Search Results - "Néliat, G"

SR141716A, a potent and selective antagonist of the brain cannabinoid receptor by Rinaldi-Carmona, Murielle, Barth, Francis, Héaulme, Michel, Shire, David, Calandra, Bernard, Congy, Christian, Martinez, Serge, Maruani, Jeanne, Néliat, Gervais, Caput, Daniel, Ferrara, Pascual, Soubrié, Philippe, Brelière, Jean Claude, Le Fur, Gérard

“…SR141716A is the first selective and orally active antagonist of the brain cannabinoid receptor. This compound displays nanomolar affinity for the central…”
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Genistein and daidzein modulate in vitro rat uterine contractile activity by Picherit, C, Dalle, M, Néliat, G, Lebecque, P, Davicco, M.J, Barlet, J.P, Coxam, V

“…The present study investigated the effect of genistein, daidzein and estradiol on in vitro rat uterine responsiveness to oxytocin (OT) and PGF 2α or luprostiol…”
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A potent and selective non-peptide antagonist of the neurokinin A (NK2) receptor by Emonds-Alt, X, Vilain, P, Goulaouic, P, Proietto, V, Van Broeck, D, Advenier, C, Naline, E, Neliat, G, Le Fur, G, Brelière, J C

“…SR 48968 is a potent and selective non-peptide antagonist of the neurokinin A (NK2) receptor. SR 48968 selectively inhibited neurokinin A binding to its…”
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The naphtosultam derivative RP 62203 (fananserin) has high affinity for the dopamine D4 receptor by HEUILLET, E, PETITET, F, MIGNAMI, S, MALLERON, J.-L, LAVAYRE, J, NELIAT, G, DOBLE, A, BLANCHARD, J.-C

“…The dopamine D4 receptor is a potential target for novel antipsychotic drugs. Most available compounds with affinity for the dopamine D4 receptor also bind to…”
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Biochemical and pharmacological properties of SR 46349B, a new potent and selective 5-hydroxytryptamine2 receptor antagonist by Rinaldi-Carmona, M, Congy, C, Santucci, V, Simiand, J, Gautret, B, Neliat, G, Labeeuw, B, Le Fur, G, Soubrie, P, Breliere, J C

“…A new potent, selective and p.o. active serotonergic [5-hydroxytryptamine (5-HT2)] receptor antagonist, SR 46349B [trans,…”
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Neurokinin A (NK2) receptor revisited with SR 48968, a potent non-peptide antagonist by Advenier, C, Rouissi, N, Nguyen, Q T, Emonds-Alt, X, Breliere, J C, Neliat, G, Naline, E, Regoli, D

“…SR 48968, a new non-peptide antagonist of NK2 receptors, has been tested in a variety of isolated smooth muscle preparations from rats, guinea pigs, rabbits,…”
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PK 11195, an antagonist of peripheral type benzodiazepine receptors, modulates Bay K8644 sensitive but not beta- or H2-receptor sensitive voltage operated calcium channels in the guinea pig heart by Mestre, M, Carriot, T, Néliat, G, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Doble, A, Le Fur, G

“…In a partially depolarized guinea pig papillary muscle preparation, BAY K8644 stimulated voltage-operated calcium channels, promoting slow action potentials;…”
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Functional modulation of gamma-aminobutyric acid A receptors by etifoxine and allopregnanolone in rodents by Verleye, M., Schlichter, R., Neliat, G., Pansart, Y., Gillardin, J.M.

“…We looked for an interaction between etifoxine and the neurosteroid allopregnanolone at central gamma-aminobutyric acid (GABA A) receptors. Etifoxine (2 μM)…”
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Functional modulation of gamma-aminobutyric acidA receptors by etifoxine and allopregnanolone in rodents by VERLEYE, M, SCHLICHTER, R, NELIAT, G, PANSART, Y, GILLARDIN, J. M

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Up‐regulation of [3H]‐des‐Arg10‐kallidin binding to the bradykinin B1 receptor by interleukin‐1β in isolated smooth muscle cells: correlation with B1 agonist‐induced PGI2 production by Galizzi, J.P., Bodinier, M.C., Chapelain, B., Ly, S.M., Coussy, L., Giraud, S., Neliat, G., Jean, T.

