Search Results - "Moyá, Diego A."
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1
Convergent Total Synthesis of Yaku'amide A
Published in Angewandte Chemie International Edition (01-03-2021)“…Total synthesis of the anticancer peptide natural product yaku'amide A is reported. Its β‐tert‐hydroxy amino acids were prepared by regioselective…”
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Journal Article -
2
Towards a streamlined synthesis of peptides containing α,β-dehydroamino acids
Published in Tetrahedron letters (22-06-2021)“…[Display omitted] •Dehydroamino acids can be inserted in peptides via a coupling/elimination sequence.•Dehydration of a Thr-containing peptide can be…”
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Journal Article -
3
Synthesis and evaluation of potent yaku'amide A analogs
Published in Chemical science (Cambridge) (16-02-2022)“…Two full-length analogs of the anticancer peptide yaku'amide A (1a) and four partial structures have been synthesized. These analogs were identified by…”
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Journal Article -
4
Convergent Total Synthesis of Yaku'amide A
Published in Angewandte Chemie (01-03-2021)“…Total synthesis of the anticancer peptide natural product yaku'amide A is reported. Its β‐tert‐hydroxy amino acids were prepared by regioselective…”
Get full text
Journal Article -
5
Synthesis and Applications of α,β-Dehydroamino Acid-Containing Peptides
Published 01-01-2022“…Yaku’amide A (YA) is a linear anticancer peptide that is rich in bulky dehydroamino acids (ΔAAs) and β-hydroxyamino acids (β-OHAAs). In our recent total…”
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Dissertation