Search Results - "Li, Tiechao"

Aryl[a]pyrrolo[3,4-c]carbazoles as selective cyclin D1-CDK4 inhibitors by SANCHEZ-MARTINEZ, Concha, SHIH, Chuan, BROOKS, Harold B, PATEL, Bharvin K. R, SCHULTZ, Richard M, DEHAHN, Tammy B, SPENCER, Charles D, WATKINS, Scott A, CONSIDINE, Eileen, DEMPSEY, Jack A, OGG, Catherine A, CAMPBELL, Robert M, FAUL, Margaret M, ANDERSON, Bryan A, WAGNER, Jill, GUOXIN ZHU, PAAL, Michael, SOMOZA, Carmen, TIECHAO LI, KUMRICH, Christine A, WINNEROSKI, Leonard L, ZHOU XUN

“…The synthesis of new analogues of Arcyriaflavin A in which one indole ring is replaced by an aryl or heteroaryl ring is described. These new series of…”
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Novel 1,3-disubstituted-5, 10-dihydro-5, 10-dioxo-1H-benzo[g] isochromene-3 carboxamides as potent antitumor agents by WUYI WANG, TIECHAO LI, MILBURN, R, YATES, J, HINNANT, E, LUZZIO, M. J, NOBLE, S. A, ATTARDO, G

“…Novel antitumor 5,10-dihydro-5,10-dioxo-1H- benzo[g]isochromene-3-carboxamides were discovered…”
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Synthesis, Structure−Activity Relationship, and Biological Studies of Indolocarbazoles as Potent Cyclin D1-CDK4 Inhibitors by Zhu, Guoxin, Conner, Scott E, Zhou, Xun, Shih, Chuan, Li, Tiechao, Anderson, Bryan D, Brooks, Harold B, Campbell, Robert Morris, Considine, Eileen, Dempsey, Jack A, Faul, Margaret M, Ogg, Cathy, Patel, Bharvin, Schultz, Richard M, Spencer, Charles D, Teicher, Beverly, Watkins, Scott A

“…Novel substituted indolocarbazoles were synthesized, and their kinase inhibitory capability was evaluated in vitro. 6-Substituted indolocarbazoles 4 were found…”
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Acyl Sulfonamide Anti-Proliferatives:  Benzene Substituent Structure−Activity Relationships for a Novel Class of Antitumor Agents by Lobb, Karen L, Hipskind, Philip A, Aikins, James A, Alvarez, Enrique, Cheung, Yiu-Yin, Considine, Eileen L, De Dios, Alfonso, Durst, Gregory L, Ferritto, Rafael, Grossman, Cora Sue, Giera, Deborah D, Hollister, Beth A, Huang, Zhongping, Iversen, Philip W, Law, Kevin L, Li, Tiechao, Lin, Ho-Shen, Lopez, Beatriz, Lopez, Jose E, Cabrejas, Luisa M. Martin, McCann, Denis J, Molero, Victoriano, Reilly, John E, Richett, Michael E, Shih, Chuan, Teicher, Beverly, Wikel, James H, White, Wesley T, Mader, Mary M

“…Two closely related diaryl acylsulfonamides were recently reported as potent antitumor agents against a broad spectrum of human tumor xenografts (colon, lung,…”
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Imidazolyl benzimidazoles and imidazo[4,5- b]pyridines as potent p38α MAP kinase inhibitors with excellent in vivo antiinflammatory properties by Mader, Mary, de Dios, Alfonso, Shih, Chuan, Bonjouklian, Rosanne, Li, Tiechao, White, Wesley, de Uralde, Beatriz López, Sánchez-Martinez, Concepción, del Prado, Miriam, Jaramillo, Carlos, de Diego, Eugenio, Martín Cabrejas, Luisa M., Dominguez, Carmen, Montero, Carlos, Shepherd, Timothy, Dally, Robert, Toth, John E., Chatterjee, Arindam, Pleite, Sehila, Blanco-Urgoiti, Jaime, Perez, Leticia, Barberis, Mario, Lorite, María José, Jambrina, Enrique, Nevill, C. Richard, Lee, Paul A., Schultz, Richard C., Wolos, Jeffrey A., Li, Li C., Campbell, Robert M., Anderson, Bryan D.

