Search Results - "Massarelli, P"

PHENOLIC COMPOUNDS, CAROTENOIDS AND ANTIOXIDANT ACTIVITY IN FIVE TOMATO CULTIVARS by Zanfini, A, Franchi, G.G, Massarelli, P, Corbini, G, Dreassi, E

“…In this study we examined the antioxidants content (polyphenols and carotenoids) and the total hydrophilic (HAA) and lipophilic (LAA) antioxidant activity of…”
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Nuclear magnetic resonance for studying recognition processes between anandamide and cannabinoid receptors by Bonechi, C., Martini, S., Brizzi, V., Brizzi, A., Massarelli, P., Bruni, G., Rossi, C.

“…The understanding of the molecular basis of cannabinoid activity has greatly improved since the discovery of CB1 and CB2 receptors. In this paper, the ligand…”
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Synthesis and in vitro pharmacological evaluation of a new series of 5-HT1A 5-HT2A and 5-HT2C receptor ligands containing a norbornene nucleus by Fiorino, F, Severino, B, De Angelis, F, Perissutti, E, Magli, E, Frecentese, F, Esposito, A, Massarelli, P, Nencini, C, Viti, B, Santagada, V, Caliendo, G

“…A series of 4-substituted piperazine derivatives bearing a norbornene nucleus have been prepared and their affinity for serotonin 5-HT1A, 5-HT2A and 5-HT2C…”
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High affinity central benzodiazepine receptor ligands: synthesis and structure-activity relationship studies of a new series of pyrazolo[4,3-c]quinolin-3-ones by Savini, L, Massarelli, P, Nencini, C, Pellerano, C, Biggio, G, Maciocco, A, Tuligi, G, Carrieri, A, Cinone, N, Carotti, A

“…A large series of 2-aryl(heteroaryl)-2,5-dihydropyrazolo[4,3-c]quinolin- 3-(3H)-ones, carrying appropriate substituents at the quinoline and N2-phenyl rings,…”
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Chelating agents as potential antitumorals. 2-quinolylhydrazones and bis-2-quinolylhydrazones. I by Savini, L, Massarelli, P, Chiasserini, L, Sega, A, Pellerano, C, Barzi, A, Nocentini, G

“…A number of pyruvic acid, methylpyruvate and pyruvic carboxaldehyde 2-quinolylhydrazones have been synthesized. Some bis-2-quinolylhydrazones were also…”
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Chelating agents as potential antitumorals: alpha-(N)-heterocyclic hydrazones and bis-alpha-(N)-heterocyclic hydrazones by Savini, L, Massarelli, P, Chiasserini, L, Nencini, C, Pellerano, C

“…A number of pyruvic acid and methylpyruvate alpha-(N)-heterocyclic hydrazones has been synthesized. Bis-heterocyclic hydrazones were obtained from reaction…”
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Mechanical and metabolic alterations in rat diaphragm during electrical stimulation by Massarelli, P S, Green, H J, Hughson, R L, Sharratt, M T

“…To investigate the hypothesis that the rate of fatigue development is not influenced by the absolute duration of contraction (train duration) and relaxation…”
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New quinoline derivatives: synthesis and evaluation for antiinflammatory and analgesic properties--Note II by Savini, L, Massarelli, P, Pellerano, C, Bruni, G

“…The synthesis of new halogenated series of 4-anilinoquinoline-3-carboxylic acids, N-[3-carboxyquinolyl(4)]anthranilic acids and their corresponding esters is…”
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Synthesis of 4-quinolylazide derivatives and evaluation of their antitumor and antimicrobial activity by Savini, L, Massarelli, P, Pellerano, C

“…Synthesis and pharmacological evaluation of a series of 4-quinolylazide derivatives are reported. These were screened against P388 lymphocitic leukemia in…”
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New 1-[quinolyl(4)]-1,2,3-triazoles: synthesis and evaluation of antiinflammatory and analgesic properties. I by Savini, L, Massarelli, P, Corti, P, Chiasserini, L, Pellerano, C, Bruni, G

