Search Results - "Lu, Ai‐Min"

An Enzymatic N‐Acylation Step Enables the Biocatalytic Synthesis of Unnatural Sialosides by Laborda, Pedro, Lyu, Yong‐Mei, Parmeggiani, Fabio, Lu, Ai‐Min, Wang, Wen‐Jiao, Huang, Ying‐Ying, Huang, Kun, Guo, Juan, Liu, Li, Flitsch, Sabine L., Voglmeir, Josef

“…Chitin is one of the most abundant and cheaply available biopolymers in Nature. Chitin has become a valuable starting material for many biotechnological…”
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Diastereoselective One‐Step Synthesis of 2‐Keto‐3‐deoxy‐d‐ glycero‐d‐galacto‐nononic acid (KDN) Analogues as Templates for the Development of Influenza Drugs by Laborda, Pedro, Wang, Su‐Yan, Lu, Ai‐Min, He, Meng, Duan, Xu‐Chu, Qian, Ying‐Juan, Jung, Yong‐Sam, Liu, Li, Voglmeir, Josef

“…Novel sialic acid scaffolds have great significance in the development of influenza neuraminidase inhibitors. Here the enzymatic synthesis of a wide range of…”
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Biocatalytic β-glucosylation/β-galactosylation of Rebaudioside C by glycosynthases by Yu, Ye-Yang, Zhang, Si-Yu, Sun, Jia-Hui, Li, Yu-Yang, Zhang, Yao-Yao, Lu, Ai-Min, Liu, Li, Voglmeir, Josef

“…Extracts of Stevia rebaudiana Bertoni plant leaves contain a mixture of diterpene glycosides which possess high sweetness and are used as non-caloric…”
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Synthesis, Characterization, and Antifungal Activity of Phenylpyrrole-Substituted Tetramic Acids Bearing Carbonates by Xu, Wen-Qin, Chen, Min, Wang, Kun-Yao, Ren, Zheng-Jiao, Lu, Ai-Min, Yang, Chun-Long

“…For the aim of discovering new fungicide, a series of phenylpyrrole-substituted tetramic acid derivatives bearing carbonates 6a-q were designed and synthesized…”
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Synthesis and fungicidal activity of phenylhydrazone derivatives containing two carbonic acid ester groups by Wang, Jun-Jun, Si, Wei-Jie, Chen, Min, Lu, Ai-Min, Zhang, Wei-Hua, Yang, Chun-Long

“…Substituted phenylhydrazone moieties and two carbonate groups were merged in one molecule scaffold to obtain 48 novel compounds. 1H and 13C NMR, MS, elemental…”
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N-acetylglucosamine 2-Epimerase from Pedobacter heparinus: First Experimental Evidence of a Deprotonation/Reprotonation Mechanism by Su-Yan Wang, Pedro Laborda, Ai-Min Lu, Xu-Chu Duan, Hong-Yu Ma, Li Liu, Josef Voglmeir

“…The control of cellular N-acetylmannosamine (ManNAc) levels has been postulated to be an effective way to modulate the decoration of cell surfaces with sialic…”
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Imidazolium labelling permits the sensitive mass-spectrometric detection of N -glycosides directly from serum by Zhang, Yao-Yao, Ghirardello, Mattia, Wang, Ting, Lu, Ai-Min, Liu, Li, Voglmeir, Josef, Galan, M Carmen

“…A novel imidazolium derivative (GITag) shows superior ionisation and consequently allows increased mass spectrometric detection capabilities of…”
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α‑Allenyl Ethers as Starting Materials for Palladium Catalyzed Suzuki–Miyaura Couplings of Allenylphosphine Oxides with Arylboronic Acids by Chen, Yao-Zhong, Zhang, Ling, Lu, Ai-Min, Yang, Fang, Wu, Lei

“…We disclose here the first palladium-catalyzed Suzuki–Miyaura couplings of aryl ethers functionalized allenylphosphine oxides with arylboronic acids. This new…”
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Potential Succinate Dehydrogenase Inhibitors Bearing a Novel Pyrazole-4-sulfonohydrazide Scaffold: Molecular Design, Antifungal Evaluation, and Action Mechanism by Chai, Jian-Qi, Mei, Yu-Dong, Tai, Lang, Wang, Xiao-Bin, Chen, Min, Kong, Xiang-Yi, Lu, Ai-Min, Li, Guo-Hua, Yang, Chun-Long

“…Aiming to develop novel antifungal agents with a distinctive molecular scaffold targeting succinate dehydrogenase (SDH), 24…”
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Design, Synthesis, Antifungal, and Antioxidant Activities of (E)‑6-((2-Phenylhydrazono)methyl)quinoxaline Derivatives by Zhang, Mao, Dai, Zhi-Cheng, Qian, Shao-Song, Liu, Jun-Yan, Xiao, Yu, Lu, Ai-Min, Zhu, Hai-Liang, Wang, Jian-Xin, Ye, Yong-Hao

