Search Results - "May, Nóra V."

New Water-Soluble Copper(II) Complexes with Morpholine–Thiosemicarbazone Hybrids: Insights into the Anticancer and Antibacterial Mode of Action by Ohui, Kateryna, Afanasenko, Eleonora, Bacher, Felix, Ting, Rachel Lim Xue, Zafar, Ayesha, Blanco-Cabra, Núria, Torrents, Eduard, Dömötör, Orsolya, May, Nóra V, Darvasiova, Denisa, Enyedy, Éva A, Popović-Bijelić, Ana, Reynisson, Jóhannes, Rapta, Peter, Babak, Maria V, Pastorin, Giorgia, Arion, Vladimir B

“…Six morpholine-(iso)­thiosemicarbazone hybrids HL 1 –HL 6 and their Cu­(II) complexes with good-to-moderate solubility and stability in water were synthesized…”
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Cu(II) and Zn(II) Complexes of New 8‑Hydroxyquinoline Schiff Bases: Investigating Their Structure, Solution Speciation, and Anticancer Potential by Côrte-Real, Leonor, Pósa, Vivien, Martins, Matilde, Colucas, Raquel, May, Nóra V., Fontrodona, Xavier, Romero, Isabel, Mendes, Filipa, Pinto Reis, Catarina, Gaspar, Maria Manuela, Pessoa, João Costa, Enyedy, Éva A., Correia, Isabel

“…We report the synthesis and characterization of three novel Schiff bases (L1–L3) derived from the condensation of 2-carbaldehyde-8-hydroxyquinoline with amines…”
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Direct ortho‐Trifluoroethylation of Aromatic Ureas by Palladium Catalyzed C‐H activation: A Missing Piece of Aromatic Substitutions by Kovács, Szabolcs, Tóth, Balázs L., Borsik, Gábor, Bihari, Tamás, May, Nóra V., Stirling, András, Novák, Zoltán

“…Development of direct late‐stage installation of alkyl groups into aromatic systems is an important and challenging task of current organic chemistry. In spite…”
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A Comparative Study on the Complexation of the Anticancer Iron Chelator VLX600 with Essential Metal Ions by Pósa, Vivien, Federa, Anja, Cseh, Klaudia, Wenisch, Dominik, Spengler, Gabriella, May, Nóra V., Lihi, Norbert, Samu, Gergely F., Jakupec, Michael A., Keppler, Bernhard K., Kowol, Christian R., Enyedy, Éva A.

“…As cancer cells exhibit an increased uptake of iron, targeting the interaction with iron has become a straightforward strategy in the fight against cancer…”
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The Role of the Cysteine Fragments of the Nickel Binding Loop in the Activity of the Ni(II)-Containing SOD Enzyme by Lihi, Norbert, Kelemen, Dóra, May, Nóra V, Fábián, István

“…Detailed equilibrium, spectroscopic, and SOD activity studies are reported on nickel­(II) complexes formed with the N-terminally free HHDLPCGVY-NH2 (NiSODHH)…”
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Binding Models of Copper(II) Thiosemicarbazone Complexes with Human Serum Albumin: A Speciation Study by May, Nóra V., Jancsó, Attila, Enyedy, Éva A.

“…Copper(II) complexes of thiosemicarbazones (TSCs) often exhibit anticancer properties, and their pharmacokinetic behavior can be affected by their interaction…”
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Impact of copper and iron binding properties on the anticancer activity of 8-hydroxyquinoline derived Mannich bases by Pape, Veronika F S, May, Nóra V, Gál, G Tamás, Szatmári, István, Szeri, Flóra, Fülöp, Ferenc, Szakács, Gergely, Enyedy, Éva A

“…The anticancer activity of 8-hydroxyquinolines relies on complex formation with redox active copper and iron ions. Here we employ UV-visible spectrophotometry…”
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Stabilization of the Nickel Binding Loop in NiSOD and Related Model Complexes: Thermodynamic and Structural Features by Lihi, Norbert, Csire, Gizella, Szakács, Bence, May, Nóra V, Várnagy, Katalin, Sóvágó, Imre, Fábián, István

“…Detailed equilibrium and spectroscopic characterization of the complex formation processes of the nickel binding loop in NiSOD and its related fragments is…”
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Gradual Changes in the Aromaticity in a Series of Hydroxypyridine-Carboxylic Acid Derivatives and Their Effect on Tautomerism and Crystal Packing by May, Nóra V., Gál, G. Tamás, Holczbauer, Tamás, Bereczki, Laura, Di Marco, Valerio B., Bombicz, Petra

“…The keto–enol tautomerism of hydroxypyridine-carboxylic acid (HPC) derivatives with proton transfer between the hydroxyl or carboxyl oxygen atoms was…”
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Complex formation of ML324, the histone demethylase inhibitor, with essential metal ions: Relationship between solution chemistry and anticancer activity by Kovács, Hilda, Jakusch, Tamás, May, Nóra V., Tóth, Szilárd, Szakács, Gergely, Enyedy, Éva A.

