Search Results - "Mochul’skaya, N. N."

MnO2-Mediated Oxidative Cyclization of “Formal” Schiff’s Bases: Easy Access to Diverse Naphthofuro-Annulated Triazines by Fatykhov, Ramil F., Khalymbadzha, Igor A., Sharapov, Ainur D., Potapova, Anastasia P., Mochulskaya, Nataliya N., Tsmokalyuk, Anton N., Ivoilova, Alexandra V., Mozharovskaia, Polina N., Santra, Sougata, Chupakhin, Oleg N.

“…A different type of MnO2-induced oxidative cyclization of dihydrotriazines has been developed. These dihydrotriazines are considered as a “formal” Schiff’s…”
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Schiff Bases Derived from 6-Formyl-3-(4-methoxyphenyl)picolinonitrile: Rational Synthetic Approach and Photophysical Properties by Kudryashova, E. A., Valieva, M. I., Shtaitz, Ya. K., Mochulskaya, N. N., Krinochkin, A. P., Kopchuk, D. S., Zyryanov, G. V., Rusinov, V. L.

“…A convenient synthetic approach to Schiff bases based on 3-(4-methoxyphenyl)-6-formylpicolinonitrile as surrogates of 2,2′-bipyridine ligands is proposed. The…”
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Bioinspired Pyrano[2,3- f ]chromen-8-ones: Ring C-Opened Analogues of Calanolide A: Synthesis and Anti-HIV-1 Evaluation by Khalymbadzha, Igor A, Fatykhov, Ramil F, Butorin, Ilya I, Sharapov, Ainur D, Potapova, Anastasia P, Muthipeedika, Nibin Joy, Zyryanov, Grigory V, Melekhin, Vsevolod V, Tokhtueva, Maria D, Deev, Sergey L, Kukhanova, Marina K, Mochulskaya, Nataliya N, Tsurkan, Mikhail V

“…We have designed and synthesized a series of bioinspired pyrano[2,3- ]coumarin-based Calanolide A analogs with anti-HIV activity. The design of these new…”
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Bioactive Pyrrolo[2,1-f][1,2,4]triazines: Synthesis, Molecular Docking, In Vitro Cytotoxicity Assay and Antiviral Studies by Mochulskaya, Nataliya N., Kotovskaya, Svetlana K., Butorin, Ilya I., Varaksin, Mikhail V., Charushin, Valery N., Rusinov, Vladimir L., Esaulkova, Yana L., Slita, Alexander V., Ilyina, Polina A., Zarubaev, Vladimir V.

“…A series of 2,4-disubstituted pyrrolo[2,1-f][1,2,4]triazines containing both aryl and thienyl substituents were synthesized by exploiting the 1,3-cycloaddition…”
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2-Thiomorpholino-5-Aryl-6H-1,3,4-Thiadiazine Hydrobromides and Their Ability to Inhibit Nonenzymatic Protein Glycosylation by Sidorova, L. P., Tseitler, T. A., Emel’yanov, V. V., Savateeva, E. A., Maksimova, N. E., Mochul’skaya, N. N., Chereshnev, V. A., Chupakhin, O. N.

“…Cyclocondensation of α-halogenacetophenones with an original 4-morpholine thiosemicarbazide was used to synthesize a group of new Captions: of the…”
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Nitroalkyl-substituted tetrahydropyrazines in syntheses of azapolycyclic compounds by Slepukhin, P. A., Mochul’skaya, N. N., Sidorova, L. P., Rusinov, G. L., Ezhikova, M. A., Kodess, M. I., Kazheva, O. N., Chekhlov, A. N., D’yachenko, O. A., Charushin, V. N.

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Synthesis of New 1,3,4-Thiadiazines Capable of Inhibiting Nonenzymatic Glycosylation of Proteins by Sidorova, L. P., Tseitler, T. A., Perova, N. M., Emel’yanov, V. V., Savateeva, E. A., Maksimova, N. E., Mochul’skaya, N. N., Chereshnev, V. A., Chupakhin, O. N.

“…A series of new 1,3,4-thiadiazines with cycloalkylamino (cyclopropylamino, cyclobutylamino, cyclopentylamino, cyclohexylamino) groups were synthesized via…”
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2-Morpholino-5-Phenyl-6H-1,3,4-Thiadiazine Corrects Metabolic Disorders during the Development of Alloxan Diabetes Mellitus in Rats by Emelianov, V. V., Savateeva, E. A., Sidorova, L. P., Tseitler, T. A., Gette, I. F., Bulavintseva, T. S., Smirnykh, S. E., Maksimova, N. E., Mochulskaya, N. N., Chupakhin, O. N., Chereshnev, V. A.

“…Metabolic disorders were evaluated in rats with alloxan diabetes mellitus after administration of 2-morpholino-5-phenyl- 6H -1,3,4-thiadiazine (compound L-17)…”
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Synthetic approaches to 2-aryl/hetaryl- and 2-(hetaryl)ylidene derivatives of fluorinated 1,3-benzothiazin-4-ones by Nosova, Emiliya V., Batanova, Olga A., Mochulskaya, Nataliya N., Lipunova, Galina N.

