Search Results - "LA COLLA, M"

In Vitro Activity and Resistance Profile of Samatasvir, a Novel NS5A Replication Inhibitor of Hepatitis C Virus by BILELLO, J. P, LALLOS, L. B, MCCARVILLE, J. F, LA COLLA, M, SERRA, I, CHAPRON, C, GILLUM, J. M, PIERRA, C, STANDRING, D. N, SEIFER, M

“…The hepatitis C virus (HCV) nonstructural 5A (NS5A) protein is a clinically validated target for drugs designed to treat chronic HCV infection. This study…”
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Quadratus Lumborum Block as Sole, Homeostatic-Preserving Anesthetic for a Patient with Multiple System Atrophy Undergoing Open Inguinal Hernia Repair: A Case Report by La Colla, M. D. Luca, Schroeder, R. M. D.

“…Quadratus Lumborum (QL) block has been successfully used for different abdominal procedures in the past. Multiple system atrophy (MSA) is a progressive…”
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P1244 FAVORABLE PRECLINICAL PROFILE OF IDX21437, A NOVEL URIDINE NUCLEOTIDE PRODRUG, FOR USE IN A DIRECT-ACTING ANTIVIRAL (DAA) REGIMEN FOR HCV by Gupta, K, Seifer, M, Serra, I, Rashidzadeh, H, Luo, S, La Colla, M, Pan-Zhou, X.-R, Chapron, C, Hernandez-Santiago, B, Mayes, B, Bhadresa, S, Moussa, A, Rush, R

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815 IDENIX NS5A HCV REPLICATION INHIBITORS WITH LOW PICOMOLAR, PAN-GENOTYPIC IN VITRO ANTIVIRAL ACTIVITY by Dousson, C.B, Chapron, C, Standring, D, Bilello, J.P, McCarville, J, La Colla, M, Seifer, M, Parsy, C, Dukhan, D, Pierra, C, Surleraux, P

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Structure-Based Design, Synthesis, and Biological Evaluation of Conformationally Restricted Novel 2-Alkylthio-6-[1-(2,6-difluorophenyl)alkyl]- 3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as Non-nucleoside Inhibitors of HIV-1 Reverse Transcriptase by Mai, Antonello, Sbardella, Gianluca, Artico, Marino, Ragno, Rino, Massa, Silvio, Novellino, Ettore, Greco, Giovanni, Lavecchia, Antonio, Musiu, Chiara, La Colla, Massimiliano, Murgioni, Chiara, La Colla, Paolo, Loddo, Roberta

“…5-Alkyl-2-(alkylthio)-6-(2,6-difluorobenzyl)-3,4-dihydropyrimidin-4(3H)-ones (S-DABOs, 2) have been recently described as a new class of human immunodeficiency…”
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20 IN VITRO ACTIVITY AND PHARMACOLOGIC PROPERTIES OF TWO NOVEL SERIES OF HCV PROTEASE INHIBITORS by Standring, D.N, Parsy, C, Alexandre, F.-R, Derock, M, Leroy, F, Convard, T, La Colla, M, Lallos, L, Loi, A.-G, Musiu, C, Marceddu, T, Poddesu, B, Vargiu, L, Liuzzi, M, Surleraux, D

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588 IN VITRO ANTIVIRAL ACTIVITY AND PHARMACOLOGY OF IDX184, A NOVEL AND POTENT INHIBITOR OF HCV REPLICATION by Cretton-Scott, E, Perigaud, C, Peyrottes, S, Licklider, L, Camire, M, Larsson, M, La Colla, M, Hildebrand, E, Lallos, L, Bilello, J, McCarville, J, Seifer, M, Liuzzi, M, Pierra, C, Badaroux, E, Gosselin, G, Surleraux, D, Standring, D.N

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Erratum to “Quadratus Lumborum Block as Sole, Homeostatic-Preserving Anesthetic for a Patient with Multiple System Atrophy Undergoing Open Inguinal Hernia Repair: A Case Report” by La Colla, M. D. Luca, Schroeder, R. M. D.

“…In the article titled “Quadratus Lumborum Block as Sole, Homeostatic-Preserving Anesthetic for a Patient with Multiple System Atrophy Undergoing Open Inguinal…”
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IDX375, A Novel Allosteric HCV Polymerase Inhibitor: In Vitro Antiviral Activity and Preclinical Profile by Dousson, C.B., Good, S.S., La Colla, M., Bilello, J., Seifer, M., Standring, D.N., Paparin, J.-L., Surleraux, D.

