Search Results - "Locco, L"

6H-Benzo[c]chromen-6-one derivatives as selective ERβ agonists by Sun, Wanying, Cama, Lovji D., Birzin, Elizabeth T., Warrier, Sudha, Locco, Louis, Mosley, Ralph, Hammond, Milton L., Rohrer, Susan P.

“…A series of 6H-benzo[c]chromen-6-one and 6H-benzo[c]chromene derivatives were prepared. Many of the analogs were found to be potent and selective ERβ agonists…”
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The discovery of tetrahydrofluorenones as a new class of estrogen receptor β-subtype selective ligands by Wilkening, R.R., Ratcliffe, R.W., Tynebor, E.C., Wildonger, K.J., Fried, A.K., Hammond, M.L., Mosley, R.T., Fitzgerald, P.M.D., Sharma, N., McKeever, B.M., Nilsson, S., Carlquist, M., Thorsell, A., Locco, L., Katz, R., Frisch, K., Birzin, E.T., Wilkinson, H.A., Mitra, S., Cai, S., Hayes, E.C., Schaeffer, J.M., Rohrer, S.P.

“…Synthesis and derivatization of a series of substituted tetrahydrofluorenone analogs giving potent, ERβ subtype-selective ligands are described. Synthesis and…”
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Endogenous syntaxins 2, 3 and 4 exhibit distinct but overlapping patterns of expression at the hepatocyte plasma membrane by Fujita, H, Tuma, P L, Finnegan, C M, Locco, L, Hubbard, A L

“…To investigate the mechanisms regulating polarized vesicle delivery to the cell surface in hepatocytes, we have characterized the endogenous plasma membrane…”
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Modeling directed design and biological evaluation of quinazolinones as non-peptidic growth hormone secretagogues by ZHIXIONG YE, YINGDUO GAO, LOCCO, L, PARMAR, R. M, CHAN, W. W.-S, SCHAEFFER, J. M, SMITH, R. G, PATCHETT, A. A, NARGUND, R. P, BAKSHI, R. K, CHEN, M.-H, ROHRER, S. P, FEIGHNER, S. D, PONG, S.-S, HOWARD, A. D, BLAKE, A, BIRZIN, E. T

“…Quinazolinone derivatives were synthesized and evaluated as non-peptidic growth hormone secretagogues. Modeling guided design of quinazolinone compound 21 led…”
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