“…A series of 2-hetaryl- and 2-(hetaryl)ylidene substituted 5-fluoro-8-nitro-1,3-benzothiazin-4-ones was synthesized by interaction of…”
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Fluorine-containing quinoline and quinoxaline styryl derivatives: synthesis and photophysical properties by Nosova, E. V., Trashakhova, T. V., Ustyugov, V. S., Mochul’skaya, N. N., Valova, M. S., Lipunova, G. N., Charushin, V. N.

“…( E )-2-Styryl-substituted 6,7-difluoroquinolines and quinoxalines were synthesized by the condensation of the corresponding 2-methylbenzazines with aromatic…”
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Fluoro-containing Heterocycles: XIV. Cyclic Adducts of 6-Fluoro-7-azidoquinoxaline and Their Transformation Products by Mochul'skaya, N. N., Nagibina, E. N., Volchenkova, Yu. S., Sidorova, L. P., Charushin, V. N.

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Antiviral Agents – Benzazine Derivatives by Mochulskaya, Nataliya N., Nosova, Emiliya V., Charushin, Valery N.

“…The review outlines the results of studies of the antiviral activity of quinoline, quinoxaline, and quinazoline derivatives published over the past 5 years…”
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2,5-Di(het)arylpyridines: synthesis by ‘‘1,2,4-triazine’’ methodology and photophysical properties by Krinochkin, Alexei P., Khasanov, Albert F., Valieva, Maria I., Kudryashova, Ekaterina A., Guda, Mallikarjuna R., Kopchuk, Dmitry S., Shabunina, Olga V., Mochulskaya, Nataliya N., Slepukhin, Pavel A., Zyryanov, Grigory V., Chupakhin, Oleg N.

“…The method for the preparation of 3,6-disubstituted 1,2,4-triazines based on condensation reaction between easily available α-imino esters and…”
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Synthesis and antimycobacterial evaluation of new (2-oxo-2H-chromen-3-yl) substituted fluoroquinolones by Charushin, Valery N., Mochulskaya, Nataliya N., Antipin, Fedor V., Kotovskaya, Svetlana K., Nosova, Emiliya V., Ezhikova, Marina A., Kodess, Mikhail I., Kravchenko, Marionella A.

“…[Display omitted] •The cyanomethyl fragment was incorporated into the benzene ring of fluoroquinolones.•Cyanomethyl fluoroquinolones was converted to…”
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Aminovinyl ketones and aminovinyl esters as CCN building blocks for the synthesis of 1H-pyrrolo[3,2-e]1,2,4-triazines by Charushin, Valery N, Mochulskaya, Nataliya N, Andreiko, Anatoly A, Filyakova, Vera I, Kodess, Mikhail I, Chupakhin, Oleg N

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Fluorinated 1,3-benzothiazin-4-ones containing fluoroquinolone fragment by Nosova, Emiliya V., Batanova, Olga A., Mochulskaya, Nataliya N., Charushin, Valery N.

“…We have developed an efficient synthetic approach to potential antibacterial agents with double mechanism of action through the combination of antibacterial…”
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Fluorinated quinolones possessing antituberculous activity by Lipunova, G. N., Nosova, É. V., Kravchenko, M. A., Mochul’skaya, N. N., Sidorova, L. P., Tsoi, E. V., Mokrushina, G. A., Chasovskikh, O. M., Charushin, V. N.

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Intermolecular and intramolecular cycloaddition reactions of 1-ethyl-1,2,4-triazinium salts with alkynes by Mochulskaya, Nataliya N., Andreiko, Anatoly A., Charushin, Valery N., Shulgin, Boris V., Raikov, Dmitry V., Solomonov, Vladimir I.

“…Azomethyne ylides generated from 3-alkylthio substituted 1-alkyl-5-aryl-1,2,4-triazinium salts 4a–c on treatment with triethylamine undergo 1,3-dipolar…”
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Use of a dual-origin temperature-controlled amplifiable replicon for optimization of human interleukin-1 beta synthesis in Escherichia coli by Mashko, S V, Mochulsky, A V, Kotenko, S V, Lebedeva, M I, Lapidus, A L, Mochulskaya, N A, Izotova, L S, Veiko, V P, Vinetsky, Y P, Ketlinsky, S A

“…A new dual-replicon recombinant plasmid, pPR53-tsr, has been constructed; it is a derivative of the expression vector pPR-TGATG-1 [Mashko et al., Gene 88…”
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MnO[sub.2]-Mediated Oxidative Cyclization of “Formal” Schiff’s Bases: Easy Access to Diverse Naphthofuro-Annulated Triazines by Fatykhov, Ramil F, Khalymbadzha, Igor A, Sharapov, Ainur D, Potapova, Anastasia P, Mochulskaya, Nataliya N, Tsmokalyuk, Anton N, Ivoilova, Alexandra V, Mozharovskaia, Polina N, Santra, Sougata, Chupakhin, Oleg N

“…A different type of MnO[sub.2]-induced oxidative cyclization of dihydrotriazines has been developed. These dihydrotriazines are considered as a "formal"…”
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