Search Results - "Lubos, Marta"

A viral insulin-like peptide inhibits IGF-1 receptor phosphorylation and regulates IGF1R gene expression by Chrudinová, Martina, Kirk, Nicholas S., Chuard, Aurelien, Venugopal, Hari, Zhang, Fa, Lubos, Marta, Gelfanov, Vasily, Páníková, Terezie, Žáková, Lenka, Cutone, Julianne, Mojares, Matthew, DiMarchi, Richard, Jiráček, Jiří, Altindis, Emrah

“…The insulin/IGF superfamily is conserved across vertebrates and invertebrates. Our team has identified five viruses containing genes encoding viral…”
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Inhibition of human and yeast 20S proteasome by analogues of trypsin inhibitor SFTI-1 by Dębowski, Dawid, Pikuła, Michał, Lubos, Marta, Langa, Paulina, Trzonkowski, Piotr, Lesner, Adam, Łęgowska, Anna, Rolka, Krzysztof

“…Starting from the primary structure of sunflower trypsin inhibitor SFTI-1, we designed novel non-covalent inhibitors of human and yeast 20S proteasomes…”
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Functional stapled fragments of human preptin of minimised length by Lubos, Marta, Mrázková, Lucie, Gwozdiaková, Petra, Pícha, Jan, Buděšínský, Miloš, Jiráček, Jiří, Kaminský, Jakub, Žáková, Lenka

“…Preptin is a 34-amino-acid-long peptide derived from the E-domain of a precursor of insulin-like growth factor 2 (pro-IGF2) with bone-anabolic and insulin…”
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Combinatorial Libraries of Bipodal Binders of the Insulin Receptor by Selicharová, Irena, Fabre, Benjamin, Soledad Garre Hernández, María, Lubos, Marta, Pícha, Jan, Voburka, Zdeněk, Mitrová, Katarína, Jiráček, Jiří

“…The binding process of insulin to its transmembrane receptor entails a sophisticated interplay between two proteins, each possessing two binding sites. Given…”
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The final walk with preptin by Mrázková, Lucie, Lubos, Marta, Voldřich, Jan, Kužmová, Erika, Zrubecká, Denisa, Gwozdiaková, Petra, Buděšínský, Miloš, Asai, Seiya, Marek, Aleš, Pícha, Jan, Tencerová, Michaela, Ferenčáková, Michaela, Barrera, Glenda Alquicer, Kaminský, Jakub, Jiráček, Jiří, Žáková, Lenka

“…Preptin, a 34-amino acid peptide derived from pro-IGF2, is believed to influence various physiological processes, including insulin secretion and the…”
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Modulation of the antagonistic properties of an insulin mimetic peptide by disulfide bridge modifications by Lubos, Marta, Pícha, Jan, Selicharová, Irena, Žák, Jíří, Buděšínský, Miloš, Mitrová, Katarína, Žáková, Lenka, Jiráček, Jiří

“…Insulin is a peptide responsible for regulating the metabolic homeostasis of the organism; it elicits its effects through binding to the transmembrane insulin…”
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Interactions between trypsin and its peptidic inhibitors studied by isothermal titration calorimetry (ITC) by Dębowski, Dawid, Wyrzykowski, Dariusz, Lubos, Marta, Rolka, Krzysztof

“…Isothermal titration calorimetry (ITC) technique was used to study the interactions of trypsin with bicyclic sunflower-derived trypsin inhibitor (SFTI-1) as…”
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Noncovalent inhibitors of human 20S and 26S proteasome based on trypsin inhibitor SFTI-1 by Dębowski, Dawid, Cichorek, Mirosława, Lubos, Marta, Wójcik, Sławomir, Łęgowska, Anna, Rolka, Krzysztof

“…Sunflower trypsin inhibitor (SFTI‐1) is recognized as an attractive scaffold to designed potent inhibitors of various proteases. We have recently found that…”
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Multipodal insulin mimetics built on adamantane or proline scaffolds by Hajduch, Jan, Fabre, Benjamin, Klopp, Benjamin, Pohl, Radek, Buděšínský, Miloš, Šolínová, Veronika, Kašička, Václav, Köprülüoglu, Cemal, Eyrilmez, Saltuk Mustafa, Lepšík, Martin, Hobza, Pavel, Mitrová, Katarína, Lubos, Marta, Hernández, María Soledad Garre, Jiráček, Jiří

“…[Display omitted] •Insulin mimetics could represent an alternative strategy for treatment of diabetes.•Multipodal compounds based on adamantane or proline…”
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Inhibition of human constitutive 20S proteasome and 20S immunoproteasome with novel N‐terminally modified peptide aldehydes and their antitumor activity by Lubos, Marta, Dębowski, Dawid, Barcińska, Ewelina, Meid, Annika, Inkielewicz‐Stepniak, Iwona, Burster, Timo, Rolka, Krzysztof

“…The conversion of primary structures of novel, highly selective and sensitive, internally quenched peptide substrates of the human 20S proteasome into peptide…”
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