Search Results - "Mukkanti, Kagga"

An Improved and Scalable Process for Celecoxib: A Selective Cyclooxygenase-2 Inhibitor by Reddy, Anumula Raghupathi, Sampath, Alla, Goverdhan, Gilla, Yakambaram, Bojja, Mukkanti, Kagga, Reddy, Padi Pratap

“…An improved, scalable and commercially viable process is developed for an active pharmaceutical ingredient, celecoxib…”
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Regioselective synthesis of isoxazole–mercaptobenzimidazole hybrids and their in vivo analgesic and anti-inflammatory activity studies by Kankala, Shravankumar, Kankala, Ranjith Kumar, Gundepaka, Prasad, Thota, Niranjan, Nerella, Srinivas, Gangula, Mohan Rao, Guguloth, Hanmanthu, Kagga, Mukkanti, Vadde, Ravinder, Vasam, Chandra Sekhar

“…Regioselective synthesis of isoxazole–mercaptobenzimidazole hybrids and their efficiency in in vivo analgesic and anti-inflammatory activity was described. A…”
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Microwave-assisted Claisen rearrangement of naphthyl 2-propynyl ethers: synthesis of naphthofurans by Prasada Rao Lingam, V.S., Dahale, Dnyaneshwar H., Mukkanti, Kagga, Gopalan, Balasubramanian, Thomas, Abraham

“…An efficient two-step approach for the synthesis of naphtho[1,2-b]furans and naphtho[2,1-b]furans has been developed. Various functionalized propargyl alcohols…”
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An Improved Process for Pioglitazone and Its Pharmaceutically Acceptable Salt by Madivada, Lokeswara Rao, Anumala, Raghupathi Reddy, Gilla, Goverdhan, Alla, Sampath, Charagondla, Kavitha, Kagga, Mukkanti, Bhattacharya, Apurba, Bandichhor, Rakeshwar

“…An improved process for pioglitazone (1) is described. The process features high-yielding transformations employing inexpensive reagents and recoverable…”
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Anti-neuroinflammatory activity of 1,5-benzodiazepine derivatives by Ha, Sang Keun, Shobha, Donthabhaktuni, Moon, Eunjung, Chari, Murugulla A., Mukkanti, Kagga, Kim, Sung-Hoon, Ahn, Kwang-Hyun, Kim, Sun Yeou

“…1,5-Benzodiazepine derivatives such as compound 3e showed a good anti-neuroinflammatory effects by suppressing iNOS enzyme activity in microglia cells. A…”
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Simple and Efficient Process for the Large-Scale Preparation of Agomelatine: An Antidepressant Drug by Vujjini, Satish Kumar, Vyala, Sunitha, Badarla, Krishna Rao, Kandala, Sreenatha Charyulu, Bandichhor, Rakeshwar, Kagga, Mukkanti, Cherukupalli, Praveen

“…A simple and efficient process for the large-scale preparation of agomelatine (1), an antidepressant drug is, described. Agomelatine was prepared in a linear…”
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Synthesis of Zolmitriptan and Related Substances by Vujjini, Satish Kumar, Mothukuri, Vivekananda Reddy, Islam, Aminul, Bandichhor, Rakeshwar, Kagga, Mukkanti, Malakondaiah, Golla China

“…Efficient and cost-effective synthesis of Zolmitriptan 1 employing Japp-Klingemann reaction and a new robust purification strategy is described…”
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Total synthesis of agomelatine via Friedel–Crafts acylation followed by Willgerodt–Kindler reaction by Vujjini, Satish Kumar, Datla, V.R. Krishnam Raju, Badarla, Krishna Rao, Vetukuri, V.N.K.V. Prasada Raju, Bandichhor, Rakeshwar, Kagga, Mukkanti, Cherukupally, Praveen

“…Total synthesis of antidepressant drug, agomelatine is reported. Regio selective Friedel–Crafts acylation followed by Willgerodt–Kindler reactions is used as…”
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An Efficient Synthesis of 1‑(2-Methoxyphenoxy)-2,3-epoxypropane: Key Intermediate of β‑Adrenoblockers by Madivada, Lokeswara Rao, Anumala, Raghupathi Reddy, Gilla, Goverdhan, Kagga, Mukkanti, Bandichhor, Rakeshwar

