Search Results - "Lenaerts, Anne J.M."

Discovery of novel isoxazolines as anti-tuberculosis agents by Tangallapally, Rajendra P., Sun, Dianqing, Rakesh, Budha, Nageshwar, Lee, Robin E.B., Lenaerts, Anne J.M., Meibohm, Bernd, Lee, Richard E.

“…Discovery of isoxazoline compound 12 as novel anti-tuberculosis agent (MIC 90 = 1.56 μg/mL) is reported. Nitrofuranyl isoxazolines with increased proteolytic…”
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Synthesis and Evaluation of Cyclic Secondary Amine Substituted Phenyl and Benzyl Nitrofuranyl Amides as Novel Antituberculosis Agents by Tangallapally, Rajendra P, Yendapally, Raghunandan, Lee, Robin E, Lenaerts, Anne J. M, Lee, Richard E

“…In an ongoing effort to develop new and potent antituberculosis agents, a second-generation series of nitrofuranyl amides was synthesized on the basis of the…”
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Synthesis and Evaluation of Nitrofuranylamides as Novel Antituberculosis Agents by Tangallapally, Rajendra P, Yendapally, Raghunandan, Lee, Robin E, Hevener, Kirk, Jones, Victoria C, Lenaerts, Anne J. M, McNeil, Michael R, Wang, Yuehong, Franzblau, Scott, Lee, Richard E

“…In an effort to develop new and more potent therapies to treat tuberculosis, a library of compounds was screened for M. tuberculosis UDP-Gal mutase inhibition…”
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Rapid In Vivo Screening of Experimental Drugs for Tuberculosis Using Gamma Interferon Gene-Disrupted Mice by LENAERTS, Anne J. M, GRUPPO, Veronica, BROOKS, Jason V, ORME, Ian M

“…Classifications Services AAC Citing Articles Google Scholar PubMed Related Content Social Bookmarking CiteULike Delicious Digg Facebook Google+ Mendeley Reddit…”
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Synthesis of new and potent analogues of anti-tuberculosis agent 5-nitro-furan-2-carboxylic acid 4-(4-benzyl-piperazin-1-yl)-benzylamide with improved bioavailability by Tangallapally, Rajendra P., Lee, Robin E.B., Lenaerts, Anne J.M., Lee, Richard E.

“…The synthesis of lead optimized analogues, their anti-tuberculosis activity, and bioavailability are reported. Previously, the lead compound…”
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