“…The p38 MAP kinase activity of two series of trisubstituted imidazoles (X = C, N) is reported, leading to compounds with highly potent cellular and in vivo…”
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Studies on cyclin-dependent kinase inhibitors: Indolo-[2,3-a]pyrrolo[3,4-c]carbazoles versus bis-indolylmaleimides by SANCHEZ-MARTINEZ, Concha, CHUAN SHIH, OGG, Catherine A, CONSIDINE, Eileen, DEMPSEY, Jack A, FAMING ZHANG, GUOXIN ZHU, TIECHAO LI, BROOKS, Harold B, PATEL, Bharvin K. R, SCHULTZ, Richard M, DEHAHN, Tammy B, SPENCER, Charles D, WATKINS, Scott A

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Studies on cyclin-dependent kinase inhibitors: indolo-[2,3-a]pyrrolo[3,4-c]carbazoles versus bis-indolylmaleimides by Sanchez-Martinez, Concha, Shih, Chuan, Zhu, Guoxin, Li, Tiechao, Brooks, Harold B, Patel, Bharvin K R, Schultz, Richard M, DeHahn, Tammy B, Spencer, Charles D, Watkins, Scott A, Ogg, Catherine A, Considine, Eileen, Dempsey, Jack A, Zhang, Faming

“…A series of indolo[2,3-a]pyrrolo[3,4-c]carbazoles and their bis-indolylmaleimides precursors have been prepared in order to compare their activity as D1-CDK4…”
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Synthetic Study of Selective Benzylic Oxidation by Wang, Wuyi, Li, Tiechao, Attardo, Giorgio

“…Oxidation of bisbenzyl ethers was studied using 2,3-dichloro-5,6-dicyanobenzoquinone (DDQ). Compared to other benzylic oxidations such as Kornblum type…”
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Dehydrogenation by air: Preparation of 1,3-disubstituted-5,1-dioxo-5,10-dihydro-1H-benzo[g] isochromene scaffold by Wang, Wuyi, Breining, Tibor, Li, Tiechao, Milburn, Robert, Attardo, Giorgio

“…Naphthaquinopyrans 5a-d, 10 and 12 have been converted to benzoisochromene IIb via base-promoted air oxidation. A mechanism is proposed to account for the…”
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Phototoxicity of some bromine-substituted rhodamine dyes: synthesis, photophysical properties and application as photosensitizers by Pal, P, Zeng, H, Durocher, G, Girard, D, Li, T, Gupta, A K, Giasson, R, Blanchard, L, Gaboury, L, Balassy, A, Turmel, C, Laperrière, A, Villeneuve, L

“…The synthesis of some bromine-substituted rhodamine derivatives viz., 4,5-dibromorhodamine methyl ester (dye 2) and 4,5-dibromorhodamine n-butyl ester (dye 3)…”
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Synthesis and Characterization of Functionalized Analogs of 1,3,6,8-Tetrakis(methylsulfanyl)pyrene and Their Electron-Conducting Radical-Cation Salts by Li, Tiechao, Giasson, Richard

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Novel 1,3-disubstituted-5,10-dihydro-5,10-dioxo-1H-mbenzo[g]isochromene-3-carboxamides as potent antitumor agents by Wang, Wuyi, Li, Tiechao, Milburn, Robert, Yates, J., Hinnant, E., Luzzio, Micheal J., Noble, Stuart A., Attardo, Giorgio

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Imidazolyl benzimidazoles and imidazo[4,5-b]pyridines as potent p38alpha MAP kinase inhibitors with excellent in vivo antiinflammatory properties by Mader, Mary, de Dios, Alfonso, Shih, Chuan, Bonjouklian, Rosanne, Li, Tiechao, White, Wesley, López de Uralde, Beatriz, Sánchez-Martinez, Concepción, del Prado, Miriam, Jaramillo, Carlos, de Diego, Eugenio, Martín Cabrejas, Luisa M, Dominguez, Carmen, Montero, Carlos, Shepherd, Timothy, Dally, Robert, Toth, John E, Chatterjee, Arindam, Pleite, Sehila, Blanco-Urgoiti, Jaime, Perez, Leticia, Barberis, Mario, Lorite, María José, Jambrina, Enrique, Nevill, Jr, C Richard, Lee, Paul A, Schultz, Richard C, Wolos, Jeffrey A, Li, Li C, Campbell, Robert M, Anderson, Bryan D

“…Herein we report investigations into the p38alpha MAP kinase activity of trisubstituted imidazoles that led to the identification of compounds possessing…”
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Novel 1,3-disubstituted-5,10-dihydro-5,10-dioxo-1 H-mbenzo[ g]isochromene-3-carboxamides as potent antitumor agents by Wang, Wuyi, Li, Tiechao, Milburn, Robert, Yates, J., Hinnant, E., Luzzio, Micheal J., Noble, Stuart A., Attardo, Giorgio

“…Novel antitumor 5,10-dihydro-5,10-dioxo-1 H-benzo[ g]isochromene-3-carboxamides were discovered. Novel antitumor 5,10-dihydro-5,10-dioxo-1 H-benzo[…”
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