Search Results - "Micetich, Ronald G"

Synthesis and antifungal activity of coumarins and angular furanocoumarins by SARDARI, S, MORI, Y, HORITA, K, MICETICH, R. G, NISHIBE, S, DANESHTALAB, M

“…Angelicin, a naturally occurring furanocoumarin, that showed antifungal activity, was considered as a lead structure for a group of synthetic coumarins…”
Get full text

In Vitro and In Vivo Activities of Syn2190, a Novel β-Lactamase Inhibitor by NISHIDA, K, KUNUGITA, C, SALAMA, S. M, ATWAL, H, MICETICH, R. G, UJI, T, HIGASHITANI, F, HYODO, A, UNEMI, N, MAITI, S. N, PHILLIPS, O. A, SPEVAK, P, ATCHISON, K. P

“…Classifications Services AAC Citing Articles Google Scholar PubMed Related Content Social Bookmarking CiteULike Delicious Digg Facebook Google+ Mendeley Reddit…”
Get full text

Interspecies Comparison of Pharmacokinetics of the Novel Triazole Antifungal Agent SYN-2869 and Its Derivatives by KHAN, J. K, MONTASERI, H, POGLOD, M, BU, H.-Z, ZHONG ZUO, SALAMA, S. M, DANESHTALAB, M, MICETICH, R. G

“…Classifications Services AAC Citing Articles Google Scholar PubMed Related Content Social Bookmarking CiteULike Delicious Digg Facebook Google+ Mendeley Reddit…”
Get full text

3-Acylamino-azetidin-2-one as a novel class of cysteine proteases inhibitors by Zhou, Nian E., Guo, Deqi, Thomas, George, Reddy, Andhe V.N., Kaleta, Jadwiga, Purisima, Enrico, Menard, Robert, Micetich, Ronald G., Singh, Rajeshwar

“…A new class of inhibitors for cysteine proteases cathepsin B, L, K and S is described. These inhibitors are based on the β-lactam ring designed to interact…”
Get full text

2-Aminoquinazoline inhibitors of cyclin-dependent kinases by Bathini, Yadagiri, Singh, Inderjit, Harvey, Patricia J., Keller, Paul R., Singh, Rajeshwar, Micetich, Ronald G., Fry, David W., Dobrusin, Ellen M., Toogood, Peter L.

“…The inhibition of cyclin-dependent kinase 4 (Cdk4) causes cell cycle arrest and restores a checkpoint that is absent in the majority of tumor cells. Compounds…”
Get full text

High-throughput Caco-2 cell permeability screening by cassette dosing and sample pooling approaches using direct injection/on-line guard cartridge extraction/tandem mass spectrometry by Bu, Hai-Zhi, Poglod, Marzena, Micetich, Ronald G., Khan, Jehangir K.

“…A method for high‐throughput Caco‐2 permeability screening of drug candidates has been developed using thirteen generic drugs as test compounds. The high…”
Get full text

SYN-1012: a new beta-lactamase inhibitor of penem skeleton by Phillips, O A, Czajkowski, D P, Spevak, P, Singh, M P, Hanehara-Kunugita, C, Hyodo, A, Micetich, R G, Maiti, S N

“…A new beta-lactamase inhibitor, SYN-1012, with a penem skeleton was synthesized and its biological activity compared with clavulanic acid, sulbactam,…”
Get more information

6-Acylamino-penam derivatives: synthesis and inhibition of cathepsins B, L, K, and S by Zhou, Nian E, Kaleta, Jadwiga, Purisima, Enrico, Menard, Robert, Micetich, Ronald G, Singh, Rajeshwar

“…The synthesis of a new series of 6-acylamino penam derivatives and their inhibition of cysteine proteases cathepsins B, L, K, and S is described. The…”
Get full text

Synthesis and biological evaluation of penam sulfones as inhibitors of β-lactamases by Phillips, Oludotun A., Reddy, Andhe V.N., Setti, Eduardo L., Spevak, Paul, Czajkowski, David P., Atwal, Herninder, Salama, Sameeh, Micetich, Ronald G., Maiti, Samarendra N.

