Search Results - "Lusi, Aino"

Syntheses and biological activities of 13-substituted avermectin aglycons by Mrozik, Helmut, Linn, Bruce O, Eskola, Philip, Lusi, Aino, Matzuk, Alexander, Preiser, Franz A, Ostlind, Dan A, Schaeffer, James M, Fisher, Michael H

“…The reactions of sulfonate esters of the allylic/homoallylic 13-alcohol of 5-O-(tert-butyldimethylsilyl)-22,23-dihydroavermectin B1a aglycon (1a) were…”
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Ivermectin, a new broad-spectrum antiparasitic agent by Chabala, John C, Mrozik, Helmut, Tolman, Richard L, Eskola, Philip, Lusi, Aino, Peterson, Louis H, Woods, Mary F, Fisher, Michael H, Campbell, William C

“…22,23-Dihydroavermectin B1, ivermectin, derived from avermectin B1 by selective hydrogenation using Wilkinson's homogenous catalyst [Ph3P)3RhCl], was shown to…”
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4″-Deoxy-4″-aminoavermectins with potent broad spectrum antiparasitic activities by Mrozik, Helmut, Eskola, Philip, Arison, Byron H., Linn, Bruce O., Lusi, Aino, Matzuk, Alexander, Shih, Thomas L., Tischler, Maureen, Waksmunski, Frank S., Wyvratt, Matthew J., Blizzard, Timothy A., Margiatto, Gaye M., Fisher, Michael H., Shoop, Wesley L., Egerton, John R.

“…Reductive amination of 4″-oxo-5-O-tert-butyldimethylsilyl-avermectins with sodium cyanoborohydride and ammonium acetate gave an epimeric mixture of…”
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Synthesis of 5-Oxothiacyclöctane by Lusi, Aino

“…There are two fundamentally different approaches possible to arrive at cyclic medium-ring-sized ketones and acyloins• The basic ring structure may be arrived…”
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Imidazo[1,2-a]pyridine anthelmintic and antifungal agents by Fisher, Michael H, Lusi, Aino

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Anthelmintic dihydroquinoxalino[2,3-b]quinoxalines by Fisher, M H, Lusi, A, Egerton, J R

“…A series of dihydroquinoxalino[2,3-b]quinoxalines was synthesized and tested for anthelmintic activity in a model assay. The most promising compound,…”
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A TRANSANNULAR REACTION IN AN EIGHT-MEMBERED RING SULFIDE by Overberger, C. G, Lusi, Aino

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Synthesis of the New 5-Phosphomethyl-6-chromanyl Acetate of Vitamin K 1(20) by a Novel Cyclization Reaction by Wagner, Arthur F., Lusi, Aino, Erickson, Robert E., Arison, Byron, Trenner, Nelson R., Folkers, Karl

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Methyl 6-(phenylsulfinyl)imidazo[1,2-a]pyridine-2-carbamate, a potent, new anthelmintic by Bochis, Richard J, Dybas, Richard A, Eskola, Philip, Kulsa, Peter, Linn, Bruce O, Lusi, Aino, Meitzner, Eric P, Milkowski, John, Mrozik, Helmut

“…A series of methyl imidazo-[11,2-a]pyridine-2-carbamates was synthesized for anthelmintic testing. The preparation of this class of compounds was simplified by…”
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New Benzimidazoles and Novel Use of 2-Formylbenzimidazole in Syntheses by Wagner, Arthur F, Wittreich, Paul E, Lusi, Aino, Folkers, Karl

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4-Amino-6-(trichloroethenyl)-1,3-benzenedisulfonamide, a new, potent fasciolicide by Mrozik, Helmut, Bochis, Richard J, Eskola, Philip, Matzuk, Alexander, Waksmunski, Frank S, Olen, Leonard E, Schwartzkopf, George, Grodski, Alex, Linn, Bruce O

“…The synthesis and fasciolicidal activity of 4-amino-6-(trichloroethenyl)-1,3-benzenedisulfonamide are reported. A single dose of 15 mg/kg was effective in…”
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Reactions in Medium-sized Cyclic Sulfides by Overberger, C. G, Barkan, Paul, Lusi, Aino, Ringsdorf, Helmut

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Coenzyme Q. XLIII. The new 5-chloromethyl-6-chromanyl acetate of vitamin K-1(20) by WAGNER, A F, WITTREICH, P E, LUSI, A, ERICKSON, R E, ARISON, B, TRENNER, N R, FOLKERS, K

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Synthesis of the New 5-Phosphomethyl-6-chromanyl Acetate of Vitamin K1(20) by a Novel Cyclization Reaction by Wagner, Arthur F, Lusi, Aino, Erickson, Robert E, Arison, Byron, Trenner, Nelson R, Folkers, Karl

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Coenzyme Q. XLVII. New 5-Phosphomethyl-6-Chromanyl Derivatives from A Novel Reaction of Interest in Oxidative Phosphorylation by Wagner, Arthur F, Lusi, Aino, Shunk, Clifford H, Linn, Bruce O, Wolf, Donald E, Hoffman, Carl H, Erickson, Robert E, Arison, Byron, Trenner, Nelson R, Folkers, Karl

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