Search Results - "Madar, Jyoti"

Design, synthesis, characterization, and biological evaluation of pyrido[1,2-a]pyrimidinone coumarins as promising anti-inflammatory agents by Madar, Jyoti M., Shastri, Lokesh A., Shastri, Samundeeswari L., Holiyachi, Megharaja, Naik, Nirmala, Kulkarni, Rashmi, Shaikh, Farzanabi, Sungar, Vinay

“…Pursuing our recent interest regarding antimicrobial and anti-inflammatory activities of coumarin derivatives, we have synthesized a series of coumarin-linked…”
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Synthesis of Naked-eye Detectable Fluorescent 2H-chromen-2-One 2, 6-Dicyanoanilines: Effect of Substituents and pH on Its Luminous Behavior by Kulkarni, Rashmi C., Samundeeswari, S., Shaikh, Farzanabi, Naik, Nirmala S., Madar, Jyoti M., Shastri, Lokesh A., Sunagar, Vinay A.

“…A variety of new coumarin derivatives containing C-4 bridged 2,6-dicyanoanilines ( 4a-4d ) were synthesized via multicomponent one pot approach. These novel…”
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Solvent-Free Synthesis, Characterization, and In Vitro Biological Activity Study of Xanthenediones and Acridinediones by Madar, Jyoti M., Samundeeswari, S., Holiyachi, Megharaja, Naik, Nirmala S., Pawar, Varsha, Gudimani, Parashuram, Shastri, Lokesh A., Kumbar, Vijay M., Sunagar, Vinay A.

“…The present work highlights the broad range of oxygen and nitrogen heterocycles and their applications in medicinal field. A facial approach has been developed…”
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3,4-Dihydropyrimidinone-coumarin analogues as a new class of selective agent against S. aureus: Synthesis, biological evaluation and molecular modelling study by Naik, Nirmala S., Shastri, Lokesh A., Joshi, Shrinivas D., Dixit, Sheshagiri R., Chougala, Bahubali M., Samundeeswari, S., Holiyachi, Megharaj, Shaikh, Farzanabi, Madar, Jyoti, Kulkarni, Rashmi, Sunagar, Vinay

“…[Display omitted] •An efficient protocol has been developed for the synthesize of dihydropyrimidin-2(1H)-one/thione derivatives of coumarin from substituted…”
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Synthesis, Antitubercular and Antimicrobial Activity of 1,2,4‐Triazolidine‐3‐thione Functionalized Coumarin and Phenyl Derivatives and Molecular Docking Studies by Shaikh, Farzanabi, Shastri, Samundeeswari L., Naik, Nirmala S., Kulkarni, Rashmi, Madar, Jyoti M., Shastri, Lokesh A., Joshi, Shrinivas D., Sunagar, Vinay

“…Tuberculosis (TB) is still a demanding worldwide health problem and mycobacterium tuberculosis (MTB) remains one of the most toxic human pathogens. In pursuit…”
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Design and synthesis of coumarin–imidazole hybrid and phenyl-imidazoloacrylates as potent antimicrobial and antiinflammatory agents by Holiyachi, Megharaja, Samundeeswari, S., Chougala, Bahubali M., Naik, Nirmala S., Madar, Jyoti, Shastri, Lokesh A., Joshi, Shrinivas D., Dixit, Sheshagiri R., Dodamani, Suneel, Jalalpure, Sunil, Sunagar, Vinay A.

“…An improved one pot, multi-component synthesis of tri- and tetrasubstituted coumarin–imidazole hybrid has been synthesized at C4 position in good to excellent…”
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Synthesis of Polyfunctionalized Fused Pyrazolo‐Pyridines: Characterization, Anticancer Activity, Protein Binding and Molecular Docking Studies by Naik, Nirmala S., Shastri, Lokesh A., Shastri, Samundeeswari L., Chougala, Bahubali M., Shaikh, Farzanabi, Madar, Jyoti M., Kulkarni, Rashmi C., Dodamani, Suneel, Jalalpure, Sunil, Joshi, Shrinivas D., Sunagar, Vinay

“…The reaction of a multi‐substituted pyrazole 1 with aryl or heteroaryl aldehydes and active methylene compounds afford unexpected pyrazolo[1,5‐a]pyridine…”
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The anti‐inflammatory Design, Synthesis and Exploiting Pharmacological Activities of 2,3‐Dihydrofuranocoumarins as Multi‐Therapeutic Agents by Madar, Jyoti M., Shastri, Lokesh A., Shastri, Samundeeswari L., Holiyachi, Megharaja, Naik, Nirmala S., Shaikh, Farzanabi, Kumbar, Vijay M., Bhat, Kishor G., Joshi, Shrinivas D., Sungar, Vinay A.

“…Our recent research interest regarding synthesis of bioactive furanocoumarin derivatives, we have developed pyridinium yield assisted synthesis of…”
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Green synthesis of coumarin-pyrazolone hybrids: In vitro anticancer and anti-inflammatory activities and their computational study on COX-2 enzyme by Kulkarni, Rashmi C., Madar, Jyoti M., Shastri, Samundeeswari L., Shaikh, Farzanabi, Naik, Nirmala S., Chougale, Ravindra B., Shastri, Lokesh A., Joshi, Shrinivas D., Dixit, Sheshagiri R., Sunagar, Vinay A.

“…A series of novel quinoline-2-carboxamides 4(a–l) were synthesized using different 2-oxo-2H-chromene-4-carbaldehyde and 3-methyl-1H-pyrazole-5(4H)-one with…”
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Design and synthesis of structurally identical coumarinotriazoles as cytotoxic and antimicrobial agents by Madar, Jyoti M., Shastri, Lokesh A., Shastri, Samundeeswari L., Guda, Ramu, Holiyachi, Megharaja, Naik, Nirmala S., Dodamani, Suneel, Jalapure, Sunil, Sungar, Vinay A.

“…Novel coumarinotriazoles have been synthesized with excellent yield by 1,3-cycloaddition reaction of substituted coumarin azides with active methylene…”
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