“…Synthesis of 2β-substituted-oxyimino and -hydrazone penam sulfones and their β-lactamase inhibitory activities against class A and C β-lactamases are…”
Get full text

Design and synthesis of 6-substituted amino-4-oxa-1-azabicyclo[3,2,0]heptan-7-one derivatives as cysteine proteases inhibitors by Zhou, Nian E, Guo, Deqi, Kaleta, Jadwiga, Purisima, Enrico, Menard, Robert, Micetich, Ronald G, Singh, Rajeshwar

“…A series of 6-substituted amino-4-oxa-1-azabicyclo[3,2,0]heptan-7-one compounds was designed and synthesized as a new class of inhibitors for cysteine…”
Get full text

Phenylpropanoid glycosides from Stellera chamaejasme by Jin, Changdong, Micetich, Ronald G, Daneshtalab, Mohsen

“…Two new phenylpropanoid glycosides, [4-(3- β- d-glucopyranosyloxy-1- E-propenyl)-2,6-dimethoxyphenyl]-6- O- β- d-gluco pyranosyl- β- d-glucopyranoside and…”
Get full text

Studies on 6-halo- and 6,6-dihalopenicillins: the rearrangement of methyl 6,6-dibromopenicillanate to 1,4-thiazepine by Micetich, Ronald G, Maiti, Samarendra N, Tanaka, Motoaki, Yamazaki, Tomio, Ogawa, Kazuo

Get full text

Synthesis and .beta.-lactamase inhibitory properties of 2.beta.-[(1,2,3-triazol-1-yl)methyl]-2.alpha.-methylpenam-3.alpha.-carboxylic acid 1,1-dioxide and related triazolyl derivatives by Micetich, Ronald G, Maiti, Samarendra N, Spevak, Paul, Hall, Tse W, Yamabe, Shigeru, Ishida, Naobumi, Tanaka, Motoaki, Yamazaki, Tomio, Nakai, Akira, Ogawa, Kazuo

Get full text

Synthesis and evaluation of 3-substituted-4-oxa-1-azabicyclo[3,2,0]heptan-7-ones as cysteine proteases inhibitors: part II by Zhou, Nian E., Reddy, Andhe V. N., Kaleta, Jadwiga, Micetich, Ronald G., Singh, Rajeshwar

Get full text

1H-NMR and NOE studies of 2-cephems and 3-cephems by Im, Chaeuk, Yim, Chul Bu, Micetich, Ronald G, Daneshtalab, Mohsen

“…The¹H-NMR signals of 2-cephems and 3-cephems have been assigned and the Nuclear Overhauser Effect (NOE) study of these compounds was undertaken…”
Get full text

A rapid and reliable solid-phase extraction-LC/MS/MS assay for the determination of two novel human leukocyte elastase inhibitors, SYN-1390 and SYN-1396, in rat plasma by KHAN, J. K, BU, H.-Z, ZHONG ZUO SAMARENDRA, MAITI, N, MICETICH, R. G

“…A rapid and rugged solid-phase extraction-liquid chromatographic-electrospray tandem mass spectrometric method has been developed to quantitate two novel human…”
Get full text

High-performance liquid chromatographic analysis of new triazole antifungal agent SYN-2869 and its derivatives in plasma by Khan, Jehangir K, Montaseri, Hashem, Poglod, Marzena, Bu, Hai-Zhi, Daneshtalab, Mohsen, Micetich, Ronald G

“…A simple reversed-phase high-performance liquid chromatography (HPLC) method with UV detection was developed and validated for the quantitation of SYN-2869, a…”
Get full text

Sensitive high-performance liquid chromatographic assay for norfloxacin utilizing fluorescence detection by Hussain, Mohammed S., Chukwumaeze-Obiajunwa, Vern, Micetich, Ronald G.

“…A rapid, sensitive and reproducible reversed-phase high-performance liquid chromatographic assay was developed for the determination of norfloxacin. Following…”
Get full text

Studies on penam sulfones III. Synthesis and β-lactamase inhibitory activity of sodium (6R)-6-(α-hydroxybenzyl)-2β-methoxyiminomethyl-2α-methylpenam-3α-carboxylate 1,1-dioxide and sodium 2β-acyl-2α-methylpenam-3α-carboxylate 1,1-dioxide by Czajkowski, David P, Reddy, Andhe V.N, Setti, Eduardo L, Phillips, Oludotun A, Micetich, Ronald G, Kunugita, Chieko, Maiti, Samarendra N

“…The synthesis and in vitro synergies of (6R)-6-(α-hydroxybenzyl)-2β-methoxyiminomethyl-2α-methylpenam-3α-carboxylate 1,1-dioxide ( 4) and…”
Get full text

Studies on Reactive Intermediates. Part VI. Synthesis of Benzo[a]quinolizines via Methylketene Dimer by Daneshtalab, Mohsen, G. Micetich, Ronald, Forghanifar, Sedighe

Get full text