Search Results - "Mondal, Susanta Kumar"

Tuning Caco-2 Permeability by Cocrystallization: Insights from Molecular Dynamics Simulation by Pandey, Noopur, Kumari, Nimmy, Roy, Parag, Kumar Mondal, Susanta, Thakur, Abhishek, Calvin Sun, Changquan, Ghosh, Animesh

“…Emerging evidence suggests that intestinal permeability can be potentially enhanced through cocrystallization. However, a mechanism for this effect remains to…”
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Development of direct compression Acetazolamide tablet with improved bioavailability in healthy human volunteers enabled by cocrystallization with p-Aminobenzoic acid by Kumari, Nimmy, Roy, Parag, Roy, Sukanta, Wang, Chenguang, Das, Sourav, Pandey, Noopur, Mondal, Susanta Kumar, Bose, Anirbandeep, Sun, Changquan Calvin, Ghosh, Animesh

“…[Display omitted] Pharmaceutical cocrystallization has been widely used to improve physicochemical properties of APIs. However, developing cocrystal…”
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Non-carboxylic acid inhibitors of aldose reductase based on N-substituted thiazolidinedione derivatives by Mohd Siddique, Mohd Usman, Thakur, Abhishek, Shilkar, Deepak, Yasmin, Sabina, Halakova, Dominika, Kovacikova, Lucia, Prnova, Marta Soltesova, Stefek, Milan, Acevedo, Orlando, Dasararaju, Gayathri, Devadasan, Velmurugan, Mondal, Susanta Kumar, Jayaprakash, Venkatesan

“…In search of dually active PPAR-modulators/aldose reductase (ALR2) inhibitors, 16 benzylidene thiazolidinedione derivatives, previously reported as partial…”
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Synthesis, anti-cancer activity and molecular docking studies of new nicotinamide containing EP4 antagonists by Ali, Md. Akram, Chakraborty, Rajib, Mondal, Susanta Kumar, Bhunia, Supriya, Chakraborty, Sabyasachi, Samanta, Subhas, Rudra, Sonali

“…•20 new EP4 antagonists compounds designed and synthesized based on the literature nicotinamide derivative AAT-008.•Evaluations of the in vitro EP4…”
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Antidiabetic activity of Diospyros malabarica Kostel bark: a preliminary investigation for possible mode of action by Mondal, Susanta Kumar, Chakraborty, Goutam, Bhaumik, Uttam Kumar, Gupta, Malaya, Mazumder, Upal Kanti

“…The defatted methanol extract of bark of Diospyros malabarica (DM) at doses of 200 and 400 mg/kg, p.o. showed significant hypoglycemic activity on normal rats…”
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Free radical scavenging property of Annona reticulata leaves by Mondal, Susanta Kumar, Saha, Prerona, Mondal, NB, Mazumder, UK

“…Annona reticulata belonging to the family Annonaceae is traditionally used as anthelmintic and it is reported to have anticancer activity. Free radicals are…”
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Chemistry of withaferin-A: chemo, regio, and stereoselective synthesis of novel spiro-pyrrolizidino-oxindole adducts of withaferin-A via one-pot three-component [3+2] azomethine ylide cycloaddition and their cytotoxicity evaluation by Bharitkar, Yogesh P., Kanhar, Satish, Suneel, Neradibilli, Mondal, Susanta Kumar, Hazra, Abhijit, Mondal, Nirup B.

“…Withaferin-A (WA) has attracted the attention of chemists as well as biologists due to its interesting structure and various bio-activities. In light of the…”
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Regio- and Stereoselective Synthesis of a Library of Bioactive Dispiro-Oxindolo/Acenaphthoquino Andrographolides via 1,3-Dipolar Cycloaddition Reaction Under Microwave Irradiation by Hazra, Abhijit, Bharitkar, Yogesh P, Chakraborty, Debanjana, Mondal, Susanta Kumar, Singal, Nupur, Mondal, Shyamal, Maity, Arindam, Paira, Rupankar, Banerjee, Sukdeb, Mondal, Nirup B

“…Dispiro-pyrrolidino/pyrrolizidino fused oxindoles/acenaphthoquinones have been derived from andrographolide via azomethine ylide cycloaddition to the…”
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Monoamine Oxidase Inhibitory Activity of Novel Pyrazoline Analogues: Curcumin Based Design and Synthesis‐II by Badavath, Vishnu Nayak, Ucar, Gulberk, Sinha, Barij Nayan, Mondal, Susanta Kumar, Jayaprakash, Venkatesan

“…In continuation with our earlier work on MAO inhibitory curcumin based pyrazoline analogues, we synthesized a series of pyrazoline derivatives (from…”
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Novel Pyrimidinone Derivatives Show Anticancer Activity and Induce Apoptosis: Synthesis, SAR and Putative Binding Mode by Roy, Ashis, Kundu, Mrinalkanti, Dhar, Pranab, Chakraborty, Arnish, Mukherjee, Soumen, Naskar, Jayatri, Rarhi, Chhanda, Barik, Rajib, Mondal, Susanta Kumar, Wani, Mushtaq Ahmad, Gajbhiye, Rahul, Roy, Kuldeep K., Maiti, Arup, Manna, Priyadarshi, Adhikari, Susanta

“…A series of novel bicyclic, substituted pyrimidinone compounds were designed, synthesized and characterized. In vitro anti‐proliferative activity of the…”
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In vitro antioxidant activity of Diospyros malabarica Kostel bark by Mondal, Susanta Kumar, Chakraborty, Goutam, Gupta, M, Mazumder, U K

“…Antioxidant activity of defatted methanol extract of D. malabarica bark was studied for its free radical scavenging property on different in vitro models e.g…”
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Determination of drug-like properties of a novel antileishmanial compound: In vitro absorption, distribution, metabolism, and excretion studies by Mondal, Susanta Kumar, Mondal, Nirup B, Banerjee, Sukdeb, Mazumder, Upal Kanti

“…In drug discovery research, the compounds should not only to be potent and selective but also must possess acceptable pharmacokinetic properties such as…”
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In vitro cytotoxic and human recombinant caspase inhibitory effect of Annona reticulata leaves by Mondal, Susanta Kumar, Mondal, Nirup Bikash, Mazumder, Upal Kanti

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Antidiabetic activity of Diospyros malabarica Kostel bark: a preliminary investigation for possible mode of action by Mondal, Susanta Kumar, Chakraborty, Goutam, Bhaumik, Uttam Kumar, Gupta, Malaya, Mazumder, Upal Kanti

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Free radical scavenging property of Annona reticulata leaves by Mondal, Susanta Kumar, Saha, Prerona, Mondal, NB, Mazumder, UK

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