Search Results - "Kruppa, Marco"

A Survey on the Synthesis of Variolins, Meridianins, and Meriolins-Naturally Occurring Marine (aza)Indole Alkaloids and Their Semisynthetic Derivatives by Kruppa, Marco, Müller, Thomas J J

“…Marine natural products are a source of essential significance due to a plethora of highly diverse biological properties. The naturally occurring (aza)indole…”
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Concise Syntheses of Marine (Bis)indole Alkaloids Meridianin C, D, F, and G and Scalaridine A via One-Pot Masuda Borylation-Suzuki Coupling Sequence by Kruppa, Marco, Sommer, Gereon A, Müller, Thomas J J

“…-Protected 3-iodoindoles were reacted with (di)azine halides in a sequentially Pd-catalyzed one-pot fashion, i.e., by Masuda borylation-Suzuki coupling (MBSC)…”
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Masuda Borylation–Suzuki Coupling (MBSC) Sequence: A One-Pot Process to Access Complex (hetero)Biaryls by Marco Kruppa, Thomas J. J. Müller

“…The direct formation of (hetero)biaryls from readily available (hetero)aryl halides under mild reaction conditions can be efficiently achieved through the…”
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Nature-Inspired (di)Azine-Bridged Bisindole Alkaloids with Potent Antibacterial In Vitro and In Vivo Efficacy against Methicillin-Resistant Staphylococcus aureus by Rehberg, Nidja, Sommer, Gereon A, Drießen, Daniel, Kruppa, Marco, Adeniyi, Emmanuel T, Chen, Shang, Wang, Lin, Wolf, Karina, Tasch, Boris O. A, Ioerger, Thomas R, Zhu, Kui, Müller, Thomas J. J, Kalscheuer, Rainer

“…Natural bisindole alkaloids such as Hyrtinadine A and Alocasin A, which are known to exhibit diverse bioactivities, provide promising chemical scaffolds for…”
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Synthesis of Bisindole Alkaloids and Their Mode of Action against Methicillin-Resistant Staphylococcus Aureus by Adeniyi, Emmanuel T., Kruppa, Marco, De Benedetti, Stefania, Ludwig, Kevin C., Krisilia, Violetta, Wassenberg, Tobias R., Both, Melissa, Schneider, Tanja, Müller, Thomas J. J., Kalscheuer, Rainer

“…About 100,000 deaths are attributed annually to infections with methicillin-resistant Staphylococcus aureus (MRSA) despite concerted efforts toward vaccine…”
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