Search Results - "MATUSZCZAK, B."

N-substituted tetrahydro-2,4-dioxoquinazolin-1-yl acetic acids as aldose reductase inhibitors by Rakowitz, D, Gmeiner, A, Matuszczak, B

“…Novel N-substituted tetrahydro-2,4-dioxoquinazolin-1-yl acetic acids characterized by formal replacement of the substituted benzyl moiety by cyclohexylmethyl…”
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Linear and cyclic N-acetyl-α-aryl-glycines: Synthesis and chemiluminescence studies by Matuszczak, B.

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PP#89 - A proof of concept study with FSC-based hybrid imaging agents for pretargeting applications by Summer, D., Mayr, S., Petrik, M., Hermann, M., Vieider, L., Matuszczak, B., Decristoforo, C.

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A proof of concept study with FSC-based hybrid imaging agents for pretargeting applications by Summer, D., Mayr, S., Petrik, M., Hermann, M., Vieider, L., Matuszczak, B., Decristoforo, C.

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Non-ionic thiolated cyclodextrins - the next generation by Moghadam, Ali, Ijaz, Muhammad, Asim, Mulazim Hussain, Mahmood, Arshad, Jelkmann, Max, Matuszczak, Barbara, Bernkop-Schnürch, Andreas

“…The current study was aimed at developing a novel mucoadhesive thiolated cyclodextrin (CD) without ionizable groups and an intact ring backbone for drug…”
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2′,3′,4′,5′-Tetraacetyl- N(3)-carboxymethylriboflavin derivatives: synthesis and fluorescence studies by Banekovich, Christian, Matuszczak, Barbara

“…[Display omitted] The hitherto not described 2′,3′,4′,5′-tetraacetyl- N(3)-carboxymethylriboflavin ( 1) could be prepared starting from…”
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Substituted Pyridazino[3,4-b][1,5]benzoxazepin-5(6H)ones as Multidrug-Resistance Modulating Agents by Ott, Ingo, Kircher, Brigitte, Heinisch, Gottfried, Matuszczak, Barbara

“…Pyridazino[3,4-b][1,5]benzoxazepin-5(6H)ones substituted with propylene-linked basic side chains were synthesized and investigated for the ability to reverse…”
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Synthesis of novel phenylacetic acid derivatives with halogenated benzyl subunit and evaluation as aldose reductase inhibitors by Rakowitz, Dietmar, Gmeiner, Andreas, Schröder, Nicole, Matuszczak, Barbara

“…In the course of our ongoing studies several substituted benzyloxyphenylacetic acids were prepared. Comparison of their aldose reductase inhibition with the…”
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Linear and cyclicN-acyl-?-arylglycines III. Synthesis and chemiluminescence studies of naphthol and phenanthrol amidoalkylation products by Matuszczak, B.

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Pyrazolo[2′,3′:3,4][1,3]oxazino[5,6- b]quinoxaline, a novel tetracyclic ring system by Banekovich, Christian, Mereiter, Kurt, Matuszczak, Barbara

“…Reaction of 2-chloro-3-(3-chloro-1 H-pyrazol-5-yl)quinoxaline and aldehydes does not afford the corresponding N-(α-hydroxyalkylated) derivatives but results in…”
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Synthesis of Novel Benzoic Acid Derivatives with Benzothiazolyl Subunit and Evaluation as Aldose Reductase Inhibitors by Rakowitz, Dietmar, Hennig, Barbara, Nagano, Marietta, Steger, Stefan, Costantino, Luca, Matuszczak, Barbara

“…Several methyl benzothiazolyloxybenzoates, S‐isosters, and the corresponding benzoic acids were synthesized and tested as aldose reductase inhibitors (ARIs)…”
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Diazine-derived guanidines, isothioureas, and isoureas: Synthesis and attempts of configurational assignment by Heinisch, Gottfried, Matuszczak, Barbara, Rakowitz, Dietmar, Mereiter, Kurt

“…The utility of diazinyl substituted carbodiimides (1a‐c) for the synthesis of novel guanidines (2), isothioureas (3), and isoureas (4) is shown. Attempts to…”
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Pyridazines 91. Synthesis of substituted tri- and tetracyclic compounds bearing a pyridazine core and their biological evaluation as antimycobacterial agents by Heinisch, G, Matuszczak, B, Planitzer, K

“…Starting from substituted 3,6-dichloropyridazine-4-carboxamides (2, 3) tri- and tetracyclic compounds (4, 5) could be smoothly prepared. Structural…”
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On the prodrug potential of novel aldose reductase inhibitors with diphenylmethyleneaminooxycarboxylic acid structure by Rakowitz, Dietmar, Matuszczak, Barbara, Gritsch, Stefan, Hofbauer, Peter, Krassnigg, Andreas, Costantino, Luca

“…Diphenylmethyleneaminooxycarboxylic acids were found to represent novel type inhibitors of the enzyme aldose reductase. Ester derivatives of the most active…”
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Synthesis of Substituted Tri- and Tetracyclic Compounds Bearing a Pyridazine Core and their Biological Evaluation as Antimycobacterial Agents by Heinisch, Gottfried, Matuszczak, Barbara, Planitzer, Karin

“…Starting from substituted 3,6‐dichloropyridazine‐4‐carboxamides (2, 3) tri‐ and tetracyclic compounds (4, 5) could be smoothly prepared. Structural…”
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On the bioisosteric potential of the pyridazine core in the systematic structural modification of antiviral agents by Heinisch, G., Easmon, J., Matuszczak, B.

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Pyridazines. 84. Pyridazino[3,4-e]pyrido[3,2-b][1,4]diazepine, a novel tricyclic ring system by Heinisch, Gottfried, Matuszczak, Barbara

“…The preparation of pyridazino[3,4‐e]pyrido[3,2‐b][1,4]diazepin‐5‐ones 8 and 9 starting from appropriately substituted pyridazine‐4‐carboxamides is reported…”
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Pyridazines, 89. On the Synthesis of Novel 1,2-Diazine Containing Tricyclic Systems: Preparation of Dipyridazinodiazepinones by Matuszczak, Barbara, Heinisch, Gottfried, Huber, Elisabeth, Mereiter, Kurt

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Pyridazines 93. an unexpected reaction behaviour of 3-aminopyridazine towards 2-methylphenylisocyanate by Heinisch, Gottfried, Hetzenauer, Alfred, Matuszczak, Barbara, Rakowitz, Dietmar, Mereiter, Kurt

“…Reaction of 3‐aminopyridazine (1) with 2‐mefhylphenylisocyante (4) affords not only the desired urea derivative (5) but also an unexpected side‐product (6),…”
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Synthesis of N-aryl-N'-heteroaryl-substituted urea and thiourea derivatives and evaluation of their anticonvulsant activity by Heinisch, G, Matuszczak, B, Rakowitz, D, Tantisira, B

“…Starting from amino(di)azines and 2-chloro-6-methyliso(thio)cyanate a series of aryl-substituted urea and thiourea derivatives was prepared and screened as…”
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