Search Results - "Mascarello, A."
-
1
Characterization and cytotoxic activity of sulfated derivatives of polysaccharides from Agaricus brasiliensis
Published in International journal of biological macromolecules (01-06-2013)“…•Polysaccharides were isolated from Agaricus brasiliensis fruiting body (FR) and mycelia (MI).•The sulfated derivatives FR-S and MI-S were prepared.•FR, FR-S,…”
Get full text
Journal Article -
2
Relation between lipophilicity of alkyl gallates and antifungal activity against yeasts and filamentous fungi
Published in Bioorganic & medicinal chemistry letters (15-03-2009)“…When the log P of each gallate was calculated and related to the different values of MIC against Microsporum gypseum it was observed that hexyl, heptyl, octyl…”
Get full text
Journal Article -
3
Novel Dihydropteridinone Derivatives As Potent Inhibitors of the Understudied Human Kinases Vaccinia-Related Kinase 1 and Casein Kinase 1δ/ε
Published in Journal of medicinal chemistry (13-06-2024)“…Vaccinia-related kinase 1 (VRK1) and the δ and ε isoforms of casein kinase 1 (CK1) are linked to various disease-relevant pathways. However, the lack of tool…”
Get full text
Journal Article -
4
Quinoxaline-substituted chalcones as new inhibitors of breast cancer resistance protein ABCG2: polyspecificity at B-ring position
Published in Drug design, development and therapy (01-01-2014)“…A series of chalcones substituted by a quinoxaline unit at the B-ring were synthesized and tested as inhibitors of breast cancer resistance protein-mediated…”
Get full text
Journal Article -
5
New structure-activity relationships of chalcone inhibitors of breast cancer resistance protein: polyspecificity toward inhibition and critical substitutions against cytotoxicity
Published in Drug design, development and therapy (01-01-2013)“…Adenosine triphosphate-binding cassette subfamily G member 2 (ABCG2) plays a major role in cancer cell multidrug resistance, which contributes to low efficacy…”
Get full text
Journal Article