Search Results - "Macri, Bryan"

Novel Transient Receptor Potential Vanilloid 1 Receptor Antagonists for the Treatment of Pain:  Structure−Activity Relationships for Ureas with Quinoline, Isoquinoline, Quinazoline, Phthalazine, Quinoxaline, and Cinnoline Moieties by Gomtsyan, Arthur, Bayburt, Erol K, Schmidt, Robert G, Zheng, Guo Zhu, Perner, Richard J, Didomenico, Stanley, Koenig, John R, Turner, Sean, Jinkerson, Tammie, Drizin, Irene, Hannick, Steven M, Macri, Bryan S, McDonald, Heath A, Honore, Prisca, Wismer, Carol T, Marsh, Kennan C, Wetter, Jill, Stewart, Kent D, Oie, Tetsuro, Jarvis, Michael F, Surowy, Carol S, Faltynek, Connie R, Lee, Chih-Hung

“…Novel transient receptor potential vanilloid 1 (TRPV1) receptor antagonists with various bicyclic heteroaromatic pharmacophores were synthesized, and their in…”
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Impact of Entropic Effects in the Classical Resolution of a 2-Arylpyrrolidine by Barnes, David M, Barkalow, Jufang, Chen, Yong, Gupta, Ashok, Haight, Anthony R, Hengeveld, John E, Kerdesky, Francis A. J, Kotecki, Brian J, Macri, Bryan, Pal, Agnes

“…The impact of entropic effects on the classical salt resolution of a 2-arylpyrrolidine is described. We have found that the crystallization of a racemic…”
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A practical stereoselective synthesis of ( 2S, 4S)-4- tert-butoxycarbonylamino-2-methylpyrrolidine by Li, Qun, Chu, Daniel T.W., Raye, Kathleen, Claiborne, Akiyo, Seif, Louis, Macri, Bryan, Plattner, Jacob J.

“…Two practical syntheses of (2S, 4S)-4-tert-butoxycarbonylamino-2-methylpyrrolidine, an important intermediate for quinolone antibacterial agents, have been…”
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