Search Results - "Maiereanu, Carmen"

3,7-Dioxa-1-azabicyclo[3.3.0]octanes Substituted at the C-5 Position − From Local to Global Stereochemistry by Darabantu, Mircea, Maiereanu, Carmen, Silaghi-Dumitrescu, Ioan, Toupet, Loïc, Condamine, Eric, Ramondenc, Yvan, Berghian, Camelia, Plé, Gérard, Plé, Nelly

“…Multiple approaches are described for the elucidation of the stereochemistry in solution (high‐resolution NMR spectroscopy) and in the solid state (X‐ray…”
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Exploring S1 plasticity and probing S1′ subsite of mammalian aminopeptidase N/CD13 with highly potent and selective aminobenzosuberone inhibitors by Revelant, Germain, Al-Lakkis-Wehbe, Mira, Schmitt, Marjorie, Alavi, Sarah, Schmitt, Céline, Roux, Lionel, Al-Masri, Mounir, Schifano-Faux, Nadège, Maiereanu, Carmen, Tarnus, Céline, Albrecht, Sébastien

“…[Display omitted] In order to probe the S1 and S1′ mammalian aminopeptidase N subsites, racemic 1- or 4-substituted 7-aminobenzocyclohepten-6-one derivatives…”
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A novel amino-benzosuberone derivative is a picomolar inhibitor of mammalian aminopeptidase N/CD13 by Maiereanu, Carmen, Schmitt, Céline, Schifano-Faux, Nadège, Le Nouën, Didier, Defoin, Albert, Tarnus, Céline

“…Some racemic amino-benzosuberones 1a–h′, were synthesised and evaluated as inhibitors of four representative members of zinc-dependent amino-peptidases. Ki…”
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Synthesis and biological evaluation of novel benzodioxinocarbazoles (BDCZs) as potential anticancer agents by Ayerbe, Nathalie, Routier, Sylvain, Gillaizeau, Isabelle, Maiereanu, Carmen, Caignard, Daniel-Henry, Pierré, Alain, Léonce, Stéphane, Coudert, Gérard

“…We report the efficient synthesis and biological evaluation of new benzodioxinoindolocarbazoles heterocycles (BDCZs) designed as potential anticancer agents…”
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Quantitative structure—retention and retention—activity relationships of some 1,3-oxazolidine systems by RP-HPTLC and PCA by Sârbu, C, Casoni, Dorina, Darabantu, M, Maiereanu, Carmen

“…A quantitative structure–retention and retention–activity relationships investigations were performed on the lipophilicities of some 1,3-oxazolidine systems as…”
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α-(3,7-Dioxa- r-1-azabicyclo[3.3.0]oct- c-5-ylmethoxy)-diazines. Part 1: Synthesis and stereochemistry. Extension to s-triazine series by Berghian, Camelia, Lameiras, Pedro, Toupet, Loïc, Condamine, Eric, Plé, Nelly, Turck, Alain, Maiereanu, Carmen, Darabantu, Mircea

“…The general and efficient synthesis of the title compounds, consisting of the (selective) replacement of chlorine in commercial α-chlorodiazines and cyanuryl…”
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α-(3,7-Dioxa- r-1-azabicyclo[3.3.0]oct- c-5-ylmethoxy)-diazines. Part 2: Functionalisation via directed ortho-metallation and cross-coupling reactions by Berghian, Camelia, Condamine, Eric, Plé, Nelly, Turck, Alain, Silaghi-Dumitrescu, Ioan, Maiereanu, Carmen, Darabantu, Mircea

“…The functionalisation of the title compounds via regioselective Directed ortho-Metallation (DoM) and cross-coupling reactions is studied. The compatibility of…”
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Ring-chain tautomerism and other versatile behaviour of 1,4-diimino- and 1,2-phenylene derivatives of some C-substituted serinols by Maiereanu, Carmen, Darabantu, Mircea, Plé, Gérard, Berghian, Camelia, Condamine, Eric, Ramondenc, Yvan, Silaghi-Dumitrescu, Ion, Mager, Sorin

“…The behaviour of the title compounds, obtained from terephthaldicarboxaldehyde or 1,2-phthaldicarboxaldehyde and certain (non)chiral C-substituted serinols is…”
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Synthesis and Stereochemistry of Some 1,3-Oxazolidine Systems Based on TRIS (α,α,α-trimethylolaminomethane) and Related Aminopolyols Skeleton. Part 2: 1-Aza-3,7-dioxabicyclo[3.3.0]octanes by Darabantu, Mircea, Plé, Gérard, Maiereanu, Carmen, Silaghi-Dumitrescu, Ion, Ramondenc, Yvan, Mager, Sorin

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Synthesis of 2-Deoxy-2-thiophenylglucosyl Azides through 1,2 Thio Migration of Thiophenyl Mannosides by Maiereanu, Carmen, Kanai, Akira, Weibel, Jean-Marc, Pale, Patrick

“…2-Deoxy-2-thio glucosyl azides bearing or not bearing an azido group at the 6-position can be conveniently obtained through a 1,2-thio migration from…”
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Synthesis and Stereochemistry of Some 1,3-Oxazolidine Systems Based on TRIS (α,α,α-Trimethylolaminomethane) and Related Aminopolyols Skeleton. Part 1: (Di)spiro-1,3-oxazolidines by Darabantu, Mircea, Plé, Gérard, Silaghi-Dumitrescu, Ion, Maiereanu, Carmen, Turos, Istvan, Silberg, Ioan A, Mager, Sorin

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