Search Results - "Lupattelli, P"

Synthesis of new methoxy derivatives of trans 2,3-diaryl-2,3-dihydrobenzofurans and evaluation of their anti-inflammatory activity by Laurita, T., Pappalardo, I., Chiummiento, L., D'Orsi, R., Funicello, M., Santarsiero, A., Marsico, M., Infantino, V., Todisco, S., Lupattelli, P.

“…[Display omitted] In the present study we synthesized new methoxy derivatives of trans 2,3-diaryl-2,3-dihydrobenzofurans, starting from suitable trans…”
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Synthesis and biological evaluation in vitro and in mammalian cells of new heteroaryl carboxyamides as HIV-protease inhibitors by Funicello, M., Chiummiento, L., Tramutola, F., Armentano, M.F., Bisaccia, F., Miglionico, R., Milella, L., Benedetti, F., Berti, F., Lupattelli, P.

“…[Display omitted] New heteroaryl HIV-protease inhibitors bearing a carboxyamide spacer were synthesized in few steps and high yield, from commercially…”
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Synthesis and biological evaluation of new simple indolic non peptidic HIV Protease inhibitors: The effect of different substitution patterns by Bonini, C., Chiummiento, L., Di Blasio, N., Funicello, M., Lupattelli, P., Tramutola, F., Berti, F., Ostric, A., Miertus, S., Frecer, V., Kong, D.-X.

“…New structurally simple indolic non peptidic HIV Protease inhibitors were synthesized from (S)-glycidol by regioselective methods. Following the concept of…”
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Asymmetric oxidation of silyl enol ethers using chiral dioxiranes derived from α-fluoro cyclohexanones by Solladié-Cavallo, A., Lupattelli, P., Jierry, L., Bovicelli, P., Angeli, F., Antonioletti, R., Klein, A.

“…Asymmetric oxidation of silyl enolethers derived from tetralone, 2-methyl-tetralone, propiophenone and deoxybenzoin using chiral dioxiranes generated in situ…”
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Isotactic polypropylene biodegradation by a microbial community: physicochemical characterization of metabolites produced by Cacciari, I, Quatrini, P, Zirletta, G, Mincione, E, Vinciguerra, V, Lupattelli, P, Giovannozzi Sermanni, G

“…From a selective enrichment culture prepared with different soil samples on starch-containing polyethylene we isolated four microaerophilic microbial…”
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anti Ethyl β-thienyl-β-amino-α-hydroxy propionate: a regio and stereoselective ring opening of trans ethyl 2-thienyl-glycidate by Solladié-Cavallo, A., Lupattelli, P., Bonini, C., De Bonis, M.

“…anti Ethyl β-thienyl-β-amino-α-hydroxy propionate was obtained regio- and diastereo-selectively in three steps and 45% overall yield, while 95% syn ethyl…”
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Synthesis Via Organoborates of (2E, 4Z)-1-Oxy-functionalized Dienes, Useful Intermediates of Natural and Bioactive Compounds by Bovicelli, P, Lupattelli, P, Mincione, E

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Synthesis, biological activity and modelling studies of two novel anti HIV PR inhibitors with a thiophene containing hydroxyethylamino core by Bonini, Carlo, Chiummiento, Lucia, Bonis, Margherita De, Funicello, Maria, Lupattelli, Paolo, Suanno, Gerardina, Berti, Federico, Campaner, Pietro

“…An efficient method has been developed for the synthesis of a versatile intermediate bearing azido, hydroxyl and ester functions, a useful precursor for…”
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Regio- and Stereoselective Ring Opening of 2,3-Diaryl Oxiranes by LiBr/Amberlyst 15:  A New Stereocontrolled Access to 1,2-Diaryl-2-bromo Alcohols by Solladié-Cavallo, Arlette, Lupattelli, Paolo, Bonini, Carlo

“…Both symmetrical and nonsymmetrical trans-2,3-diaryloxiranes are regio- and stereoselectively opened by the LiBr/Amberlyst 15 system. In the case of…”
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Single Route to Chiral syn- and anti-2-Amino-1,2-diphenylethanols via a New Stereodivergent Opening of trans-1,2-Diphenyloxirane by LUPATTELLI, Paolo, BONINI, Carlo, CARUSO, Leonilde, GAMBACORTA, Augusto

