development of systemic…”
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Practical and efficient ipso-iodination of arylboronic acids via KF/I2 system by Tramutola, Francesco, Chiummiento, Lucia, Funicello, Maria, Lupattelli, Paolo

“…[Display omitted] A facile and effective iododeboronation of variously substituted aryl and heteroarylboronic acids through activation and subsequent…”
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New Dihydroxytyrosyl Esters from Dicarboxylic Acids: Synthesis and Evaluation of the Antioxidant Activity In Vitro (ABTS) and in Cell-Cultures (DCF Assay) by Roma, Elia, Mattoni, Elena, Lupattelli, Paolo, Moeini, Seyed Sepehr, Gasperi, Tecla, Bernini, Roberta, Incerpi, Sandra, Tofani, Daniela

“…New dihydroxytyrosyl esters of dicarboxylic acids were synthesized from methyl orthoformate protected hydroxytyrosol and diacyl chlorides. New compounds were…”
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Targeting Viral and Cellular Cysteine Proteases for Treatment of New Variants of SARS-CoV-2 by Gentile, Davide, Chiummiento, Lucia, Santarsiere, Alessandro, Funicello, Maria, Lupattelli, Paolo, Rescifina, Antonio, Venuti, Assunta, Piperno, Anna, Sciortino, Maria Teresa, Pennisi, Rosamaria

“…The continuous emergence of SARS-CoV-2 variants caused the persistence of the COVID-19 epidemic and challenged the effectiveness of the existing vaccines. The…”
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Unveiling the Relationship between Structure and Anticancer Properties of Permethylated Anigopreissin A: A Study with Thirteen Analogues by Caivano, Ilaria, Santarsiere, Alessandro, Amati, Mario, Convertini, Paolo, Funicello, Maria, Lupattelli, Paolo, Chiummiento, Lucia, Santarsiero, Anna

“…Permethylated anigopreissin A (PAA), a fully protected form of the natural anigopreissin A, was found in our previous study to be active against several cancer…”
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The Pseudo-Symmetric N -benzyl Hydroxyethylamine Core in a New Series of Heteroarylcarboxyamide HIV-1 Pr Inhibitors: Synthesis, Molecular Modeling and Biological Evaluation by D'Orsi, Rosarita, Funicello, Maria, Laurita, Teresa, Lupattelli, Paolo, Berti, Federico, Chiummiento, Lucia

“…Here, we report the synthesis, enzyme inhibition and structure-activity relationship studies of a new potent class of HIV-1 protease inhibitors, which contain…”
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Asymmetric Synthesis of Spirooxindoles via Nucleophilic Epoxidation Promoted by Bifunctional Organocatalysts by Miceli, Martina, Mazziotta, Andrea, Palumbo, Chiara, Roma, Elia, Tosi, Eleonora, Longhi, Giovanna, Abbate, Sergio, Lupattelli, Paolo, Mazzeo, Giuseppe, Gasperi, Tecla

“…Taking into account the postulated reaction mechanism for the organocatalytic epoxidation of electron-poor olefins developed by our laboratory, we have…”
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Oxidized Palladium Supported on Ceria Nanorods for Catalytic Aerobic Oxidation of Benzyl Alcohol to Benzaldehyde in Protic Solvents by Seyed Sepehr Moeini, Chiara Battocchio, Stefano Casciardi, Igor Luisetto, Paolo Lupattelli, Daniela Tofani, Simonetta Tuti

“…In the present study, the catalytic activity of palladium oxide (PdOx) supported on ceria nanorods (CeO2-NR) for aerobic selective oxidation of benzyl alcohol…”
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Novel wild type and mutate HIV-1 protease inhibitors containing heteroaryl carboxamides in P2: Synthesis, biological evaluations and in silico ADME prediction by Francesca Armentano, Maria, Lupattelli, Paolo, Bisaccia, Faustino, D'Orsi, Rosarita, Miglionico, Rocchina, Nigro, Ilaria, Santarsiere, Alessandro, Berti, Federico, Funicello, Maria, Chiummiento, Lucia

