Search Results - "Markov, Pavel O."

Cyclodextrin Polymers as a Promising Drug Carriers for Stabilization of Meropenem Solutions by Yakupova, Linara R, Skuredina, Anna A, Markov, Pavel O, Le-Deygen, Irina M, Kudryashova, Elena V

“…Here we report the development of new drug carriers for meropenem based on the hydroxypropyl-β-cyclodextrin (HPCD) polymers with variable linkers, namely,…”
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Preclinical Optimization of gp120 Entry Antagonists as anti-HIV‑1 Agents with Improved Cytotoxicity and ADME Properties through Rational Design, Synthesis, and Antiviral Evaluation by Curreli, Francesca, Ahmed, Shahad, Benedict Victor, Sofia M, Iusupov, Ildar R, Belov, Dmitry S, Markov, Pavel O, Kurkin, Alexander V, Altieri, Andrea, Debnath, Asim K

“…We previously reported a milestone in the optimization of NBD-11021, an HIV-1 gp120 antagonist, by developing a new and novel analogue, NBD-14189 (Ref1), which…”
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Design of gp120 HIV-1 entry inhibitors by scaffold hopping via isosteric replacements by Iusupov, Ildar R., Curreli, Francesca, Spiridonov, Evgeniy A., Markov, Pavel O., Ahmed, Shahad, Belov, Dmitry S., Manasova, Ekaterina V., Altieri, Andrea, Kurkin, Alexander V., Debnath, Asim K.

“…We present the development of alternative scaffolds and validation of their synthetic pathways as a tool for the exploration of new HIV gp120 inhibitors based…”
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Design, Synthesis, and Antiviral Activity of the Thiazole Positional Isomers of a Potent HIV‐1 Entry Inhibitor NBD‐14270 by Kurkin, Alexander V., Curreli, Francesca, Iusupov, Ildar R., Spiridonov, Evgeniy A., Ahmed, Shahad, Markov, Pavel O., Manasova, Ekaterina V., Altieri, Andrea, Debnath, Asim K.

“…The envelope glycoprotein gp120 of human immunodeficiency virus type 1 (HIV‐1) plays a critical role in virus entry to the cells by binding to the host…”
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Front Cover: Design, Synthesis, and Antiviral Activity of the Thiazole Positional Isomers of a Potent HIV‐1 Entry Inhibitor NBD‐14270 (ChemMedChem 22/2022) by Kurkin, Alexander V., Curreli, Francesca, Iusupov, Ildar R., Spiridonov, Evgeniy A., Ahmed, Shahad, Markov, Pavel O., Manasova, Ekaterina V., Altieri, Andrea, Debnath, Asim K.

“…The Front Cover shows the interactions of the HIV‐1 envelope glycoprotein gp120 with two sets of NBD compounds (HIV‐1 entry inhibitors) representing three…”
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