“…Oxiranyl ring opening of trans-stilbene oxide gave rise to anti- or syn-2-bromo-1,2-diphenylethanols, using either MgBr(2).Et(2)O or MgBr(2).Et(2)O, NaBr, and…”
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Cyclohexanones derived from dihydrocarvone as precursor of chiral dioxiranes for epoxidation of olefins by Solladié-Cavallo, Arlette, Jierry, Loïc, Lupattelli, Paolo, Bovicelli, Paolo, Antonioletti, Roberto

“…New ketones having an axial α-fluorine atom and substituents other than fluorine at C8, derived from commercially available (+)-dihydrocarvone, have been…”
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Synthesis of a first thiophene containing analog of the HIV protease inhibitor nelfinavir by Bonini, Carlo, Chiummiento, Lucia, De Bonis, Margherita, Funicello, Maria, Lupattelli, Paolo

“…A stereoselective and efficient preparation of a thiophene containing intermediate 2 from ethyl 3-thienyl propenoate 4 as the core of new possible HIV protease…”
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Oxidation of 3-arylisochromans by dimethyldioxirane. An easy route to substituted 3-arylisocoumarins by Bovicelli, Paolo, Lupattelli, Paolo, Crescenzi, Benedetta, Sanetti, Anna, Bernini, Roberta

“…The selective oxidation of the two different benzylethereal position of 3-arylisochromans by dimethyldioxirane as a function of different substituents on the…”
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Opening of Diaryl Epoxides: ortho-Fluorophenyl and 2-Pyridyl Epoxides by Solladié-Cavallo, Arlette, Lupattelli, Paolo, Marsol, Claire, Isarno, Thomas, Bonini, Carlo, Caruso, Leonilde, Maiorella, Angelica

“…Opening of epoxides with LiAlH4, MgBr2·2OEt2 (solution in Et2O), MgBr2·OEt2 (suspension in Et2O), and NaBr/Amberlyst‐15 has been studied. While 2‐pyridyl…”
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Oxyfunctionalisation of activated methylenes by dimethyldioxirane: An easy conversion of isochromans into isocoumarins by Bovicelli, Paolo, Sanetti, Anna, Bernini, Roberta, Lupattelli, Paolo

“…the concerted activating effect of two groups allowed the oxidation of methylene carbons, otherwise almost inert, by dimethyldioxirane. The method permitted an…”
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Improved procedure for 3,4-dihydro-1H-2-benzopyran ring closure. A general access to 3-substituted isochromanes by Antonioletti, Roberto, Bovicelli, Paolo, Crescenzi, Benedetta, Lupattelli, Paolo

“…A general method for the ring closure of 1-substituted 2-(-hydroxymethyl)-phenylethanols to 3-substituted isochromanes using p-TsOH supported on silica gel is…”
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Regioselective oxidation of azidodiols, bromodiols and triol derivatives by dimethyldioxirane by Bovicelli, Paolo, Truppa, Danilo, Sanetti, Anna, Bernini, Roberta, Lupattelli, Paolo

“…Azidodiols, bromodiols and triol derivatives were regioselectively monooxidised to the corresponding ketols using dimethyldioxirane. This regioselectivity is…”
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Fine regioselective tuning in the oxidation of sec,sec 1,2-diols by dimethyldioxirane by Bovicelli, Paolo, Sanetti, Anna, Lupattelli, Paolo

“…Non symmetric sec,sec 1.2-diols and their O-isopropylidene derivatives undergo a regioselective oxidation by dimethyldioxirane depending on the electronic…”
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An efficient oxyfunctionalisation by dimethyldioxirane of the benzylethereal carbon of flavonoids; a general and useful way to anthocyanidins by Bernini, Roberta, Mincione, Enrico, Sanetti, Anna, Bovicelli, Paolo, Lupattelli, Paolo

“…compounds with flavonoid structure were selectively oxyfunctionalised at the C-2 carbon atom by DMD. The reaction permitted a new route to flavylium salts…”
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Regio- and Stereoselective Epoxidation of Steroidal 1,4-Diene 3-Ones by Dimethyldioxirane: A New Access to A-Norsteroids and to a Class of Estrogen Synthetase Inhibitors by Bovicelli, Paolo, Lupattelli, Paolo, Mincione, Enrico

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