Search Results - "Miyazaki, Anna"

Icing after eccentric contraction-induced muscle damage perturbs the disappearance of necrotic muscle fibers and phenotypic dynamics of macrophages in mice by Kawashima, Masato, Kawanishi, Noriaki, Tominaga, Takaki, Suzuki, Katsuhiko, Miyazaki, Anna, Nagata, Itsuki, Miyoshi, Makoto, Miyakawa, Motoi, Sakuraya, Tohma, Sonomura, Takahiro, Arakawa, Takamitsu

“…Icing is still one of the most common treatments to acute skeletal muscle damage in sports medicine. However, previous studies using rodents reported the…”
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Synthesis and evaluation of [18F]FBNAF, a STAT3-targeting probe, for PET imaging of tumor microenvironment by Miyazaki, Anna, Kanai, Yasukazu, Wakamori, Keita, Mizuguchi, Serina, Futatsugi, Mikiya, Hirano, Fuko, Kondo, Naoya, Temma, Takashi

“…Background Signal transducer and activator of transcription 3 (STAT3) is a protein that regulates cell proliferation and differentiation, and it is attracting…”
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PET probe detecting non-small cell lung cancer susceptible to epidermal growth factor receptor tyrosine kinase inhibitor therapy by Makino, Akira, Miyazaki, Anna, Tomoike, Ayaka, Kimura, Hiroyuki, Arimitsu, Kenji, Hirata, Masahiko, Ohmomo, Yoshiro, Nishii, Ryuichi, Okazawa, Hidehiko, Kiyono, Yasushi, Ono, Masahiro, Saji, Hideo

“…[Display omitted] Tyrosine kinase inhibitors for epidermal growth factor receptor (EGFR-TKIs) are used as molecular targeted therapy for non-small cell lung…”
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18F‑Labeled Pyrido[3,4‑d]pyrimidine as an Effective Probe for Imaging of L858R Mutant Epidermal Growth Factor Receptor by Kimura, Hiroyuki, Okuda, Haruka, Ishiguro, Masumi, Arimitsu, Kenji, Makino, Akira, Nishii, Ryuichi, Miyazaki, Anna, Yagi, Yusuke, Watanabe, Hiroyuki, Kawasaki, Ikuo, Ono, Masahiro, Saji, Hideo

“…In nonsmall-cell lung carcinoma patients, L858R mutation of epidermal growth factor receptor (EGFR) is often found, and molecular target therapy using EGFR…”
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Application of liquid chromatography–tandem mass spectrometry for the determination of opioidmimetics in the brain dialysates from rats treated with opioidmimetics intraperitoneally by Igarashi, Kazuo, Murabayashi, Yuki, Hotta, Koichiro, Kitamura, Youji, Kasuya, Fumiyo, Shiotani, Kimitaka, Tingyou, Li, Miyazaki, Anna, Tsuda, Yuko, Okada, Yoshio, Fukushima, Shoji

“…We have determined three opioidmimetics (compounds I– III) in the rat brain dialysates after intraperitoneal (i.p.) administration of compounds I– III using a…”
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Icing after skeletal muscle injury with necrosis in a small fraction of myofibers limits inducible nitric oxide synthase-expressing macrophage invasion and facilitates muscle regeneration by Nagata, Itsuki, Kawashima, Masato, Miyazaki, Anna, Miyoshi, Makoto, Sakuraya, Tohma, Sonomura, Takahiro, Oyanagi, Eri, Yano, Hiromi, Arakawa, Takamitsu

“…Growing evidence from animal experiments suggests that icing after skeletal muscle injury is harmful to muscle regeneration. However, these previous…”
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Icing after skeletal muscle injury decreases M1 macrophage accumulation and TNF-α expression during the early phase of muscle regeneration in rats by Miyazaki, Anna, Kawashima, Masato, Nagata, Itsuki, Miyoshi, Makoto, Miyakawa, Motoi, Sugiyama, Megumi, Sakuraya, Tohma, Sonomura, Takahiro, Arakawa, Takamitsu