“…An efficient process for the preparation of 1-(2-methoxyphenoxy)-2,3-epoxypropane, a key intermediate for the synthesis of ranolazine is described…”
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An Improved and Scalable Process for the Synthesis of 5‑Azacytidine: An Antineoplastic Drug by Vujjini, Satish Kumar, Varanasi, Ganesh, Arevelli, Srinivas, Kandala, Sreenatha Charyulu, Tirumalaraju, Satyanarayana Raju, Bandichhor, Rakeshwar, Kagga, Mukkanti, Cherukupally, Praveen

“…An improved, practical, and scalable process for the manufacture of antineoplastic drug, 5-azacytidine (1), is described. A thorough understanding of the…”
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Synthesis and Characterization of Related Substances of Deferasirox, an Iron (Fe3+) Chelating Agent by Rao, Vascuri Janardhana, Mukkanti, Kagga, Vekariya, N. A., Gupta, P. Badrinadh, Islam, Aminul

“…Deferasirox is an orally active iron chelating agent, and during process development for deferasirox, we observed six related substances (impurities), namely…”
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An efficient synthesis of dexlansoprazole employing asymmetric oxidation strategy by Raju, Manne Naga, Kumar, Neelam Uday, Reddy, Baddam Sudhakar, Anitha, Naredla, Srinivas, Gangula, Bhattacharya, Apurba, Mukkanti, Kagga, Kolla, Naveenkumar, Bandichhor, Rakeshwar

“…An alternative and scalable synthesis of dexlansoprazole (( R)-(+)- 1); the ( R)-enantiomer of Lansoprazole with an enantiomeric excess of >99.8% is presented…”
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Practical One-Pot and Large-Scale Synthesis of N-(tert-Butyloxycarbonyl)-3-pyrroline by Rajesh, Tammana, Azeez, Shaik Abdul, Naresh, Erragunta, Madhusudhan, Gutta, Mukkanti, Kagga

“…N-(tert-Butyloxycarbonyl)-3-pyrroline was prepared with high purity in large scale starting from cis-1,4-dichloro-2-butene via delepine reaction and subsequent…”
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New and Improved Manufacturing Process for Valsartan by .N, Senthil Kumar, Reddy, Shankar B, Sinha, Brajesh Kumar, Mukkanti, Kagga, Dandala, Ramesh

“…A new and improved industrially viable manufacturing process for valsartan, an antihypertension drug, is described…”
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Synthesis of (±)-trans-hexahydropyrrolo[3,4-d]oxazol-2-one and its derivatives by using N-(tert-butyloxycarbonyl)-3-pyrroline as precursor by Rajesh, Tammana, Rao, Sambangi Polinaini Narayana, Suresh, Kopparthi, Madhusudhan, Gutta, Mukkanti, Kagga

“…Synthetic method for the preparation of (±)‐trans‐hexahydropyrrolo[3,4‐d]oxazol‐2‐one and its derivatives has been developed. By one route, an efficient…”
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Alternative Synthesis of Tadalafil: PDE5 Inhibitor by Anumula, Raghupathi Reddy, Madivada, Lokeswara Rao, Gilla, Goverdhan, Raju, V. V. N. K. Prasad, Kagga, Mukkanti, Reddy, Padi Pratap, Bhattacharya, Apurba, Bandichhor, Rakeshwar

“…Two-step alternative synthesis of tadalafil (1) is described. The synthesis features Pictet-Spengeler type reaction and DCC…”
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Preparation of Optically Pure Esomeprazole and Its Related Salt by Raju, Satya V. N, Purandhar, Koilkonda, Reddy, Padi Pratap, Reddy, Ghanta Mahesh, Reddy, Lekkala Amarnath, Reddy, Kikkuri Srirami, Sreenath, Keshaboina, Mukkanti, Kagga, Reddy, Ganji Santhi

“…The magnesium salt of (S)-isomer of omeprazole, with a trade name of Nexium, is the first proton-pump inhibitor developed as a single isomer for the treatment…”
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A novel validated RP-HPLC method development for the estimation of rimonabant hydrochloride in bulk and tablet dosage forms by Nama, Sreekanth

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