“…N-(3-(dimethylamino)propyl-4-(8-hydroxyquinolin-6-yl)benzamide (ML324, HL) is a potent inhibitor of the iron-containing histone demethylase KDM4, a recognized…”
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Solution Equilibrium Studies on Salicylidene Aminoguanidine Schiff Base Metal Complexes: Impact of the Hybridization with L-Proline on Stability, Redox Activity and Cytotoxicity by Dömötör, Orsolya, May, Nóra V, Gál, G Tamás, Spengler, Gabriella, Dobrova, Aliona, Arion, Vladimir B, Enyedy, Éva A

“…The proton dissociation processes of two tridentate salicylidene aminoguanidine Schiff bases (SISC, Pro-SISC-Me), the solution stability and electrochemical…”
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Synthesis of dihydrotestosterone derivatives modified in the A-ring with (hetero)arylidene, pyrazolo[1,5-a]pyrimidine and triazolo[1,5-a]pyrimidine moieties and their targeting of the androgen receptor in prostate cancer by Kiss, Márton A., Peřina, Miroslav, Bazgier, Václav, May, Nóra V., Baji, Ádám, Jorda, Radek, Frank, Éva

“…[Display omitted] •Novel 2-arylidene derivatives of 5α-dihydrotestosterone have been synthesized.•Heterocyclizations of the α,β-enones were performed with…”
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Copper Coordination Chemistry of Sulfur Pendant Cyclen Derivatives: An Attempt to Hinder the Reductive-Induced Demetalation in 64/67Cu Radiopharmaceuticals by Tosato, Marianna, Dalla Tiezza, Marco, May, Nóra V, Isse, Abdirisak Ahmed, Nardella, Sonia, Orian, Laura, Verona, Marco, Vaccarin, Christian, Alker, André, Mäcke, Helmut, Pastore, Paolo, Di Marco, Valerio

“…The Cu2+ complexes formed by a series of cyclen derivatives bearing sulfur pendant arms,…”
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Diagnosis of Melanoma with 61Cu-Labeled PET Tracer by Bunda, Szilvia, Kálmán-Szabó, Ibolya, Lihi, Norbert, Képes, Zita, Szikra, Dezső, Peline Szabo, Judit, Timári, István, Szücs, Dániel, May, Nóra V., Papp, Gábor, Trencsényi, György, Kálmán, Ferenc K.

“…Until the recent years, substances containing radioactive 61Cu were strongly considered as potential positron-emitting radiopharmaceuticals for use in positron…”
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Structural and solution speciation studies on selected [Cu(NN)(OO)] complexes and an investigation of their biomimetic activity, ROS generation and their cytotoxicity in normoxic, hypoxic and anoxic environments in MCF-7 breast cancer-derived cells by Jenkins, Hollie, MacLean, Louise, McClean, Siobhán, Cooke, Gordon, Devereux, Michael, Howe, Orla, Pereira, Marcos D., May, Nóra V., Enyedy, Éva A., Creaven, Bernadette S.

“…Reactive oxygen species(ROS) generation with subsequent DNA damage is one of the principle mechanisms of action assigned to copper-based anticancer complexes…”
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Copper(II) Complexes of Pyridine-2,6-dicarboxamide Ligands with High SOD Activity by Diószegi, Róbert, Bonczidai-Kelemen, Dóra, Bényei, Attila Cs, May, Nóra V, Fábián, István, Lihi, Norbert

“…Copper­(II) complexes of pyridine-based ligands functionalized with alanine (PydiAla) and tyrosine (PydiTyr) moieties have been synthesized as novel superoxide…”
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Copper(II) Complexes of Sulfonated Salan Ligands: Thermodynamic and Spectroscopic Features and Applications for Catalysis of the Henry Reaction by Bunda, Szilvia, May, Nóra V, Bonczidai-Kelemen, Dóra, Udvardy, Antal, Ching, H. Y. Vincent, Nys, Kevin, Samanipour, Mohammad, Van Doorslaer, Sabine, Joó, Ferenc, Lihi, Norbert

“…Copper­(II) complexes formed with sulfonated salan ligands (HSS) have been synthesized, and their coordination chemistry has been characterized using…”
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Comparative solution equilibrium studies of antitumor ruthenium(η 6 -p-cymene) and rhodium(η 5 -C 5 Me 5 ) complexes of 8-hydroxyquinolines by Dömötör, Orsolya, Pape, Veronika F S, May, Nóra V, Szakács, Gergely, Enyedy, Éva A

“…Complex formation processes of [Ru(η -p-cymene)(H O) ] and [Rh(η -C Me )(H O) ] organometallic cations with 8-hydroxyquinoline (HQ) ligands were studied in…”
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8-Hydroxyquinoline-Amino Acid Hybrids and Their Half-Sandwich Rh and Ru Complexes: Synthesis, Anticancer Activities, Solution Chemistry and Interaction with Biomolecules by Pivarcsik, Tamás, Dömötör, Orsolya, Mészáros, János P, May, Nóra V, Spengler, Gabriella, Csuvik, Oszkár, Szatmári, István, Enyedy, Éva A

“…Solution chemical properties of two novel 8-hydroxyquinoline-D-proline and homo-proline hybrids were investigated along with their complex formation with [Rh(η…”
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Effect of the Additional Carboxyl Group in Half‐Sandwich Organometallic 2,4‐Dipicolinate Complexes on Solution Speciation and Structure by Mészáros, János P., Németi, Gábor, Poljarevic, Jelena M., Holczbauer, Tamás, May, Nóra V., Enyedy, Éva A.

“…Solution speciation of Rh(η5‐C5Me5), Ru(η6‐p‐cymene) and Ru(η6‐toluene) complexes of 2,4‐pyridinedicarboxylic acid (2,4‐dipicH2) was studied and compared to…”
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