Search Results - "NAKAO, Kazuya"

All-optical 2-bit header recognition and packet switching using polarization bistable VCSELs by Hayashi, Daisuke, Nakao, Kazuya, Katayama, Takeo, Kawaguchi, Hitoshi

“…We propose and evaluate an all-optical 2-bit header recognition and packet switching method using two 1.55-µm polarization bistable vertical-cavity…”
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Structures of TMC-95A−D:  Novel Proteasome Inhibitors from Apiospora montagnei Sacc. TC 1093 by KOHNO, Jun, KOGUCHI, Yutaka, NISHIO, Maki, NAKAO, Kazuya, KURODA, Masataka, SHIMIZU, Ryo, OHNUKI, Tetsuo, KOMATSUBARA, Saburo

“…Four novel proteasome inhibitors, TMC-95A-D (1-4) have been isolated from the fermentation broth of Apiospora montagnei Sacc. TC 1093, isolated from a soil…”
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Virtual Screening System for Finding Structurally Diverse Hits by Active Learning by Fujiwara, Yukiko, Yamashita, Yoshiko, Osoda, Tsutomu, Asogawa, Minoru, Fukushima, Chiaki, Asao, Masaaki, Shimadzu, Hideshi, Nakao, Kazuya, Shimizu, Ryo

“…Two virtual screening strategies, “query by bagging” (QBag) and “query by bagging with descriptor-sampling” (QBagDS), based on active learning were devised…”
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The usefulness of an artificial membrane accumulation index for estimation of the bioconcentration factor of organophosphorus pesticides by Fujikawa, Masaaki, Nakao, Kazuya, Shimizu, Ryo, Akamatsu, Miki

“…The bioconcentration factor ( BCF) is an important ecotoxicological parameter that describes the accumulation of chemicals in organisms. As many studies have…”
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Novel Synthesis of (−)-Bestatin from L-Aspartic Acid by SEKI, Masahiko, NAKAO, Kazuya

“…Oxazoline-4-acetate derivative 3 that could be readily obtained from L-aspartic acid was subjected to highly stereoselective hydroxylation, and subsequent…”
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QSAR study on permeability of hydrophobic compounds with artificial membranes by Fujikawa, Masaaki, Nakao, Kazuya, Shimizu, Ryo, Akamatsu, Miki

“…To investigate PAMPA permeability of hydrophobic compounds, we experimentally measured the P app-pampa of compounds with high hydrophobicity, including several…”
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In silico Prediction of Human Oral Absorption Based on QSAR Analyses of PAMPA Permeability by Akamatsu, Miki, Fujikawa, Masaaki, Nakao, Kazuya, Shimizu, Ryo

“…The parallel artificial membrane permeation assay (PAMPA) was developed as a model for the prediction of transcellular permeation in the process of drug…”
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Optical control of neuronal firing via photoinduced electron transfer in donor-acceptor conjugates by Takano, Yuta, Numata, Tomohiro, Fujishima, Kazuto, Miyake, Kazuaki, Nakao, Kazuya, Grove, Wesley David, Inoue, Ryuji, Kengaku, Mineko, Sakaki, Shigeyoshi, Mori, Yasuo, Murakami, Tatsuya, Imahori, Hiroshi

“…A series of porphyrin-fullerene linked molecules has been synthesized to evaluate the effects of substituents and molecular structures on their…”
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QSAR application for the prediction of compound permeability with in silico descriptors in practical use by Nakao, Kazuya, Fujikawa, Masaaki, Shimizu, Ryo, Akamatsu, Miki

“…The parallel artificial membrane permeation assay (PAMPA) was developed as a model for the prediction of transcellular permeation in the process of drug…”
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Relationships between structure and high-throughput screening permeability of diverse drugs with artificial membranes: Application to prediction of Caco-2 cell permeability by Fujikawa, Masaaki, Ano, Rieko, Nakao, Kazuya, Shimizu, Ryo, Akamatsu, Miki

“…To evaluate the absorption of drugs with diverse structures across a membrane via the transcellular route, their permeability was measured by the parallel…”
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Optical control of neuronal firing viaphotoinduced electron transfer in donor-acceptor conjugates by Takano, Yuta, Numata, Tomohiro, Fujishima, Kazuto, Miyake, Kazuaki, Nakao, Kazuya, Grove, Wesley David, Inoue, Ryuji, Kengaku, Mineko, Sakaki, Shigeyoshi, Mori, Yasuo, Murakami, Tatsuya, Imahori, Hiroshi