“…1 Binding of the specific bradykinin B1 receptor agonist, [3H]‐des‐Arg10‐kallidin (‐KD) was investigated in smooth muscle cells (SMC) isolated from rabbit…”
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Biochemical and pharmacological activities of SR 144190, a new potent non-peptide tachykinin NK2 receptor antagonist by EMONDS-ALT, X, ADVENIER, C, PROIETTO, V, VAN BROECK, D, VILAIN, P, SOUBRIE, P, LE FUR, G, MAFFRAND, J. P, BRELIERE, J. C, COGNON, C, CROCI, T, DAOUI, S, DUCOUX, J. P, LANDI, M, NALINE, E, NELIAT, G, PONCELET, M

“…(R)-3-(1-[2-(4-benzoyl-2-(3,4-difluorophenyl)-morpholin-2-yl)- ethyl]-4-phenylpiperidin-4-yl)-1-dimethylurea (SR 144190) is a new non-peptide antagonist of…”
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Interleukin-1 impairs both vascular contraction and relaxation in rabbit isolated aorta by Robert, R, Chapelain, B, Jean, T, Néliat, G

“…Incubation of rabbit aortic rings with interleukin-1 (100 U/ml) in vitro led to a depressed contractile response to norepinephrine, whether the endothelium was…”
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Lack of Effect of Repeated Administration of Milnacipran, a Double Noradrenaline and Serotonin Reuptake Inhibitor, on the β-adrenoceptor-linked Adenylate Cyclase System in the Rat Cerebral Cortex by NELIAT, G., BODINIER, M.-C., PANCONI, E., BRILEY, M.

“…The effects of subacute administration of the double noradrenaline and serotonin uptake inhibitor antidepressant, milnacipran, and the tricyclic…”
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Modulation of the spontaneous transient outward currents by histamine in single vascular smooth muscle cells by Neliat, G, Masson, F, Gargouil, Y M

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Different effects of interleukin-1 on reactivity of arterial vessels isolated from various vascular beds in the rabbit by Robert, R, Chapelain, B, Néliat, G

“…During septic shock, arterial smooth muscle is thought to be hyporeactive to vasoconstrictors. This hyporeactivity, however, seems to be different from one…”
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In vitro and in vivo biological activities of SR140333, a novel potent non-peptide tachykinin NK1 receptor antagonist by Emonds-Alt, X, Doutremepuich, J D, Heaulme, M, Neliat, G, Santucci, V, Steinberg, R, Vilain, P, Bichon, D, Ducoux, J P, Proietto, V

“…(S)1-(2-[3-(3,4-dichlorophenyl)-1-(3-isopropoxyphenylacetyl)pip eridin-3- yl]ethyl)-4-phenyl-1-azoniabicyclo[2.2.2]octane chloride (SR140333) is a new…”
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Effects of butoprozine on ionic currents in frog atrial and ferret ventricular fibres. Comparison with amiodarone and verapamil by Néliat, G, Ducouret, P, Moreau, M, Gargouïl, Y M

“…The effects of butoprozine on cardiac membrane currents of frog atrial and ferret ventricular fibres were investigated in voltage clamp conditions by means of…”
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SR120819A, an orally-active and selective neuropeptide Y Y1 receptor antagonist by Serradeil-Le Gal, Claudine, Valette, Gérard, Rouby, Pierre-Eric, Pellet, Alain, Oury-Donat, Florence, Brossard, Gabrielle, Lespy, Liliane, Marty, Eléonore, Neliat, Gervais, de Cointet, Paul, Maffrand, Jean-Pierre, Le Fur, Gérard

“…An orally-active antagonist of neuropeptide Y (NPY) Y 1 receptors, SR 120819A, has been characterized. This compound displays highly selective and competitive…”
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Electrophysiological effects of butoprozine on isolated heart preparations. Comparison with amiodarone and verapamil by Néliat, G, Moreau, M, Ducouret, P, Gargouïl, Y M

“…The electrophysiological effects of butoprozine, a relatively new antiarrhythmic agent, were investigated in sheep cardiac Purkinje fibres using a…”
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Functional modulation of gamma-aminobutyric acid sub(A) receptors by etifoxine and allopregnanolone in rodents by Verleye, M, Schlichter, R, Neliat, G, Pansart, Y, Gillardin, J M

“…We looked for an interaction between etifoxine and the neurosteroid allopregnanolone at central gamma-aminobutyric acid (GABA sub(A)) receptors. Etifoxine (2…”
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