Search Results - "Krüll, Jasmin"

Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach by Engel, Julian, Richters, André, Getlik, Matthäus, Tomassi, Stefano, Keul, Marina, Termathe, Martin, Lategahn, Jonas, Becker, Christian, Mayer-Wrangowski, Svenja, Grütter, Christian, Uhlenbrock, Niklas, Krüll, Jasmin, Schaumann, Niklas, Eppmann, Simone, Kibies, Patrick, Hoffgaard, Franziska, Heil, Jochen, Menninger, Sascha, Ortiz-Cuaran, Sandra, Heuckmann, Johannes M., Tinnefeld, Verena, Zahedi, René P., Sos, Martin L., Schultz-Fademrecht, Carsten, Thomas, Roman K., Kast, Stefan M., Rauh, Daniel

“…Receptor tyrosine kinases represent one of the prime targets in cancer therapy, as the dysregulation of these elementary transducers of extracellular signals,…”
Get full text

[18F]Fluorine‐Labeled Pharmaceuticals: Direct Aromatic Fluorination Compared to Multi‐Step Strategies by Krüll, Jasmin, Heinrich, Markus R.

“…Positron emission tomography (PET) presents an important tool for medicinal and pharmaceutical investigations, with applications ranging from fundamental…”
Get full text

Inhibitors to Overcome Secondary Mutations in the Stem Cell Factor Receptor KIT by Kaitsiotou, Helena, Keul, Marina, Hardick, Julia, Mühlenberg, Thomas, Ketzer, Julia, Ehrt, Christiane, Krüll, Jasmin, Medda, Federico, Koch, Oliver, Giordanetto, Fabrizio, Bauer, Sebastian, Rauh, Daniel

“…In modern cancer therapy, the use of small organic molecules against receptor tyrosine kinases (RTKs) has been shown to be a valuable strategy. The association…”
Get full text

Microwave‐Assisted Rapid One‐Pot Synthesis of Fused and Non‐Fused Indoles and 5‐[18F]Fluoroindoles from Phenylazocarboxylates by Krüll, Jasmin, Hubert, Anja, Nebel, Natascha, Prante, Olaf, Heinrich, Markus R.

“…Substituted indoles can be prepared from phenylazocarboxylates through a rapid one‐pot sequence featuring a microwave‐assisted Fischer indole synthesis as a…”
Get full text

Sustainable Synthesis of Balsalazide and Sulfasalazine Based on Diazotization with Low Concentrations of Nitrogen Dioxide in Air by Hofmann, Dagmar, Gans, Eva, Krüll, Jasmin, Heinrich, Markus R.

“…Low concentrations of nitrogen dioxide, which arises as a side product from a range of industrial processes, can effectively be recycled through the…”
Get full text

Inside Cover: Sustainable Synthesis of Balsalazide and Sulfasalazine Based on Diazotization with Low Concentrations of Nitrogen Dioxide in Air (Chem. Eur. J. 17/2017) by Hofmann, Dagmar, Gans, Eva, Krüll, Jasmin, Heinrich, Markus R.

“…From waste to valuables: The industrial production of copper nitrate from copper produces large amounts of toxic NO2. Instead of costly denitrification, this…”
Get full text

Tuning the Polarity of Antibiotic‐Cy5 Conjugates Enables Highly Selective Labeling of Binding Sites by Graßl, Fabian, Konrad, Maike M. B., Krüll, Jasmin, Pezerovic, Azra, Zähnle, Leon, Burkovski, Andreas, Heinrich, Markus R.

“…Multidrug‐resistant bacteria pose a major threat to global health, even as newly introduced antibiotics continue to lose their therapeutic value. Against this…”
Get full text

Selective Functionalization of Graphene at Defect‐Activated Sites by Arylazocarboxylic tert‐Butyl Esters by Halbig, Christian E., Lasch, Roman, Krüll, Jasmin, Pirzer, Anna S., Wang, Zhenping, Kirchhof, Jan N., Bolotin, Kirill I., Heinrich, Markus R., Eigler, Siegfried

“…The development of versatile functionalization concepts for graphene is currently in the focus of research. Upon oxo‐functionalization of graphite, the full…”
Get full text

Synthesis, Radiosynthesis and Biological Evaluation of Buprenorphine‐Derived Phenylazocarboxamides as Novel μ‐Opioid Receptor Ligands by Krüll, Jasmin, Fehler, Stefanie K., Hofmann, Laura, Nebel, Natascha, Maschauer, Simone, Prante, Olaf, Gmeiner, Peter, Lanig, Harald, Hübner, Harald, Heinrich, Markus R.

“…Targeted structural modifications have led to a novel type of buprenorphine‐derived opioid receptor ligand displaying an improved selectivity profile for the…”
Get full text

Selective functionalization of graphene at defect activated sites by arylazocarboxylic tert-butylesters by Eigler, Siegfried, Heinrich, Markus R, Halbig, Christian E, Lasch, Roman, Krüll, Jasmin, Prizer, Anna, Wang, Zhenping, Kirchhof, Jan N, Bolotin, Kirill I

“…The development of versatile functionalization concepts for graphene are currently in the focus of research. With oxo-functionalization of graphite the full…”
Get full text

Selektive Funktionalisierung von Graphen an defektaktivierten Bereichen durch Arylazocarbonsäure‐tert‐butylester by Halbig, Christian E., Lasch, Roman, Krüll, Jasmin, Pirzer, Anna S., Wang, Zhenping, Kirchhof, Jan N., Bolotin, Kirill I., Heinrich, Markus R., Eigler, Siegfried

“…Die Entwicklung vielseitiger Funktionalisierungskonzepte für Graphen steht derzeit im Fokus der Forschung. Mittels Oxo‐Funktionalisierung von Graphit wird die…”
Get full text

Selektive Funktionalisierung von Graphen an defektaktivierten Bereichen durch Arylazocarbonsäure‐ tert ‐butylester by Halbig, Christian E., Lasch, Roman, Krüll, Jasmin, Pirzer, Anna S., Wang, Zhenping, Kirchhof, Jan N., Bolotin, Kirill I., Heinrich, Markus R., Eigler, Siegfried

“…Abstract Die Entwicklung vielseitiger Funktionalisierungskonzepte für Graphen steht derzeit im Fokus der Forschung. Mittels Oxo‐Funktionalisierung von Graphit…”
Get full text