“…A series of porphyrin-fullerene linked molecules has been synthesized to evaluate the effects of substituents and molecular structures on their…”
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Optical control of neuronal firing via photoinduced electron transfer in donor–acceptor conjugates† †Electronic supplementary information (ESI) available: Experimental procedures and spectroscopic data for all new compounds, supplementary characterizations, and optimized structures by theoretical calculations. See DOI: 10.1039/c5sc04135j by Takano, Yuta, Numata, Tomohiro, Fujishima, Kazuto, Miyake, Kazuaki, Nakao, Kazuya, Grove, Wesley David, Inoue, Ryuji, Kengaku, Mineko, Sakaki, Shigeyoshi, Mori, Yasuo, Murakami, Tatsuya, Imahori, Hiroshi

“…A rationally designed donor–acceptor conjugate efficiently generates a photoinduced charge-separated state in a cellular environment, achieving photoinduction…”
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Drug Screening of GPCR Using Active Learning by Fujiwara, Yukiko, Yamashita, Yoshiko, Osoda, Tsutomu, Asogawa, Minoru, Doi, Shun, Asao, Masaaki, Kushiyama, Emi, Nakao, Kazuya, Kuroda, Masataka, Wada, Kazuteru, Ogaru, Takanori, Fukushima, Chiaki, Shimizu, Ryo

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Optical control of neuronal firing photoinduced electron transfer in donor-acceptor conjugates by Takano, Yuta, Numata, Tomohiro, Fujishima, Kazuto, Miyake, Kazuaki, Nakao, Kazuya, Grove, Wesley David, Inoue, Ryuji, Kengaku, Mineko, Sakaki, Shigeyoshi, Mori, Yasuo, Murakami, Tatsuya, Imahori, Hiroshi

“…A series of porphyrinfullerene linked molecules has been synthesized to evaluate the effects of substituents and molecular structures on their…”
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Novel hydroxyphenylurea dual inhibitor against Acyl-CoA by Nakao, Kazuya, Kubota, Hitoshi, Yasuhara, Mikiko, Saito, Keiko, Suzuki, Toshikazu, Ohmizu, Hiroshi, Shimizu, Ryo

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Erratum to “( Z)-selective β-bromination of N-formyl- α, β-dehydroamino acid esters” [Tetrahedron 52 (1996) 5751] by Yamada, Masaki, Nakao, Kazuya, Fukui, Toshio, Nunami, Ken-ichi

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Structures of TMC-95A−D:  Novel Proteasome Inhibitors from Apiospora m ontagnei Sacc. TC 1093 by Kohno, Jun, Koguchi, Yutaka, Nishio, Maki, Nakao, Kazuya, Kuroda, Masataka, Shimizu, Ryo, Ohnuki, Tetsuo, Komatsubara, Saburo

“…Four novel proteasome inhibitors, TMC-95A−D (1−4) have been isolated from the fermentation broth of Apiospora montagnei Sacc. TC 1093, isolated from a soil…”
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Novel hydroxyphenylurea dual inhibitor against Acyl-CoA: cholesterol acyltransferase (ACAT) and low density lipoprotein (LDL) oxidation as antiatherosclerotic agent by Nakao, Kazuya, Kubota, Hitoshi, Yasuhara, Mikiko, Saito, Keiko, Suzuki, Toshikazu, Ohmizu, Hiroshi, Shimizu, Ryo

“…Novel hydroxyphenylurea derivatives were synthesized and their inhibitory potency evaluated against acyl-CoA: cholesterol acyltransferase (ACAT). Quantitative…”
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Quantitative Structure–Activity Analyses of Novel Hydroxyphenylurea Derivatives as Antioxidants by Nakao, Kazuya, Shimizu, Ryo, Kubota, Hitoshi, Yasuhara, Mikiko, Hashimura, Yoshimasa, Suzuki, Toshikazu, Fujita, Toshio, Ohmizu, Hiroshi

“…A series of substituted hydroxyphenylureas was synthesized, the chemical structure of which was designed based on structures of natural antioxidants, vitamin E…”
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(Z)-selective β-bromination ofN-formyl-α, β-dehydroamino acid esters by Yamada, Masaki, Nakao, Kazuya, Fukui, Toshio, Nunami, Ken-ichi

“…Stereoselective β-bromination ofN-formyl-α, β-dehydroamino acid esters 5 was investigated. A reaction of 5 with NBS affordedα-bromo-N-formylimines 10 which…”
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