Search Results - "PRUNEAU, D"

Stable expression of human kinin B 1 receptor in 293 cells: pharmacological and functional characterization by Bastian, S., Loillier, B., Paquet, J. L., Pruneau, D.

“…We compared the binding properties of [ 3 H]‐desArg 10 ‐[Leu 9 ]‐kallidin, a radiolabelled kinin B 1 receptor antagonist, to membranes from IMR‐90 human…”
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Effect of warming and flow rate conditions of blood warmers on red blood cell integrity by Poder, T. G., Pruneau, D., Dorval, J., Thibault, L., Fisette, J.-F., Bédard, S. K., Jacques, A., Beauregard, P.

“…Background and Objectives Fluid warmers are routinely used to reduce the risk of hypothermia and cardiac complications associated with the infusion of cold…”
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Effects of LF 16-0687 Ms, a bradykinin B2 receptor antagonist, on brain edema formation and tissue damage in a rat model of temporary focal cerebral ischemia by ZAUSINGER, S, LUMENTA, D. B, PRUNEAU, D, SCHMID-ELSAESSER, R, PLESNILA, N, BAETHMANN, A

“…Bradykinin, an endogenous nonapeptide produced by activation of the kallikrein-kinin system, promotes neuronal tissue damage as well as disturbances in…”
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Activation of liver X receptors promotes lipid accumulation but does not alter insulin action in human skeletal muscle cells by Cozzone, D, Debard, C, Dif, N, Ricard, N, Disse, E, Vouillarmet, J, Rabasa-Lhoret, R, Laville, M, Pruneau, D, Rieusset, J, Lefai, E, Vidal, H

“…The aim of this study was to investigate the effects of liver X receptor (LXR) activation on lipid metabolism and insulin action in human skeletal muscle cells…”
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Detrimental role of bradykinin B2 receptor in a murine model of diffuse brain injury by Hellal, F, Pruneau, D, Palmier, B, Faye, P, Croci, N, Plotkine, M, Marchand-Verrecchia, C

“…Inhibition of the bradykinin B2 receptor type (B2R) has been shown to improve neurological outcome in models of focal traumatic brain injury. However, the…”
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Neuroprotective effects of a postischemic treatment with a bradykinin B2 receptor antagonist in a rat model of temporary focal cerebral ischemia by LUMENTA, D. B, PLESNILA, N, KLÄSNER, B, BAETHMANN, A, PRUNEAU, D, SCHMID-ELSAESSER, R, ZAUSINGER, S

“…Bradykinin, an endogenous nonapeptide produced by activation of the kallikrein-kinin system, promotes neuronal tissue damage as well as disturbances in…”
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Neuroprotective effects of a postischemic treatment with a bradykinin B 2 receptor antagonist in a rat model of temporary focal cerebral ischemia by Lumenta, D.B., Plesnila, N., Kläsner, B., Baethmann, A., Pruneau, D., Schmid-Elsaesser, R., Zausinger, S.

“…Bradykinin, an endogenous nonapeptide produced by activation of the kallikrein–kinin system, promotes neuronal tissue damage as well as disturbances in…”
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Antinociceptive pharmacology of N-[[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]methyl]-2-[2-[[(4-methoxy-2,6-dimethylphenyl) sulfonyl]methylamino]ethoxy]-N-methylacetamide, fumarate (LF22-0542), a novel nonpeptidic bradykinin B1 receptor antagonist by Porreca, F, Vanderah, T W, Guo, W, Barth, M, Dodey, P, Peyrou, V, Luccarini, J M, Junien, J-L, Pruneau, D

“…The antinociceptive pharmacology of N-[[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]methyl]-2-[2-[[(4-methoxy-2,6-dimethylphenyl)…”
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Stable expression of human kinin B1 receptor in 293 cells: pharmacological and functional characterization by Bastian, S., Loillier, B., Paquet, J. L., Pruneau, D.