“…Following skeletal muscle injury, both myogenic and immune cells interact closely during the regenerative process. Although icing is still a common acute…”
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Studies on the structure-activity relationship of 2', 6'-dimethyl-L-tyrosine (Dmt) derivatives: bioactivity profile of H-Dmt-NH-CH3 by FUJITA, Yoshio, TSUDA, Yuko, BRYANT, Sharon D, LAZARUS, Lawrence H, OKADA, Yoshio, MOTOYAMA, Takashi, LI, Tingyou, MIYAZAKI, Anna, YOKOI, Toshio, SASAKI, Yusuke, AMBO, Akihiro, NIIZUMA, Hideko, JINSMAA, Yunden

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A solvent-dependent chirality-switchable thia-Michael addition to α,β-unsaturated carboxylic acids using a chiral multifunctional thiourea catalyst by Hayama, Noboru, Kobayashi, Yusuke, Sekimoto, Eriko, Miyazaki, Anna, Inamoto, Kiyofumi, Kimachi, Tetsutaro, Takemoto, Yoshiji

“…An asymmetric thia-Michael addition of arylthiols to α,β-unsaturated carboxylic acids using a thiourea catalyst that bears arylboronic acid and tertiary amine…”
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Studies on the Mechanism of 1,2-Dihydropyrazin-2-one Ring Formation from Dipeptidyl Chloromethyl Ketone and Its Chemical Properties: Immediate Deamination during Catalytic Hydrogenation by Miyazaki, Anna, Fujisawa, Yutaka, Shiotani, Kimitaka, Fujita, Yoshio, Li, Tingyou, Tsuda, Yuko, Yokoi, Toshio, Bryant, Sharon D., Lazarus, Lawrence H., Okada, Yoshio

“…1,2-Dihydropyrazin-2-one derivatives, which have two aminoalkyl groups at the positions 3 and 6, were found to be efficient tools for the construction of…”
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A solvent-dependent chirality-switchable thia-Michael addition to α,β-unsaturated carboxylic acids using a chiral multifunctional thiourea catalyst† †Electronic supplementary information (ESI) available: Experimental procedures, spectroscopic data, copies of 1H and 13C NMR spectra, and HPLC chromatograms. See DOI: 10.1039/d0sc01729a by Hayama, Noboru, Kobayashi, Yusuke, Sekimoto, Eriko, Miyazaki, Anna, Inamoto, Kiyofumi, Kimachi, Tetsutaro, Takemoto, Yoshiji

“…An asymmetric thia-Michael addition of arylthiols to α,β-unsaturated carboxylic acids using a thiourea catalyst that bears arylboronic acid and tertiary amine…”
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Synthesis of opioidmimetics, 3-[H-Dmt-NH(CH(2))(m)]-6-[H-Dmt-NH(CH(2))(n)]-2(1H)-pyrazinones, and studies on structure-activity relationships by Shiotani, Kimitaka, Miyazaki, Anna, Li, Tingyou, Tsuda, Yuko, Yokoi, Toshio, Ambo, Akihiro, Sasaki, Yusuke, Bryant, Sharon D, Jinsmaa, Yunden, Lazarus, Lawrence H, Okada, Yoshio

“…Opioidmimetics containing 3-[H-Dmt-NH-(CH(2))(m)]-6-[H-Dmt-NH-(CH(2))(n)]-2(1H)-pyrazinone symmetric (m = n, 1-4) (1 - 4) and asymmetric (m, n = 1 - 4)…”
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Inhibitory effect of novel somatostatin peptide analogues on human cancer cell growth based on the selective inhibition of DNA polymerase β by Kuriyama, Isoko, Miyazaki, Anna, Tsuda, Yuko, Yoshida, Hiromi, Mizushina, Yoshiyuki

“…The present study was designed to investigate the anticancer activity of novel nine small peptides (compounds 1–9) derived from TT-232, a somatostatin…”
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Immediate deamination from the aminomethyl group attached to 1,2-dihydropyrazin-2-one derivative during catalytic hydrogenation by Okada, Yoshio, Fujisawa, Yutaka, Morishita, Akihisa, Shiotani, Kimitaka, Miyazaki, Anna, Fujita, Yoshio, Li, Tingyou, Tsuda, Yuko, Yokoi, Toshio, Bryant, Sharon D., Lazarus, Lawrence H.

