Search Results - "Khatab, Tamer K"
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Biological Evaluation and Molecular Docking with In Silico Physicochemical, Pharmacokinetic and Toxicity Prediction of Pyrazolo[1,5- a ]pyrimidines
Published in Molecules (Basel, Switzerland) (21-03-2020)“…Pyrazolo[1,5- ]pyrimidines - , - and - were synthesized for evaluation of their in vitro antimicrobial properties against some microorganisms and their…”
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2
Synthesis and characterization of curcumin-encapsulated loaded on carboxymethyl cellulose with docking validation as α-amylase and α-glucosidase inhibitors
Published in Polish journal of chemical technology (01-09-2024)“…In reaction to the expanding predominance of diabetes mellitus, curcumin nanoparticles stacked on carboxymethyl cellulose (CMC) composite were effectively…”
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V2O5 based quadruple nano‐perovskite as a new catalyst for the synthesis of bis and tetrakis heterocyclic compounds
Published in Applied organometallic chemistry (01-05-2019)“…In this article, we presented a novel, efficient and facile approach for using strontium titanate supported catalyst in organic synthesis. Bis and tetrakis of…”
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4
Pulsed laser ablated zeolite nanoparticles: A novel nano‐catalyst for the synthesis of 1,8‐dioxo‐octahydroxanthene and N‐aryl‐1,8‐dioxodecahydroacridine with molecular docking validation
Published in Applied organometallic chemistry (01-02-2020)“…There is an increasing interest in the synthesis of metal nanoparticles (NPs) from bulk metals using pulsed laser ablation in liquids (PLAL), as it offers an…”
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5
Copper–Vit B3 MOF preparation, characterization and catalytic evaluation in a one-pot synthesis of benzoxanthenones with docking validation as anti H. pylori
Published in RSC advances (27-06-2024)“…Copper–Vit B3 MOF was successfully prepared by efficient and eco hydrothermal method. The prepared MOF was characterized as a tetragonal crystal copper-MOF…”
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6
Copper-Vit B 3 MOF preparation, characterization and catalytic evaluation in a one-pot synthesis of benzoxanthenones with docking validation as anti H. pylori
Published in RSC advances (27-06-2024)“…Copper-Vit B MOF was successfully prepared by efficient and eco hydrothermal method. The prepared MOF was characterized as a tetragonal crystal copper-MOF…”
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7
Synthesis and molecular docking studies of some new thiosemicarbazone derivatives as HCV polymeraseinhibitors
Published in Synthetic communications (03-06-2019)“…Series of new thiosemicarbazones was prepared and molecular studied as inhibitors of HCV 4WTG polymerase. Thus, the thiosemicarbazone derivatives (3a-k) were…”
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8
Design and Synthesis Pairing Between Xanthene and Tetrazole in Pentacyclic System Using Tetrachlorosilane with Aurora Kinase Inhibitor Validation
Published in Journal of heterocyclic chemistry (01-07-2017)“…A competent new one‐pot synthesis for tetrahydrobenzo[f]chromeno[3,2‐c]tetrazolo[1,5‐a]azepines through the catalytic synthesis of related xanthenes…”
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9
Red-sea dolomite as a sustainable catalyst in the synthesis of bis-indolyl methanes with molecular docking validation as HIV-1 replication inhibitor
Published in Bulletin of the Chemical Society of Ethiopia (01-09-2021)“…Dolomite minerals were collected from the Red Sea Mountains around the Sokhna region. The rock was collected, rinsed, and crushed using a ball mailing machine…”
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10
Copper-based glass-ceramic as an efficient catalyst in the synthesis of pyrazolo[1,5-a] pyrimidineunder solvent-free condition with docking validation as Covid-19 main protease (Mpro) inhibitor
Published in Bulletin of the Chemical Society of Ethiopia (01-01-2021)“…Copper-based oxide glass-ceramic was successfully synthesized through the single-step melt annealing technique. Synthesized glass-ceramics was characterized…”
