Search Results - "OZLEM TEMIZ-ARPACI"

Evaluation of Mutagenic Activities of Antimicrobial Benzoxazole Derivatives by Aydoğan, Zeliha, Foto, Fatma Zilifdar, Foto, Egemen, Temiz-Arpaci, Özlem, Diril, Nuran

“…Benzoxazoles are heterocyclic compounds containing fused benzene and oxazole rings, which have been reported to possess antibacterial, antitubercular,…”
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DFT, docking, MD simulation, and vibrational spectra with SERS analysis of a benzoxazole derivative: an anti-cancerous drug by Sheena Mary, Y., Shyma Mary, Y., Temiz-Arpaci, Ozlem, Yadav, Rohitash, Celik, Ismail

“…Spectroscopic, DFT, and SERS studies of antimicrobial bioactive 2-(p-bromophenyl)-5-(2-(4-(p-chlorophenyl)piperazine-1-yl)acetamido)benzoxazole (BCAB) have…”
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Synthesis, molecular docking and ADME prediction of some new benzimidazole carboxamidines derivatives as antimicrobial agents by Erol, Meryem, Celik, Ismail, Temiz-Arpaci, Ozlem, Goker, Hakan, Kaynak-Onurdag, Fatma, Okten, Suzan

“…In this study, 15 new 1 H -benzimidazole-5-carboxamidine derivative compounds that could be new antimicrobial agents were synthesized and their antimicrobial…”
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Spectroscopic, quantum mechanical and molecular docking studies of a new benzoxazole compound with an oxidoreductase enzyme and DNA by Zeyrek, Celal Tuğrul, Boyacioglu, Bahadir, Temiz-Arpaci, Özlem, Ünver, Hüseyin, Elmali, Ayhan

“…The spectroscopic, theoretical molecular structure, full vibrational band assignments, MEP, NBO, frontier molecular orbitals, and NLO effects, and molecular…”
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Synthesis, biological evaluation and 2D-QSAR analysis of benzoxazoles as antimicrobial agents by Ertan, Tugba, Yildiz, Ilkay, Tekiner-Gulbas, Betul, Bolelli, Kayhan, Temiz-Arpaci, Ozlem, Ozkan, Semiha, Kaynak, Fatma, Yalcin, Ismail, Aki, Esin

“…A new series of 5(or 6)-nitro/amino-2-(substituted phenyl/benzyl)benzoxazole derivatives ( 1a– 1m, 2a– 2l) were synthesized and evaluated for antibacterial and…”
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Some new bi- and ter-benzimidazole derivatives as topoisomerase I inhibitors by Alper, Sabiha, Temiz Arpaci, Özlem, Şener Aki, Esin, Yalçin, Ismail

“…The discovery of DNA topoisomerases has added a new dimension to the study of anticancer drugs. In the last years detailed investigation of bi- and…”
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Synthesis, antimicrobial activity, pharmacophore analysis of some new 2-(substitutedphenyl/benzyl)-5-[(2-benzofuryl)carboxamido]benzoxazoles by Alper-Hayta, Sabiha, Arisoy, Mustafa, Temiz-Arpaci, Özlem, Yildiz, Ilkay, Aki, Esin, Özkan, Semiha, Kaynak, Fatma

“…The synthesis and antimicrobial activity of a new series of 2-(substitutedphenyl/benzyl)-5-[(2-benzofuryl)carboxamido]benzoxazole derivatives 3– 12 were…”
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Vibrational spectroscopic studies and ab initio calculations of 5-methyl-2-( p-methylaminophenyl)benzoxazole by Ambujakshan, K.R., Madhavan, V.S., Varghese, Hema Tresa, Panicker, C. Yohannan, Temiz-Arpaci, Ozlem, Tekiner-Gulbas, Betul, Yildiz, Ilkay

“…FT-IR spectra of 5-methyl-2-( p-methylaminophenyl)benzoxazole was recorded and analysed. The vibrational frequencies of the compound have been computed using…”
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Synthesis and biological activity of some new benzoxazoles by Temiz-Arpacı, Özlem, Yıldız, İlkay, Özkan, Semiha, Kaynak, Fatma, Akı-Şener, Esin, Yalçın, İsmail

“…The synthesis and antimicrobial activity of a new series of 5-ethylsulphonyl-2-(substituted-phenyl/substituted-benzyl and/or phenylethyl)benzoxazole…”
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Synthesis and microbiological activity of some N-(2-hydroxy-4-substitutedphenyl)benzamides, phenylacetamides and furamides as the possible metabolites of antimicrobial active benzoxazoles by Akı-Şener, Esin, Bingöl, Kamuran K., Temiz-Arpacı, Özlem, Yalçın, İsmail, Altanlar, Nurten

