Search Results - "Lazaro, Horacio"

Microwave synthesis of 1-aryl-1H-pyrazole-5-amines by Everson, Nikalet, Yniguez, Kenya, Loop, Lauren, Lazaro, Horacio, Belanger, Briana, Koch, Grant, Bach, Jordan, Manjunath, Aashrita, Schioldager, Ryan, Law, Jarvis, Grabenauer, Megan, Eagon, Scott

“…[Display omitted] •Pyrazole-5-amines appear in molecules with a diverse range of activities.•A microwave-mediated method was developed to produce products in…”
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Microwave mediated synthesis of 2-aminooxazoles by Klug, Trevan, Cronin, Adam, O'Brien, Eli, Schioldager, Ryan, Johnson, Hunter, Gleason, Cameron, Schmid, Connor, Soderberg, Nathan, Manjunath, Aashrita, Liyanage, Duminda, Lazaro, Horacio, Kimball, Joshua J., Eagon, Scott

“…[Display omitted] A microwave mediated synthesis of 2-aminooxazoles at 150 °C was developed, providing products with a variety of functional groups. The…”
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Synthesis and activity of β-carboline antimalarials targeting the Plasmodium falciparum heat shock 90 protein by Viswanathan, Neil K., Chirgwin, Michael E., Gibbs, Julia, Kalaj, Brianna N., Durham, Sierra, Tran, Jennifer, Gomez, Maximillian, Lazaro, Horacio, Chen, Ming, Mansfield, Christopher R., Derbyshire, Emily R., Eagon, Scott

“…[Display omitted] A collection of β-carbolines based on the natural product harmine, a compound known to target the heat shock 90 protein of Plasmodium…”
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Synthesis of benzoxazoles via a silver mediated oxidation by Wong, Chloe D., Ganjooi, Kimiya, Verbarendse, Maetja, Travis, Jessica M., Troftgruben, Mark H. S., Mora, Hannah R., Oldenburg, Isabella, Lammert, Robert, Lazaro, Horacio, Eagon, Scott

“…A silver carbonate-based method to synthesize benzoxazoles from imines has been developed. The reaction is extremely mild, tolerates several heterocycles and…”
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Antimalarial activity of tetrahydro-β-carbolines targeting the ATP binding pocket of the Plasmodium falciparum heat shock 90 protein by Eagon, Scott, Hammill, Jared T., Bach, Jordan, Everson, Nikalet, Sisley, Tyler A., Walls, Michael J., Durham, Sierra, Pillai, Dylan R., Falade, Mofolusho O., Rice, Amy L., Kimball, Joshua J., Lazaro, Horacio, DiBernardo, Celine, Kiplin Guy, R.

“…[Display omitted] •The natural product harmine is known to have antimalarial activity.•We report a new series of harmine derivatives that show improved…”
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Synthesis and Structure–Activity Relationship of Dual-Stage Antimalarial Pyrazolo[3,4‑b]pyridines by Eagon, Scott, Hammill, Jared T, Sigal, Martina, Ahn, Kevin J, Tryhorn, Julia E, Koch, Grant, Belanger, Briana, Chaplan, Cory A, Loop, Lauren, Kashtanova, Anna S, Yniguez, Kenya, Lazaro, Horacio, Wilkinson, Steven P, Rice, Amy L, Falade, Mofolusho O, Takahashi, Rei, Kim, Katie, Cheung, Ashley, DiBernardo, Celine, Kimball, Joshua J, Winzeler, Elizabeth A, Eribez, Korina, Mittal, Nimisha, Gamo, Francisco-Javier, Crespo, Benigno, Churchyard, Alisje, García-Barbazán, Irene, Baum, Jake, Anderson, Marc O, Laleu, Benoît, Guy, R. Kiplin

“…Malaria remains one of the most deadly infectious diseases, causing hundreds of thousands of deaths each year, primarily in young children and pregnant…”
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