Search Results - "LORENZI, Simone"

MUST dome design based on dome seeing quantitative evaluation by Zhang, Yuchen, Lao, Junsen, Wang, Zhuoxiao, Cai, Zheng, Guo, Liquan, Bian, Qi, Zheng, Yamin, Zhuang, Yongchen, Zhang, Yifan, Li, Pei, Wang, Zichao, Dai, Xiaodong, Lu, Lu, Marchiori, Gianpietro, De Lorenzi, Simone, Huang, Lei

“…ABSTRACT The Multiplexed Survey Telescope (MUST) project is led by Tsinghua University, which entrusted the European Industrial Engineering (EIE) GROUP with…”
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Analysis of Structure−Activity Relationships for MT2 Selective Antagonists by Melatonin MT1 and MT2 Receptor Models by Rivara, Silvia, Lorenzi, Simone, Mor, Marco, Plazzi, Pier Vincenzo, Spadoni, Gilberto, Bedini, Annalida, Tarzia, Giorgio

“…Three-dimensional homology models of human MT1 and MT2 melatonin receptors were built with the aim to investigate the structure−activity relationships (SARs)…”
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MT2 selective melatonin receptor antagonists: design and structure-activity relationships by Rivara, Silvia, Mor, Marco, Lorenzi, Simone, Lodola, Alessio, Spadoni, Pier Vincenzo Plazzi Gilberto, Bedini, Annalida, Tarzia, Giorgio

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Da “Freaky Stiley” a “Jack Frusciante”: le prime prove narrative di Enrico Brizzi (pp. 186-206) by De Lorenzi, Simone

“…Il lavoro prende in esame il romanzo d’esordio di Enrico Brizzi Jack Frusciante è uscito dal gruppo (1994) evidenziando le connessioni con tre antecedenti…”
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Use of Experimental Design To Optimize Docking Performance: The Case of LiGenDock, the Docking Module of Ligen, a New De Novo Design Program by Beato, Claudia, Beccari, Andrea R, Cavazzoni, Carlo, Lorenzi, Simone, Costantino, Gabriele

“…On route toward a novel de novo design program, called LiGen, we developed a docking program, LiGenDock, based on pharmacophore models of binding sites,…”
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Biological and Biophysical Properties of the Histone Deacetylase Inhibitor Suberoylanilide Hydroxamic Acid Are Affected by the Presence of Short Alkyl Groups on the Phenyl Ring by Oger, Frédérik, Lecorgne, Aurélien, Sala, Elisa, Nardese, Vanessa, Demay, Florence, Chevance, Soizic, Desravines, Danielle C, Aleksandrova, Nataliia, Guével, Rémy Le, Lorenzi, Simone, Beccari, Andrea R, Barath, Peter, Hart, Darren J, Bondon, Arnaud, Carettoni, Daniele, Simonneaux, Gérard, Salbert, Gilles

“…Inhibition of histone deacetylases (HDACs) leads to growth arrest, differentiation, or apoptosis of tumor cell lines, suggesting HDACs as promising targets for…”
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Design and Synthesis of N-(3,3-Diphenylpropenyl)alkanamides as a Novel Class of High-Affinity MT2-Selective Melatonin Receptor Ligands by Bedini, Annalida, Spadoni, Gilberto, Gatti, Giuseppe, Lucarini, Simone, Tarzia, Giorgio, Rivara, Silvia, Lorenzi, Simone, Lodola, Alessio, Mor, Marco, Lucini, Valeria, Pannacci, Marilou, Scaglione, Francesco

“…A novel series of melatonin receptor ligands was discovered by opening the cyclic scaffolds of known classes of high affinity melatonin receptor antagonists,…”
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Validation of a histamine H3 receptor model through structure-activity relationships for classical H3 antagonists by LORENZI, Simone, MOR, Marco, BORDI, Fabrizio, RIVARA, Silvia, RIVARA, Mirko, MORINI, Giovanni, BERTONI, Simona, BALLABENI, Vigilio, BAROCELLI, Elisabetta, PLAZZI, Pier Vincenzo

“…Histamine H(3) receptor is a G protein-coupled receptor whose activation inhibits the synthesis and release of histamine and other neurotransmitters from nerve…”
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Dibasic non-imidazole histamine H3 receptor antagonists with a rigid biphenyl scaffold by MORINI, Giovanni, COMINI, Mara, BAROCELLI, Elisabetta, PLAZZI, Pier Vincenzo, RIVARA, Mirko, RIVARA, Silvia, LORENZI, Simone, BORDI, Fabrizio, MOR, Marco, FLAMMINI, Lisa, BERTONI, Simona, BALLABENI, Vigilio

“…A class of rigid, dibasic, non-imidazole H3 antagonists was developed, starting from a series of previously described flexible compounds. The original…”
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Dibasic non-imidazole histamine H 3 receptor antagonists with a rigid biphenyl scaffold by Morini, Giovanni, Comini, Mara, Rivara, Mirko, Rivara, Silvia, Lorenzi, Simone, Bordi, Fabrizio, Mor, Marco, Flammini, Lisa, Bertoni, Simona, Ballabeni, Vigilio, Barocelli, Elisabetta, Plazzi, Pier Vincenzo

