Search Results - "Montoir, David"

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  1. 1

    Differential Functionalization of 1,6-Naphthyridin-2(1H)-ones through Sequential One-Pot Suzuki-Miyaura Cross-Couplings by Montoir, David, Tonnerre, Alain, Duflos, Muriel, Bazin, Marc-Antoine

    Published in European journal of organic chemistry (01-03-2014)
    “…A practical synthesis of 7‐chloro‐3‐iodo‐1‐methyl‐1,6‐naphthyridin‐2(1H)‐one is described that starts from 2‐chloro‐4‐(methylamino)nicotinaldehyde. The dihalo…”
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  2. 2

    Crystal Structure of N-(7-{[2-(Dimethylamino)ethyl]amino}-1-methyl-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl)-3,4,5-trimethoxybenzamide by GUILLON, Jean, MONTOIR, David, MARCHIVIE, Mathieu, DUFLOS, Muriel, BAZIN, Marc-Antoine

    Published in X-ray Structure Analysis Online (2017)
    “…The X-ray crystal structure of N-(7-{[2-(dimethylamino)ethyl]amino}-1-methyl-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl)-3,4,5-trimethoxybenzamide, a potential…”
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  3. 3

    Synthesis of (1 → 2)-S-Linked Saccharides and S‑Linked Glycoconjugates via a Palladium-G3-XantPhos Precatalyst Catalysis by AL-Shuaeeb, Riyadh Ahmed Atto, Montoir, David, Alami, Mouad, Messaoudi, Samir

    Published in Journal of organic chemistry (07-07-2017)
    “…Buchwald–Hartwig–Migita cross-coupling of 1-thiosugars with 2-iodoglycals has been accomplished under mild and operationally simple reaction conditions through…”
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  4. 4

    New azole antifungals with a fused triazinone scaffold by Montoir, David, Guillon, Rémi, Gazzola, Sophie, Ourliac-Garnier, Isabelle, Soklou, Kossi Efouako, Tonnerre, Alain, Picot, Carine, Planchat, Aurélien, Pagniez, Fabrice, Le Pape, Patrice, Logé, Cédric

    Published in European journal of medicinal chemistry (01-03-2020)
    “…We identified a new series of azole antifungal agents bearing a pyrrolotriazinone scaffold. These compounds exhibited a broad in vitro antifungal activity…”
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  5. 5

    Synthesis of aryl-thioglycopeptides through chemoselective Pd-mediated conjugation by Montoir, David, Amoura, Mehdi, Ababsa, Zine El Abidine, Vishwanatha, T M, Yen-Pon, Expédite, Robert, Vincent, Beltramo, Massimiliano, Piller, Véronique, Alami, Mouad, Aucagne, Vincent, Messaoudi, Samir

    Published in Chemical science (Cambridge) (14-12-2018)
    “…We describe herein a Pd-catalyzed methodology for the thioglycoconjugation of iodoaryl peptides and aminoacids. This operationally simple process occurs under…”
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    Structure–Activity Relationship Studies of Retro‑1 Analogues against Shiga Toxin by Abdelkafi, Hajer, Michau, Aurélien, Pons, Valérie, Ngadjeua, Flora, Clerget, Alexandra, Ait Ouarab, Lilia, Buisson, David-Alexandre, Montoir, David, Caramelle, Lucie, Gillet, Daniel, Barbier, Julien, Cintrat, Jean-Christophe

    Published in Journal of medicinal chemistry (13-08-2020)
    “…High-throughput screening has shown that Retro-1 inhibits ricin and Shiga toxins by diminishing their intracellular trafficking via the retrograde route, from…”
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  8. 8

    Efficient one-pot synthesis of 3,7-disubstituted 1,6-naphthyridin-2(1H)-ones through regioselective palladium-catalyzed cross-coupling and SNAr reactions by Montoir, David, Tonnerre, Alain, Duflos, Muriel, Bazin, Marc-Antoine

    Published in Tetrahedron (27-05-2015)
    “…An efficient synthesis of original 3,7-disubstituted 1,6-naphthyridones via one-pot palladium-catalyzed cross-coupling and SNAr reactions is reported…”
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  11. 11

    Novel 1,6-naphthyridin-2(1H)-ones as potential anticancer agents targeting Hsp90 by Montoir, David, Barillé-Nion, Sophie, Tonnerre, Alain, Juin, Philippe, Duflos, Muriel, Bazin, Marc-Antoine

    Published in European journal of medicinal chemistry (25-08-2016)
    “…Hsp90 is an ATP-dependent chaperone known to be overexpressed in many cancers. This way, Hsp90 is an important target for drug discovery. Novobiocin, an…”
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