“…[Display omitted] The Virus HIV-1 infection still represents a serious disease even if actually it is transformed in chronic pathology. Considering the crucial…”
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Two Novel Precursors of the HIV-1 Protease Inhibitor Darunavir Target the UPR/Proteasome System in Human Hepatocellular Carcinoma Cell Line HepG2 by Rinaldi, Roberta, Miglionico, Rocchina, Nigro, Ilaria, D'Orsi, Rosarita, Chiummiento, Lucia, Funicello, Maria, Lupattelli, Paolo, Laurenzana, Ilaria, Sgambato, Alessandro, Monné, Magnus, Bisaccia, Faustino, Armentano, Maria Francesca

“…Several pre-clinical and clinical reports suggest that HIV-1 protease inhibitors, in addition to the antiretroviral properties, possess pleiotropic…”
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Heterocycles in peptidomimetics and pseudopeptides: design and synthesis by Cerminara, Iole, Chiummiento, Lucia, Funicello, Maria, Guarnaccio, Ambra, Lupattelli, Paolo

“…This minireview provides a brief outline of the peculiar aspects of the preparation of peptidomimetic and pseudopeptidic structures containing heterocycles. In…”
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1,2‐Diarylethanols by Alternative Regioselective Reductive Ring‐Opening of 2,3‐Diaryloxiranes by Di Blasio, Nadia, Lopardo, Maria Teresa, Lupattelli, Paolo

“…Non‐symmetrical trans‐2,3‐diaryloxiranes have been regioselectively opened by catalytic hydrogenation over Pd/C, NaBH4/Pd and [Cp2TiCl]/H2O. Although in the…”
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Regio- and Stereoselective Ring Opening of 2,3-Diaryl Oxiranes by LiBr/Amberlyst 15:  A New Stereocontrolled Access to 1,2-Diaryl-2-bromo Alcohols by Solladié-Cavallo, Arlette, Lupattelli, Paolo, Bonini, Carlo

“…Both symmetrical and nonsymmetrical trans-2,3-diaryloxiranes are regio- and stereoselectively opened by the LiBr/Amberlyst 15 system. In the case of…”
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Synthesis and elaboration of trans 2,3-diaryloxiranes by Bonini, Carlo, Lupattelli, Paolo

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Single Route to Chiral syn- and anti-2-Amino-1,2-diphenylethanols via a New Stereodivergent Opening of trans-1,2-Diphenyloxirane by LUPATTELLI, Paolo, BONINI, Carlo, CARUSO, Leonilde, GAMBACORTA, Augusto

“…Oxiranyl ring opening of trans-stilbene oxide gave rise to anti- or syn-2-bromo-1,2-diphenylethanols, using either MgBr(2).Et(2)O or MgBr(2).Et(2)O, NaBr, and…”
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Desymmetrisation of meso-methylcyclooctanones. Highly enantioselective synthesis of C8 syn-isoprenoid and syn,syn-deoxypropionate subunits from a bicyclo[3.3.1]nonane precursor by Gambacorta, Augusto, Tofani, Daniela, Lupattelli, Paolo, Tafi, Andrea

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Electrotriggered Confined Self-assembly of Metal–Polyphenol Nanocoatings Using a Morphogenic Approach by Maerten, Clément, Lopez, Lionel, Lupattelli, Paolo, Rydzek, Gaulthier, Pronkin, Sergey, Schaaf, Pierre, Jierry, Loïc, Boulmedais, Fouzia

“…Supramolecular metal-phenolic thin films attract an increasing interest since they allow the design of new types of self-assembling materials, such as tunable…”
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A liquid chromatography-mass spectrometry method for the enantioselective multiresidue determination of nine chiral agrochemicals in urine using an enrichment procedure based on graphitized carbon black by Lucci, Elena, Antonelli, Lorenzo, Gherardi, Monica, Fanali, Chiara, Fanali, Salvatore, Scipioni, Anita, Lupattelli, Paolo, Gentili, Alessandra, Chankvetadze, Bezhan

“…Many agrochemicals are chiral molecules, and most of them are marketed as racemates or diastereomeric mixtures. Stereoisomers that are not the active…”
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