“…A class of rigid dibasic H 3 antagonists is reported. Compound 5 with subnanomolar affinity for human H 3 receptor was identified. A class of rigid, dibasic,…”
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Validation of a histamine H 3 receptor model through structure–activity relationships for classical H 3 antagonists by Lorenzi, Simone, Mor, Marco, Bordi, Fabrizio, Rivara, Silvia, Rivara, Mirko, Morini, Giovanni, Bertoni, Simona, Ballabeni, Vigilio, Barocelli, Elisabetta, Plazzi, Pier Vincenzo

“…Histamine H 3 receptor is a G protein-coupled receptor whose activation inhibits the synthesis and release of histamine and other neurotransmitters from nerve…”
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Synthesis, Enantiomeric Resolution, and Structure-Activity Relationship Study of a Series of 10,11-Dihydro-5H-Dibenzo[a,d]cycloheptene MT2 Receptor Antagonists by Spadoni, Gilberto, Bedini, Annalida, Diamantini, Giuseppe, Tarzia, Giorgio, Rivara, Silvia, Lorenzi, Simone, Lodola, Alessio, Mor, Marco, Lucini, Valeria, Pannacci, Marilou, Caronno, Alessia, Fraschini, Franco

“…Racemic N‐(8‐methoxy‐10,11‐dihydro‐5H‐dibenzo[a,d]cyclohepten‐10‐ylmethyl)acetamide (compound 5) was previously identified as a novel selective MT2 antagonist…”
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Analysis of Structure−Activity Relationships for MT 2 Selective Antagonists by Melatonin MT 1 and MT 2 Receptor Models by Rivara, Silvia, Lorenzi, Simone, Mor, Marco, Plazzi, Pier Vincenzo, Spadoni, Gilberto, Bedini, Annalida, Tarzia, Giorgio

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Design and Synthesis of N -(3,3-Diphenylpropenyl)alkanamides as a Novel Class of High-Affinity MT 2 -Selective Melatonin Receptor Ligands by Bedini, Annalida, Spadoni, Gilberto, Gatti, Giuseppe, Lucarini, Simone, Tarzia, Giorgio, Rivara, Silvia, Lorenzi, Simone, Lodola, Alessio, Mor, Marco, Lucini, Valeria, Pannacci, Marilou, Scaglione, Francesco

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Synthesis, Enantiomeric Resolution, and Structure–Activity Relationship Study of a Series of 10,11‐Dihydro‐5 H ‐Dibenzo[a,d]cycloheptene MT 2 Receptor Antagonists by Spadoni, Gilberto, Bedini, Annalida, Diamantini, Giuseppe, Tarzia, Giorgio, Rivara, Silvia, Lorenzi, Simone, Lodola, Alessio, Mor, Marco, Lucini, Valeria, Pannacci, Marilou, Caronno, Alessia, Fraschini, Franco

“…Abstract Racemic N ‐(8‐methoxy‐10,11‐dihydro‐5 H ‐dibenzo[a,d]cyclohepten‐10‐ylmethyl)acetamide (compound 5 ) was previously identified as a novel selective MT…”
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Evaluation of the efficacy of personal protective equipment against occupational exposure to cold by Rossi, Simone Lorenzi, Bortolosso, Heléia, Silva, Ricardo, de Mello, Josiane Maria Muneron, Costella, Marcelo Fabiano

“…The temperature of climate controlled areas in the food industry varies from -35°C to 12°C to ensure the quality of food. However, this temperature range might…”
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Dibasic non-imidazole histamine H sub(3) receptor antagonists with a rigid biphenyl scaffold by Morini, Giovanni, Comini, Mara, Rivara, Mirko, Rivara, Silvia, Lorenzi, Simone, Bordi, Fabrizio, Mor, Marco, Flammini, Lisa, Bertoni, Simona, Ballabeni, Vigilio, Barocelli, Elisabetta, Plazzi, Pier Vincenzo

“…A class of rigid, dibasic, non-imidazole H sub(3) antagonists was developed, starting from a series of previously described flexible compounds. The original…”
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Avaliação da eficácia dos equipamentos de proteção individual para a exposição ocupacional ao frio by Rossi, Simone Lorenzi, Bortolosso, Heléia, Silva, Ricardo, Mello, Josiane Maria Muneron de, Costella, Marcelo Fabiano

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Evaluation of the efficacy of personal protective equipment against occupational exposure to cold/Avaliacao da eficacia dos equipamentos de protecao individual para a exposicao ocupacional ao frio by Rossi, Simone Lorenzi, Bortolosso, Heleia, Silva, Ricardo, de Mello, Josiane Maria Muneron, Costella, Marcelo Fabiano

“…Background: The temperature of climate controlled areas in the food industry varies from -35[degrees]C to 12[degrees]C to ensure the quality of food. However,…”
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Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors by Mor, Marco, Rivara, Silvia, Lodola, Alessio, Lorenzi, Simone, Bordi, Fabrizio, Plazzi, Pier Vincenzo, Spadoni, Gilberto, Bedini, Annalida, Duranti, Andrea, Tontini, Andrea, Tarzia, Giorgio

“…Quantitative structure–activity relationships (QSARs) are frequently employed in medicinal chemistry projects, both to rationalize structure–activity…”
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