“…1 We compared the binding properties of [3H]‐desArg10‐[Leu9]‐kallidin, a radiolabelled kinin B1 receptor antagonist, to membranes from IMR‐90 human embryonic…”
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Therapeutical efficacy of a novel non-peptide bradykinin B2 receptor antagonist on brain edema formation and ischemic tissue damage in focal cerebral ischemia by Zausinger, S, Lumenta, D B, Pruneau, D, Schmid-Elsaesser, R, Plesnila, N, Baethmann, A

“…Bradykinin has been identified as a mediator of secondary brain damage in acute insults. We currently studied neuroprotective properties of a bradykinin B2…”
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Pharmacological and molecular evidence for kinin B1 receptor expression in urinary bladder of cyclophosphamide‐treated rats by Belichard, P, Luccarini, J M, Defrêne, E, Faye, P, Franck, R M, Duclos, H, Paquet, J L, Pruneau, D

“…In the present study, we developed an experimental model of cystitis induced by cyclophosphamide (CYP). In order to characterize des‐Arg9‐BK‐induced…”
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A Rational Approach to the Design and Synthesis of a New Bradykinin B1 Receptor Antagonist by Bedos, Philippe, Amblard, Muriel, Subra, Gilles, Dodey, Pierre, Luccarini, Jean-Michel, Paquet, Jean-Luc, Pruneau, Didier, Aumelas, André, Martinez, Jean

“…We have previously synthesized a potent and selective B1 bradykinin receptor antagonist, JMV1645 (H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH), containing a…”
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Induction of kinin B1 receptor‐dependent vasoconstriction following balloon catheter injury to the rabbit carotid artery by Pruneau, D., Luccarini, J.M., Robert, C., Bélichard, P.

“…1 Balloon catheter injury to the rabbit carotid artery damaged the endothelium and induced neointima formation over 7 days. The area of intima, expressed as a…”
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Pharmacological and functional characterization of the guinea‐pig B2 bradykinin receptor stably expressed in CHO‐K1 cell line by Robert, C, Pruneau, D, Paquet, J ‐L

“…In the present study, pharmacological properties of a bradykinin B2 receptor amplified either from guinea‐pig ileum or lung and homologous to the previously…”
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Pharmacological characterization of the bradykinin B2 receptor: inter‐species variability and dissociation between binding and functional responses by Paquet, J ‐L, Luccarini, J ‐M, Fouchet, C, Defrêne, E, Loillier, B, Robert, C, Bélichard, P, Cremers, B, Pruneau, D

“…The present study addresses the differences in binding profiles and functional properties of the human and rat bradykinin (BK) B2 receptor using various kinin…”
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Induction of kinin B 1 receptor‐dependent vasoconstriction following balloon catheter injury to the rabbit carotid artery by Pruneau, D., Luccarini, J.M., Robert, C., Bélichard, P.

“…Balloon catheter injury to the rabbit carotid artery damaged the endothelium and induced neointima formation over 7 days. The area of intima, expressed as a…”
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LF16-0687 a novel non-peptide bradykinin B2 receptor antagonist reduces vasogenic brain edema from a focal lesion in rats by Schulz, J, Plesnila, N, Eriskat, J, Stoffel, M, Pruneau, D, Baethmann, A

“…Head injury world wide is still the most frequent cause of morbidity and mortality among the population under 45 years. Approximately 50% of patients dying…”
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Comparison of contractile responses to 5‐hydroxytryptamine and sumatriptan in human isolated coronary artery: synergy with the thromboxane A2‐receptor agonist, U46619 by Cocks, T.M., Kemp, B.K., Pruneau, D., Angus, J.A.

“…1 The interaction between the thromboxane A2 receptor agonist, U46619 and two 5‐hydroxytryptamine (5‐HT) receptor agonists, the non‐selective, naturally…”
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ω‐Conotoxin GVIA is a potent inhibitor of sympathetic neurogenic responses in rat small mesenteric arteries by Pruneau, D., Angus, J.A.

“…1 We have investigated the effects of the N‐type calcium channel blocker, ω‐conotoxin GVIA, on contractile responses to nerve stimulation, noradrenaline and…”
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Interleukin 8 (IL-8) induces the expression of kinin B1 receptor in human lung fibroblasts by Bastian, S, Paquet, J L, Robert, C, Cremers, B, Loillier, B, Larrivée, J F, Bachvarov, D R, Marceau, F, Pruneau, D

“…Kinin B1 receptors are induced by various inflammatory mediators. The aim of the present study was to investigate the effect of the CXC chemokine IL-8 on kinin…”
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