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2,6-Bis(3,4,5-trihydroxybenzylydene) derivatives of cyclohexanone: novel potent HIV-1 integrase inhibitors that prevent HIV-1 multiplication in cell-based assays by Costi, Roberta, Santo, Roberto Di, Artico, Marino, Massa, Silvio, Ragno, Rino, Loddo, Roberta, La Colla, Massimiliano, Tramontano, Enzo, La Colla, Paolo, Pani, Alessandra

“…A number of 2,6-bisbenzylidenecyclohexane-1-one derivatives have been synthesized and tested as HIV-1 integrase (IN) inhibitors with the aim of obtaining…”
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Simple, Short Peptide Derivatives of a Sulfonylindolecarboxamide (L-737,126) Active in Vitro against HIV-1 Wild Type and Variants Carrying Non-Nucleoside Reverse Transcriptase Inhibitor Resistance Mutations by Silvestri, Romano, Artico, Marino, De Martino, Gabriella, La Regina, Giuseppe, Loddo, Roberta, La Colla, Massimiliano, La Colla, Paolo

“…Non-nucleoside reverse transcriptase inhibitors (NNRTIs) active against NNRTI-resistant mutants were obtained by introducing two methyl groups at positions 3…”
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Structure-Based Design, Parallel Synthesis, Structure−Activity Relationship, and Molecular Modeling Studies of Thiocarbamates, New Potent Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitor Isosteres of Phenethylthiazolylthiourea Derivatives by Ranise, Angelo, Spallarossa, Andrea, Cesarini, Sara, Bondavalli, Francesco, Schenone, Silvia, Bruno, Olga, Menozzi, Giulia, Fossa, Paola, Mosti, Luisa, La Colla, Massimiliano, Sanna, Giuseppina, Murreddu, Marta, Collu, Gabriella, Busonera, Bernardetta, Marongiu, Maria Elena, Pani, Alessandra, La Colla, Paolo, Loddo, Roberta

“…In this paper we describe our structure-based ligand design, synthetic strategy, and structure−activity relationship (SAR) studies that led to the…”
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In-water reactivity of nucleosides and nucleotides: one-step preparation and biological evaluation of novel ferrocenyl-derivatives by de Champdoré, Marcella, Di Fabio, Giovanni, Messere, Anna, Montesarchio, Daniela, Piccialli, Gennaro, Loddo, Roberta, La Colla, Massimiliano, La Colla, Paolo

“…The reactivity in water of a series of nucleosides and nucleotides towards ferrocenemethanol was investigated. Several adducts incorporating the…”
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Synthesis and antiproliferative activity of 3-aryl-2-(1 H-benzotriazol-1-yl)acrylonitriles. Part III by Carta, Antonio, Sanna, Paolo, Palomba, Michele, Vargiu, Laura, La Colla, Massimiliano, Loddo, Roberta

“…A new series of 30 3-aryl-2-(1 H-benzotriazol-1-yl)acrylonitriles were synthesized and tested for biological activity as part of our research in the…”
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344 PRECLINICAL PROFILES OF IDX136 AND IDX316, TWO NOVEL MACROCYCLIC HCV PROTEASE INHIBITORS by Lallos, L.B, Bilello, J.P, Soubasakos, M.A, Gillum, J, Colla, M. La, Liuzzi, M, Carville, J. Mc, Seifer, M, Good, S.S, Larsson, M, Selden, J, Parsy, C, Surleraux, D, Standring, D.N

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Simple, Short Peptide Derivatives of a Sulfonylindolecarboxamide (L-737,126) Active in Vitro against HIV-1 Wild Type and Variants Carrying Non-Nucleoside Reverse Transcriptase Inhibitor Resistance Mutations by Silvestri, R., Artico, M., DeMartino, G., LaRegina, G., Loddo, R., LaColla, M., Mura, M., LaColla, P.

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6-Aryl-2,4-dioxo-5-hexenoic acids, novel integrase inhibitors active against HIV-1 multiplication in cell-based assays by Costi, Roberta, Santo, Roberto Di, Artico, Marino, Roux, Alessandra, Ragno, Rino, Massa, Silvio, Tramontano, Enzo, La Colla, Massimiliano, Loddo, Roberta, Marongiu, M.Elena, Pani, Alessandra, Colla, Paolo La

“…A series of 6-aryl-2,4-dioxo-5-hexenoic acids, were synthesized and tested against HIV-1 in cell-based assays and against recombinant HIV-1 integrase (rIN) in…”
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Quadratus Lumborum Block as Sole, Homeostatic-Preserving Anesthetic for a Patient with Multiple System Atrophy Undergoing Open Inguinal Hernia Repair: A Case Report by La Colla, Luca, La Colla, M D Luca, Schroeder, Rebecca, Schroeder, R M D

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