“…The synthesis of new 1-[quinolyl(4)]-1,2,3-triazoles is reported. These have been obtained by reacting 4-azidoquinolines with ethyl p-nitrobenzoylacetate. The…”
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New 5-hydroxytryptamine(1A) receptor ligands containing a norbornene nucleus: synthesis and in vitro pharmacological evaluation by Fiorino, Ferdinando, Perissutti, Elisa, Severino, Beatrice, Santagada, Vincenzo, Cirillo, Donatella, Terracciano, Sara, Massarelli, Paola, Bruni, Giancarlo, Collavoli, Elga, Renner, Christian, Caliendo, Giuseppe

“…New arylpiperazine derivatives were prepared to identify highly selective and potent ligands for the 5-hydroxytryptamine 1A (5-HT(1A)) receptor as potential…”
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Anti-inflammatory and analgesic effects of Spartium junceum L. flower extracts: a preliminary study by Menghini, Luigi, Massarelli, Paola, Bruni, Giancarlo, Pagiotti, Rita

“…Our objective was to study the anti-inflammatory and analgesic activity of extract of Spartium junceum L. flowers. Samples of flowers were collected from wild…”
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Pyrazolo[4,3-c]quinolines, synthesis and specific inhibition of benzodiazepine receptor binding. Note II by Savini, L, Massarelli, P, Corti, P, Pellerano, C, Bruni, G, Romeo, M R

“…Two new series of 2-arylpyrazolo[4,3-c]quinolin-3-ones (6,8-difluoro- and 7,9-dichloro-derivatives) have been synthesized and tested for their ability to…”
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Pyrazolo [4,3-c] quinolines synthesis and specific inhibition of benzodiazepine receptor binding (Note I) by Savini, L, Massarelli, P, Pellerano, C, Fiorini, I, Bruni, G, Romeo, M R

“…A series of 2-arylpyrazolo[4,3-c] quinolin-3-one derivatives, bearing different substituents in the two aromatic rings, were prepared and tested for their…”
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Preliminary evaluation on anti-inflammatory and analgesic effects of Sideritis syriaca L. herba extracts by Menghini, Luigi, Massarelli, Paola, Bruni, Giancarlo, Menghini, Alessandro

“…We studied the anti-inflammatory and analgesic activity of extracts of Sideritis syriaca L. herba. Samples were collected from the wild plant, dried, powdered,…”
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Synthesis of 6beta-D-glucosyl and 6-nitroxy (-)-galanthamine derivatives as acetylcholinesterase inhibitors by Perissutti, E, Fiorino, F, Severino, B, Frecentese, F, Massarelli, P, Nencini, C, Santagada, V, Caliendo, G

“…Galanthamine is an alkaloid approved for the treatment of Alzheimer's disease. In this paper the syntheses and the anticholinesterase activities of new…”
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New 5-Hydroxytryptamine sub(1A) Receptor Ligands Containing a Norbornene Nucleus: Synthesis and in Vitro Pharmacological Evaluation by Fiorino, F, Perissutti, E, Severino, B, Santagada, V, Cirillo, D, Terracciano, S, Massarelli, P, Bruni, G, Collavoli, E, Renner, C, Caliendo, G

“…New arylpiperazine derivatives were prepared to identify highly selective and potent ligands for the 5-hydroxytryptamine 1A (5-HT sub(1A)) receptor as…”
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Antiinflammatory and Analgesic Activities of Two Dicyclic Analogues of Acetaminophen and Its Regioisomer 3-Hydroxyacetanilide by Iakovou, K., Varvaresou, A., Bruni, G., Massarelli, P., Vavayannis, A., Kazanis, M.

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Synthesis of oxypropanolamine derivatives of 3,4-dihydro-2H-1,4-benzoxazine, β-adrenergic affinity, inotropic, chronotropic and coronary vasodilating activities by IAKOVOU, K, KAZANIS, M, VAVAYANNIS, A, BRUNI, G, ROMEO, M. R, MASSARELLI, P, TERAMOTO, S, FUJIKI, H, MORI, T

“…Aseries of oxypropanolamine derivatives of 3,4-dihydro-2H-1,4-benzoxazine were synthesized and evaluated for inotropic, chronotropic and coronary vasodilating…”
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The relationship between single-breath diffusion capacity of the lung for nitric oxide and carbon monoxide during various exercise intensities by Zavorsky, Gerald S, Quiron, Karine Badra, Massarelli, Philip S, Lands, Larry C

“…To determine the relationship between single-breath diffusion capacity of the lung for nitric oxide (DLNO) and single-breath diffusion capacity of the lung for…”
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