“…Different substituted phenylhydrazone groups were linked to the quinoxaline scaffold to provide 26 compounds (6a–6z). Their structures were confirmed by 1H and…”
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2種類の炭酸エステル基を有するフェニルヒドラゾン誘導体の合成及び抗菌活性

“…2位と6位に2つの炭酸エステル基を有するアセトフェノンと置換フェニルヒドラゾンの縮合により新規な置換フェニルヒドラゾン化合物48個を合成した．1Hおよび13C NMR, MS，元素分析とX線単結晶回折により，それらの構造を確認した．バイオアッセイの結果，Botrytis cinerea, Rhizoctonia…”
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Synthesis and antifungal activity of novel amide derivatives from quinic acid against the sweet potato pathogen Ceratocystis fimbriata by Jiang, Yong‐Hui, Shi, Xin‐Chi, Wu, Ting, Du, Hao, Pang, Yi‐Bo, Zhou, Rong, Yin, Hong‐Ping, Herrera‐Balandrano, Daniela D, Yang, Dong‐Jing, Lu, Ai‐Min, Laborda, Pedro, Polo, Victor, Wang, Su‐Yan

“…Abstract BACKGROUND Ceratocystis fimbriata is a fungal pathogen that infects sweet potato roots, producing enormous economic losses. Cyclic polyhydroxy…”
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Design, synthesis and herbicidal activity of novel cyclohexanedione derivations containing pyrazole and pyridine groups as potential HPPD inhibitors by Hou, Shuai-Tao, Han, Ling, Li, Wen-Rui, Dai, Guang-Yu, Liu, Yu, Lu, Ai-Min, Yang, Chun-Long, Chen, Min

“…4-Hydroxyphenylpyruvate dioxygenase (EC 1.13.11.27; HPPD) is one of the important target enzymes in the development of herbicides. To discover novel HPPD…”
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QSAR studies of phenylhydrazine-substituted tetronic acid derivatives based on the 1 H NMR and 13 C NMR chemical shifts by Chen, Min, Lu, Ai-Min, Hu, Ying, Yang, Chun-Long

“…The quantitative structure-activity relationship models of 40 phenylhydrazine-substituted tetronic acid derivatives were established between the H nuclear…”
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QSAR studies of phenylhydrazine‐substituted tetronic acid derivatives based on the 1H NMR and 13C NMR chemical shifts by Chen, Min, Lu, Ai‐Min, Hu, Ying, Yang, Chun‐Long

“…The quantitative structure–activity relationship models of 40 phenylhydrazine‐substituted tetronic acid derivatives were established between the 1H nuclear…”
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Synthesis, biological evaluation and 3D-QSAR study of novel 4,5-dihydro-1H-pyrazole thiazole derivatives as BRAF(V⁶⁰⁰E) inhibitors by Zhao, Meng-Yue, Yin, Yong, Yu, Xiao-Wei, Sangani, Chetan B, Wang, Shu-Fu, Lu, Ai-Min, Yang, Li-Fang, Lv, Peng-Cheng, Jiang, Ming-Guo, Zhu, Hai-Liang

“…Many reports implied that the BRAF serine/threonine kinase was mutated in various types of human tumors, which were related with cell growth, survival and…”
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Metal-free synthesis of chlorinated and brominated phosphinoyl 1,3-butadiene derivatives and its synthetic applications by Liu, Teng, Xia, Yun-Tao, Zhu, Jie, Lu, Ai-Min, Wu, Lei

“…[Display omitted] We report here an efficient and transition-metal free strategy for the synthesis of chlorinated and brominated phosphinoyl 1,3-butadienes and…”
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Design, synthesis, and antifungal activity of novel cyanoacrylate derivatives containing a naphthalene moiety as potential myosin-5 inhibitor by Jin, Fei, Peng, Feng, Li, Wen-Rui, Chai, Jian-Qi, Chen, Min, Lu, Ai-Min, Yang, Chun-Long, Zhou, Ming-Guo

“…In search of innovative antifungal solutions for the control of plant diseases, a series of cyanoacrylate derivatives containing naphthalene groups were…”
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6,7-Dihydrobenzo[f]benzo[4,5]imidazo[1,2-d][1,4]oxazepine derivatives as selective inhibitors of PI3Kα by Yin, Yong, Zhang, Yan-Qing, Jin, Biao, Sha, Shao, Wu, Xun, Sangani, Chetan B., Wang, She-Feng, Qiao, Fang, Lu, Ai-Min, Lv, Peng-Cheng, Zhu, Hai-Liang

“…Twenty eight new 6,7-dihydrobenzo[f]benzo[4,5]imidazo[1,2-d][1,4]oxazepine derivatives have been synthesized and evaluated for biological activities as PI3Kα…”
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Access to Cyano-Containing Isoxazolines via Copper-Catalyzed Domino Cyclization/Cyanation of Alkenyl Oximes by Meng, Fei, Zhang, Honglin, Guo, Kang, Dong, Jiayue, Lu, Ai-Min, Zhu, Yingguang

“…A highly efficient copper-catalyzed cyclization/cyanation cascade of unactivated olefins bearing oximes is described. A variety of cyano-containing…”
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