Search Results - "Montéro, Jean Louis"

Water-Dispersible Sugar-Coated Iron Oxide Nanoparticles. An Evaluation of their Relaxometric and Magnetic Hyperthermia Properties by Lartigue, Lenaic, Innocenti, Claudia, Kalaivani, Thangavel, Awwad, Azzam, Sanchez Duque, Maria del Mar, Guari, Yannick, Larionova, Joulia, Guérin, Christian, Montero, Jean-Louis Georges, Barragan-Montero, Véronique, Arosio, Paolo, Lascialfari, Alessandro, Gatteschi, Dante, Sangregorio, Claudio

“…Synthesis of functionalized magnetic nanoparticles (NPs) for biomedical applications represents a current challenge. In this paper we present the synthesis and…”
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Carbonic anhydrase IX: A new druggable target for the design of antitumor agents by Winum, Jean-Yves, Rami, Marouan, Scozzafava, Andrea, Montero, Jean-Louis, Supuran, Claudiu

“…Carbonic anhydrases (CAs, EC 4.2.1.1) are a family of enzymes widespread in all life kingdoms. In mammals, isozyme CA IX is highly overexpressed in many cancer…”
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Therapeutic potential of sulfamides as enzyme inhibitors by Winum, Jean-Yves, Scozzafava, Andrea, Montero, Jean-Louis, Supuran, Claudiu T.

“…Sulfamide, a quite simple molecule incorporating the sulfonamide functionality, widely used by medicinal chemists for the design of a host of biologically…”
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Sulfamates and their therapeutic potential by Winum, Jean-Yves, Scozzafava, Andrea, Montero, Jean-Louis, Supuran, Claudiu T.

“…Starting from the very simple molecule sulfamic acid, O‐substituted‐, N‐substituted‐, or di‐/tri‐substituted sulfamates may be obtained, which show specific…”
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Design of zinc binding functions for carbonic anhydrase inhibitors by Winum, Jean-Yves, Scozzafava, Andrea, Montero, Jean-Louis, Supuran, Claudiu T

“…Zinc ion plays a crucial role in the protein's functions and is linked to a variety of physiological processes. It constitutes an essential component of…”
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Antiangiogenic activity of neutral lipids, glycolipids, and phospholipids fractions of Pinus halepensis Mill. seeds by Kadri, Nabil, Khettal, Bachra, Adjebli, Ahmed, Cresteil, Thierry, Yahiaoui-Zaidi, Rachida, Barragan-Montero, Veronique, Montero, Jean-Louis

“…•Lipid fractions (neutral lipids, glycolipids and phospholipids) of Pinus halepensis Mill. seeds were complexed by β-Cyclodextrin.•No cytotoxicity effect was…”
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Analysis of polar lipid fraction of Pinus halepensis Mill. seeds from North Algeria by Kadri, Nabil, Khettal, Bachra, Yahiaoui-zaidi, Rachida, Barragan-Montero, Veronique, Montero, Jean-Louis

“…•Herein, the lipid fraction of Pinus halepensis Mill. seeds has been characterized.•The lipids fractions were separated by LC and the lipids sub fractions were…”
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A Very Efficient Synthesis of a Mannosyl Orthoester [2]Rotaxane and Mannosidic [2]Rotaxanes by Coutrot, Frédéric, Busseron, Eric, Montero, Jean-Louis

“…The direct preparation of mannosyl[2]rotaxane derivatives by O-glycosylation from tetra-O-acetyl-α-d-mannosyltrichloroacetimidate and a tert-butylanilinium…”
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Inhibition of carbonic anhydrase IX: a new strategy against cancer by Winum, Jean-Yves, Scozzafava, Andrea, Montero, Jean-Louis, Supuran, Claudiu T

“…Of the thirteen active carbonic anhydrase (CA) isozymes, the transmembrane isoform CA IX has been shown to be linked with carcinogenesis. CA IX presents an…”
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New zinc binding motifs in the design of selective carbonic anhydrase inhibitors by Winum, Jean-Yves, Scozzafava, Andrea, Montero, Jean-Louis, Supuran, Claudiu T

“…The carbonic anhydrases (CAs, EC 4.2.1.1) are ubiquitous zinc enzymes which catalyze a very simple physiological reaction, the interconversion between carbon…”
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BiX3 as an efficient and selective reagent for the halogen exchange reaction by Boyer, Bernard, Keramane, El Mehdi, Arpin, Sèverine, Montéro, Jean-Louis, Roque, Jean-Pierre

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Carbonic anhydrase inhibitors: Copper(II) complexes of polyamino-polycarboxylamido aromatic/heterocyclic sulfonamides are very potent inhibitors of the tumor-associated isoforms IX and XII by Rami, Marouan, Winum, Jean-Yves, Innocenti, Alessio, Montero, Jean-Louis, Scozzafava, Andrea, Supuran, Claudiu T.

