Search Results - "Min, Jong Pil"
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Discovery of DA-1229: A potent, long acting dipeptidyl peptidase-4 inhibitor for the treatment of type 2 diabetes
Published in Bioorganic & medicinal chemistry letters (15-06-2011)“…The synthesis and SAR studies of β-amino amide DPP-4 inhibitor 5f are reported. A series of β-amino amide containing substituted piperazine-2-one derivatives…”
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2
Efficient Synthesis of (±)-Juglomycin A
Published in Synthetic communications (31-12-2004)“…(±)-Juglomycin A has been synthesized in 8 steps from 1-hydroxy-5-methoxynaphthalene…”
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3
Dipeptidyl peptidase-4 inhibitor with β-amino amide scaffold: Synthesis, SAR and biological evaluation
Published in Bioorganic & medicinal chemistry letters (01-09-2012)“…The SAR studies and evaluation of β-amino amide DPP4 inhibitor 5m are reported. Inhibitors of dipeptidyl peptidase-4 (DPP4) have been shown to be effective…”
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A HIGHLY PRACTICAL ROUTE TO 2-METHYLCHROMONES FROM 2-ACETOXYBENZOIC ACIDS
Published in Synthetic communications (01-01-2001)“…2-Methylchromones were accessed via a keto ester condensation on 2-acetoxybenzoyl chloride, followed by cyclization and decarboxylation. No column…”
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5
Dipeptidyl peptidase-4 inhibitor with [beta]-amino amide scaffold: Synthesis, SAR and biological evaluation
Published in Bioorganic & medicinal chemistry letters (01-09-2012)“…Inhibitors of dipeptidyl peptidase-4 (DPP4) have been shown to be effective treatments for type 2 diabetes. Several series of [beta]-amino amide containing…”
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