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11
New Approach for Tetrachlorosilane Promoted One-Pot, Condensation Reaction for Tetrahydrobenzo[a]Xanthene-11-Ones with Docking Validation as Aurora Kinase Inhibitor
Published in SILICON (01-03-2018)“…An efficient synthesis is reported for tetrahydrobenzo[a]xanthene-11-ones through a one-pot catalytic reaction by mixing β-naphthol, demidone and aromatic…”
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12
V2O5/SiO2 as a Heterogeneous Catalyst in the Synthesis of bis(indolyl)methanes Under Solvent Free Condition
Published in SILICON (01-05-2018)“…The heterogeneous catalyst of V 2 O 5 /SiO 2 was prepared and characterized with Fourier transform infrared spectroscopy (FTIR), X-ray diffraction (XRD) and…”
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13
TCS/ZnCl2 as a controlled reagent for the Michael addition and heterocyclic cyclization based on the phenyl pyrazolone scaffold with docking validation as a Covid-19 protease inhibitor
Published in Bulletin of the Chemical Society of Ethiopia (01-01-2024)“…TCS/ZnCl2 is presented as a new catalyst for achieving the Michael addition adduct 5a-g by the reaction of phenyl pyrazolone 4 as the Michael donor and…”
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14
A new and facile tetrachlorosilane-promoted one-pot condensation for the synthesis of a novel series of tetracyclic 1,5-thiazepines
Published in Tetrahedron letters (29-10-2014)“…A new and facile approach for the one-pot synthesis of a novel series of tetracyclic 1,5-thiazepines is described. The reaction occurs through…”
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15
Chemistry of Phosphorus Ylides: Part 46—Efficient Synthesis and Biological Evaluation of New Phosphorus, Sulfur, and Selenium Pyrazole Derivatives
Published in Journal of heterocyclic chemistry (01-12-2018)“…1,5‐Dimethyl‐3‐oxo‐2‐phenyl‐2,3‐dihydro‐1H‐pyrazole‐4‐carbaldehyde was allowed to react with different phosphorus, sulfur, and selenium reagents. The reaction…”
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16
Utilization of bromine azide to access vicinal-azidobromides from arylidene malononitrile
Published in Chinese chemical letters (01-09-2016)“…An efficient and facile approach for tetrachlorosilane as an in situ mediated transformation via a one-pot, synthesis of vicinal bromoazides through the…”
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17
Evaluation of the Optical and Structural Properties of Constructed Bis-indole Derivatives Using (Sm2O3/SiO2) Catalyst
Published in SILICON (01-09-2018)“…(SiO 2 /Sm 2 O 3 ) was successfully synthesized and examined using scanning electron microscopy; X-ray diffraction and Fourier transform infrared spectroscopy…”
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18
An efficient synthesis of β-acylureas via a three-component, one-pot synthesis using TCS/ZnCl2
Published in Tetrahedron letters (30-03-2011)“…A simple and efficient one-pot, three-component synthesis of new trisubstituted ureas containing diastereotopic protons is achieved via the reaction of…”
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19
Efficient One-pot Synthesis, Antimicrobial and Docking Studies of Some Newer Tetrahydro-4H-benzo [1,3-e]oxazines and Related [beta]-Acylamino Ketone Derivatives
Published in Journal of heterocyclic chemistry (01-03-2017)“…A concise one-step procedure was developed for the synthesis of some newer tetrahydro-4H-benzo[1,3-e]oxazines and [beta]-acylamino ketone derivatives via…”
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20
Biosynthesized Selenium nanoparticles as a new catalyst in the synthesis of quinazoline derivatives in pentacyclic system with docking validation as (TRPV1) inhibitor
Published in Journal of organometallic chemistry (01-07-2021)“…In recent years, a lot of benefits of Selenium have been discovered for humans, animals and chemical uses. Nano-Selenium was biosynthesized and characterized…”
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