“…Reaction of EDTA/DTPA dianhydride with aromatic/heterocyclic sulfonamides afforded a series of derivatives incorporating polyaminopolycarboxylate tails and…”
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Regio- and stereospecificity in radical cascade cyclizations of TMS-alcyne containing allyl bromomethyldimethylsilyl ethers by Belval, Florence, Chavis, Claude, Fruchier, Alain, Montéro, Jean-Louis, Lucas, Marc

“…Tandem radical cyclization of (E) and (Z) TMS-homopropargyl allyl bromomethyl-dimethylsilyl ethers is reported to provide an all- cis substituted…”
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Synthesis of Mannose-6-Phosphate Analogues and their Utility as Angiogenesis Regulators by Barragan-Montero, Véronique, Awwad, Azzam, Combemale, Stéphanie, de Santa Barbara, Pascal, Jover, Bernard, Molès, Jean-Pierre, Montero, Jean-Louis

“…Sweet utility: An efficient approach, using a key cyclic sulfate intermediate is reported for the synthesis of mannose‐6‐phosphate (M6P) analogues modified at…”
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Carbonic Anhydrase Inhibitors: Design of Membrane-Impermeant Copper(II) Complexes of DTPA-, DOTA-, and TETA-Tailed Sulfonamides Targeting the Tumor-Associated Transmembrane Isoform IX by Rami, Marouan, Cecchi, Alessandro, Montero, Jean-Louis, Innocenti, Alessio, Vullo, Daniela, Scozzafava, Andrea, Winum, Jean-Yves, Supuran, Claudiu T.

“…The synthesis and carbonic anhydrase (CA, EC 4.2.1.1) inhibitory activity of two series of aromatic sulfonamides and their CuII derivatives, incorporating…”
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Targeting of the Brucella suis Virulence Factor Histidinol Dehydrogenase by Histidinol Analogues Results in Inhibition of Intramacrophagic Multiplication of the Pathogen by JOSEPH, Pascale, ABDO, Marie-Rose, BOIGEGRAIN, Rose-Anne, MONTERO, Jean-Louis, WINUM, Jean-Yves, KÖHLER, Stephan

“…Classifications Services AAC Citing Articles Google Scholar PubMed Related Content Social Bookmarking CiteULike Delicious Digg Facebook Google+ Mendeley Reddit…”
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Carbonic Anhydrase Inhibitors: Glycosylsulfanilamides Act as Subnanomolar Inhibitors of the Human Secreted Isoform VI by Winum, Jean-Yves, Montero, Jean-Louis, Vullo, Daniela, Supuran, Claudiu T

“…A series of sulfonamides incorporating sugar moieties and the sulfanilamide scaffold have been investigated for their interaction with the secretory isoform of…”
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Metal binding functions in the design of carbonic anhydrase inhibitors by Winum, Jean-Yves, Scozzafava, Andrea, Montero, Jean-Louis, Supuran, Claudiu T

“…The carbonic anhydrases (CAs, EC 4.2.1.1) are zinc containing metalloenzymes which catalyse efficiently the reversible hydration of carbon dioxide to…”
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Carbonic Anhydrase Activators: Gold Nanoparticles Coated with Derivatized Histamine, Histidine, and Carnosine Show Enhanced Activatory Effects on Several Mammalian Isoforms by Saada, Mohamed-Chiheb, Montero, Jean-Louis, Vullo, Daniela, Scozzafava, Andrea, Winum, Jean-Yves, Supuran, Claudiu T

“…Lipoic acid moieties were attached to amine or amino acids showing activating properties against the zinc enzyme carbonic anhydrase (CA, EC 4.2.1.1). The…”
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A new β-carbonic anhydrase from Brucella suis, its cloning, characterization, and inhibition with sulfonamides and sulfamates, leading to impaired pathogen growth by Joseph, Pascale, Ouahrani-Bettache, Safia, Montero, Jean-Louis, Nishimori, Isao, Minakuchi, Tomoko, Vullo, Daniela, Scozzafava, Andrea, Winum, Jean-Yves, Köhler, Stephan, Supuran, Claudiu T.

“…A β-carbonic anhydrase (CA, EC 4.2.1.1) from the bacterial pathogen Brucella suis, bsCA II, has been cloned, purified, and characterized kinetically. bsCA II…”
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