“…The catalytic hydrogenation of 3,6-bis(benzyloxycarbonylaminomethyl)-5-methyl-1,2-dihydropyrazin-2-one to remove benzyloxycarbonyl (Z) groups resulted in a…”
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Inhibitory effect of novel somatostatin peptide analogues on human cancer cell growth based on the selective inhibition of DNA polymerase I2 by Kuriyama, Isoko, Miyazaki, Anna, Tsuda, Yuko, Yoshida, Hiromi, Mizushina, Yoshiyuki

“…The present study was designed to investigate the anticancer activity of novel nine small peptides (compounds 1a9) derived from TT-232, a somatostatin…”
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Synthesis and preliminary characterization of radioiodinated benzofuran-3-yl-(indol-3-yl)maleimide derivatives as potential SPECT imaging probes for the detection of glycogen synthase kinase-3β (GSK-3β) in the brain by Ono, Masahiro, Kitada, Ayane, Watanabe, Hiroyuki, Miyazaki, Anna, Kimura, Hiroyuki, Saji, Hideo

“…We report on the synthesis and preliminary characterization of two radioiodinated benzofuran‐3‐yl‐(indol‐3‐yl)maleimides,…”
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Synthesis and preliminary characterization of radioiodinated benzofuran-3-yl-(indol-3-yl)maleimide derivatives as potential SPECT imaging probes for the detection of glycogen synthase kinase-3[beta] (GSK-3[beta]) in the brain by Ono, Masahiro, Kitada, Ayane, Watanabe, Hiroyuki, Miyazaki, Anna, Kimura, Hiroyuki, Saji, Hideo

“…We report on the synthesis and preliminary characterization of two radioiodinated benzofuran-3-yl-(indol-3-yl)maleimides,…”
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18 F-Labeled Pyrido[3,4- d ]pyrimidine as an Effective Probe for Imaging of L858R Mutant Epidermal Growth Factor Receptor by Kimura, Hiroyuki, Okuda, Haruka, Ishiguro, Masumi, Arimitsu, Kenji, Makino, Akira, Nishii, Ryuichi, Miyazaki, Anna, Yagi, Yusuke, Watanabe, Hiroyuki, Kawasaki, Ikuo, Ono, Masahiro, Saji, Hideo

“…In nonsmall-cell lung carcinoma patients, L858R mutation of epidermal growth factor receptor (EGFR) is often found, and molecular target therapy using EGFR…”
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Bifunctional [2‘,6‘-Dimethyl-l-tyrosine]endomorphin-2 Analogues Substituted at Position 3 with Alkylated Phenylalanine Derivatives Yield Potent Mixed μ-Agonist/δ-Antagonist and Dual μ-Agonist/δ-Agonist Opioid Ligands by Li, Tingyou, Shiotani, Kimitaka, Miyazaki, Anna, Tsuda, Yuko, Ambo, Akihiro, Sasaki, Yusuke, Jinsmaa, Yunden, Marczak, Ewa, Bryant, Sharon D, Lazarus, Lawrence H, Okada, Yoshio

“…Endomorphin-2 (H-Tyr-Pro-Phe-Phe-NH2) and [Dmt1]EM-2 (Dmt = 2‘,6‘-dimethyl-l-tyrosine) analogues, containing alkylated Phe3 derivatives, 2‘-monomethyl (2, 2‘),…”
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Inhibitory Effect of Somatostatin Peptide Analogues on DNA Polymerase Activity and Human Cancer Cell Proliferation by KURIYAMA, Isoko, MIYAZAKI, Anna, TSUDA, Yuko, YOKOI, Toshio, OKADA, Yoshio, TAKEUCHI, Toshifumi, SUGAWARA, Fumio, YOSHIDA, Hiromi, MIZUSHINA, Yoshiyuki

“…It was previously reported that ten small peptides derived from TT-232, somatostatin structural analogue (compounds 1-10), synthesised by a solution-phase…”
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