Search Results - "Kuzemko, Michael A"

3-Aryl-2-(3'-substituted-1',2',4'-oxadiazol-5'-yl)tropane analogs of cocaine: affinities at the cocaine binding site at the dopamine, serotonin, and norepinephrine transporters by Carroll, F. Ivy, Gray, Jeffrey L, Abraham, Philip, Kuzemko, Michael A, Lewin, Anita H, Boja, John W, Kuhar, Michael J

“…Previous studies have shown that 3 beta-(substituted phenyl)tropan-2 beta-carboxylic acid esters possess high affinity for the cocaine binding site on the…”
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A Green Chemistry Comparative Analysis of the Syntheses of (E)-4-Cyclobutyl-2-[2-(3-nitrophenyl)ethenyl] Thiazole, Ro 24-5904 by Kuzemko, Michael A, Van Arnum, Susan D, Niemczyk, Henry J

“…The malonic acid, the Wittig−Horner, and Claisen syntheses for the preparation of Ro 24-5904 (1) are analyzed using the Andraos' reaction analysis metrics…”
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Use of dilithiomethane equivalent in a novel one-flask [2 + 1 + 2] cyclopentannulation reaction: a highly efficient total synthesis of (.+-.)-hirsutene by Ramig, Keith, Kuzemko, Michael A, McNamara, Kevin, Cohen, Theodore

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Synthesis, Ligand Binding, and QSAR (CoMFA and Classical) Study of 3.beta.-(3'-Substituted phenyl)-, 3.beta.-(4'-Substituted phenyl)-, and 3.beta.-(3',4'-Disubstituted phenyl)tropane-2.beta.-carboxylic Acid Methyl Esters by Carroll, F. Ivy, Mascarella, S. Wayne, Kuzemko, Michael A, Gao, Yigong, Abraham, Philip, Lewin, Anita H, Boja, John W, Kuhar, Michael J

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Cocaine and 3.beta.-(4'-Substituted phenyl)tropane-2.beta.-carboxylic Acid Ester and Amide Analogs. New High-Affinity and Selective Compounds for the Dopamine Transporter by Carroll, F. Ivy, Kotian, Pravin, Dehghani, Ali, Gray, Jeffrey L, Kuzemko, Michael A, Parham, Karol A, Abraham, Philip, Lewin, Anita H, Boja, John W, Kuhar, Michael J

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Proton-transfer reactions. 4. Near-unity kinetic isotope effects for hydron exchange and dehydrofluorination reactions by Koch, Heinz F, Dahlberg, Donald B, Lodder, Gerrit, Root, Karen S, Touchette, Nancy A, Solsky, Robert L, Zuck, Robin M, Wagner, Linda J, Koch, Nanci H, Kuzemko, Michael A

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Cocaine and 3β-(4'-substituted phenyl)tropane-2β-carboxylic acid ester and amide analogues. New high-affinity and selective compounds for the dopamine transporter by CARROLL, F. I, KOTIAN, P, ALI DEHGHANI, GRAY, J. L, KUZEMKO, M. A, PARHAM, K. A, ABRAHAM, P, LEWIN, A. H, BOJA, J. W, KUHAR, M. J

“…Several 2 beta-carboxylic acid ester and amide analogues of cocaine and of 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid were prepared. The…”
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Synthesis, ligand binding, and QSAR (CoMFA and classical) study of 3β-(3'-substituted phenyl)-, 3β-(4'-substituted phenyl)-, and 3β-(3',4'-disubstituted phenyl)tropane-2β-carboxylic acid methyl esters by CARROLL, F. I, MASCARELLA, S. W, KUZEMKO, M. A, YIGONG GAO, ABRAHAM, P, LEWIN, A. H, BOJA, J. W, KUHAR, M. J

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