“…The synthesis of some N-(2-hydroxy-4-substitutedphenyl)benzamides, phenylacetamides and furamides as the possible metabolites of benzoxazoles ( II 1– 15 ) was…”
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A Target Site for Template-Based Design of Measles Virus Entry Inhibitors by Plemper, Richard K., Erlandson, Karl J., Lakdawala, Ami S., Sun, Aiming, Prussia, Andrew, Boonsombat, Jutatip, Aki-Sener, Esin, Yalcin, Ismail, Yildiz, Ilkay, Temiz-Arpaci, Ozlem, Tekiner, Betul, Liotta, Dennis C., Snyder, James P., Compans, Richard W., Palese, Peter

“…Measles virus (MV) constitutes a principal cause of worldwide mortality, accounting for almost 1 million deaths annually. Although a live-attenuated vaccine…”
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Benzimidazole and Benzoxazole Derivatives Against Alzheimer's Disease by Faydalı, Nagihan, Arpacı, Özlem Temiz

“…Benzimidazole and benzoxazole derivatives are included in the category of medical drugs in a wide range of areas such as anticancer, anticoagulant,…”
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Synthesis and Antimicrobial Activity of New 2-[p-Substituted-benzyl]-5-[substituted-carbonylamino]benzoxazoles by Yildiz-Oren, Ilkay, Tekiner-Gulbas, Betul, Yalcin, Ismail, Temiz-Arpaci, Ozlem, Akı-Sener, Esin, Altanlar, Nurten

“…A series of 23 new 2‐[p‐substituted‐benzyl]‐5‐[p‐substituted‐phenyl/benzyl‐carbonylamino]benzoxazole derivatives has been synthesized by reacting…”
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Induction of Apoptosis and Necrosis by Resistance Modifiers Benzazoles and Benzoxazines on Tumour Cell Line Mouse Lymphoma L5718 Mdr+cells by ANDRAS VARGA, ESIN AKI-SENER, ISMAIL YALCIN, OZLEM TEMIZ-ARPACI, BETUL TEKINER-GULBAS, GEORGY CHEREPNEV, JOSEPH MOLNAR

“…Eighteen new fused heterocyclic compounds of benzazoles and benzoxazines were investigated for induction and inhibition of apoptosis on tumor cells (L5718,…”
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Design, synthesis, molecular docking, density functional theory and antimicrobial studies of some novel benzoxazole derivatives as structural bioisosteres of nucleotides by Erol, Meryem, Celik, Ismail, Temiz-Arpaci, Ozlem, Kaynak-Onurdag, Fatma, Okten, Suzan

“…A series of some novel 2-(p-tert-butylphenyl)-5-(3-substituted-propionamido)benzoxazole derivatives have been designed, synthesized, evaluated for…”
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Evaluation of Activity of Some 2,5-Disubstituted Benzoxazole Derivatives against Acetylcholinesterase, Butyrylcholinesterase and Tyrosinase: ADME Prediction, DFT and Comparative Molecular Docking Studies by Celik, Ismail, Erol, Meryem, Temiz Arpaci, Ozlem, Sezer Senol, Fatma, Erdogan Orhan, Ilkay

“…In this study, p-tert-butyl at position 2 and acetamide bridged 4-substituted piperazine/piperidine at position 5 bearing benzoxazole derivatives were…”
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Synthesis, quantum mechanical calculations, antimicrobial activities and molecular docking studies of five novel 2,5-disubstituted benzoxazole derivatives by Temiz-Arpaci, Ozlem, Zeyrek, Celal Tuğrul, Arisoy, Mustafa, Erol, Meryem, Celik, Ismail, Kaynak-Onurdag, Fatma

“…•The synthesis procedure of new five novel 2,5-disubstituted benzoxazole derivatives is given in detail.•The benzoxazole compounds have been characterized by…”
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Synthesis and Antimicrobial Activity of Some 2-[p-Substituted-phenyl]benzoxazol-5-yl-arylcarboxyamides by Temiz-Arpaci, Özlem, Aki-Şener, Esin, Yalçin, Ismail, Altanlar, Nurten

“…New 2‐[p‐substituted‐phenyl ]benzoxazol‐5‐yl‐arylcarboxyamides derivatives have been synthesized by reacting 5‐amino‐2‐[p‐substituted‐phenyl ]benzoxazoles with…”
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Spectroscopic, antimicrobial and computational study of novel benzoxazole derivative by Beegum, Shargina, Mary Y, Sheena, Panicker, C. Yohannan, Armaković, Stevan, Armaković, Sanja J., Arisoy, Mustafa, Temiz-Arpaci, Ozlem, Van Alsenoy, Christian

“…A benzoxazole derivative, 2-(p-methylphenyl)-5-(2-(4-ethylpiperazine-1-yl)acetamido) benzoxazole (PMPEPAB) has been synthesized and investigated for its…”
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Synthesis and Antimicrobial Evaluation of 2-(p-Substituted Phenyl)-5-[(4-substituted piperazin-1-yl)acetamido]-benzoxazoles by Arisoy, Mustafa, Temiz-Arpaci, Ozlem, Kaynak-Onurdag, Fatma, Ozgen, Selda

“…series of 2-(p-substituted phenyl)-5-(2-{4-[(p-chloro-fluorophenyl)=phenyl] piperazin-1-yl}- acetamido)-benzoxazoles were synthesized and tested for their…”
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