Search Results - "Maeda, D Y"

CXCR2 expression during melanoma tumorigenesis controls transcriptional programs that facilitate tumor growth by Yang, J, Bergdorf, K, Yan, C, Luo, W, Chen, S C, Ayers, G D, Liu, Q, Liu, X, Boothby, M, Weiss, V L, Groves, S M, Oleskie, A N, Zhang, X, Maeda, D Y, Zebala, J A, Quaranta, V, Richmond, A

“…Though the CXCR2 chemokine receptor is known to play a key role in cancer growth and response to therapy, a direct link between expression of CXCR2 in tumor…”
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A Sigma-1 receptor selective analogue of BD1008. A potential substitute for (+)-opioids in sigma receptor binding assays by MAEDA, D. Y, WILLIAMS, W, BOWEN, W. D, COOP, A

“…A simple, achiral monoamine sigma-1 (sigma1) receptor selective ligand (sigma2Ki/sigma1Ki>2000) is described, which could replace the chiral (+)-pentazocine or…”
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Synthesis and Evaluation of Isothiocyanate-Containing Derivatives of the δ-Opioid Receptor Antagonist Tyr-Tic-Phe-Phe (TIPP) as Potential Affinity Labels for δ-Opioid Receptors by Maeda, Dean Y, Berman, Fred, Murray, Thomas F, Aldrich, Jane V

“…Derivatives of the δ-opioid receptor-selective peptide antagonist H-Tyr-Tic-Phe-Phe-OH (TIPP) containing an isothiocyanate moiety at the para position of…”
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Synthesis and Evaluation of N,N-Dialkyl Enkephalin-Based Affinity Labels for δ Opioid Receptors by Maeda, Dean Y, Ishmael, Jane E, Murray, Thomas F, Aldrich, Jane V

“…To develop affinity labels for δ opioid receptors based on peptide antagonists, the Phe4 residues of N,N-dibenzylleucine enkephalin and…”
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Identification of a New Class of Molecules, the Arachidonyl Amino Acids, and Characterization of One Member That Inhibits Pain by Huang, S M, Bisogno, T, Petros, T J, Chang, S Y, Zavitsanos, P A, Zipkin, R E, Sivakumar, R, Coop, A, Maeda, D Y, De Petrocellis, L, Burstein, S, Di Marzo, V, Walker, J M

“…In mammals, specific lipids and amino acids serve as crucial signaling molecules. In bacteria, conjugates of lipids and amino acids (referred to as lipoamino…”
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Binding characteristics of the gamma-hydroxybutyric acid receptor antagonist [(3)H](2E)-(5-hydroxy-5,7,8,9-tetrahydro-6H-benzo[a][7]annulen-6-ylidene) ethanoic acid in the rat brain by Mehta, A K, Muschaweck, N M, Maeda, D Y, Coop, A, Ticku, M K

“…Radioligand binding studies with [(3)H](2E)-(5-hydroxy-5,7,8,9-tetrahydro-6H-benzo[a][7]annulen-6-ylidene) ethanoic acid ([(3)H]NCS-382), an antagonist of…”
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Bivalent inhibitors of glutathione S-transferase: The effect of spacer length on isozyme selectivity by Maeda, Dean Y., Mahajan, Sumit S., Atkins, William M., Zebala, John A.

“…Bivalent inhibitors based on ethacrynic acid (EA) were synthesized and evaluated for inhibition of glutathione S-transferase (GST) A1-1 and GST P1-1…”
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N-Arylalkylpiperidines as High-Affinity Sigma-1 and Sigma-2 Receptor Ligands: Phenylpropylamines as Potential Leads for Selective Sigma-2 Agents by Maeda, Dean Y., Williams, Wanda, Kim, Wes E., Thatcher, Linn N., Bowen, Wayne D., Coop, Andrew

“…To delineate the differences between the structural requirements necessary for recognition at sigma-1 and sigma-2 receptors, a range of phenethyl- and…”
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Studies into the Direct Conversion of Indolomorphinans to their 4-Phenolic Derivatives by Maeda, Dean Y, Coop, Andrew

“…A one step method to convert 3- O-methyl substituted indolomorphinans into their 4-phenolic derivatives through reductive opening of the 4,5-bridge is…”
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