Search Results - "Khachatryan, Derenik S"

New Hydrazinothiazole Derivatives of Usnic Acid as Potent Tdp1 Inhibitors by Filimonov, Aleksander S, Chepanova, Arina A, Luzina, Olga A, Zakharenko, Alexandra L, Zakharova, Olga D, Ilina, Ekaterina S, Dyrkheeva, Nadezhda S, Kuprushkin, Maxim S, Kolotaev, Anton V, Khachatryan, Derenik S, Patel, Jinal, Leung, Ivanhoe K H, Chand, Raina, Ayine-Tora, Daniel M, Reynisson, Johannes, Volcho, Konstantin P, Salakhutdinov, Nariman F, Lavrik, Olga I

“…Tyrosyl-DNA phosphodiesterase 1 (Tdp1) is a promising therapeutic target in cancer therapy. Combination chemotherapy using Tdp1 inhibitors as a component can…”
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Albumin-Functionalized Iron Oxide Nanoparticles for Theranostics: Engineering and Long-Term In Situ Imaging by Bychkova, Anna V, Yakunina, Marina N, Lopukhova, Mariia V, Degtyarev, Yevgeniy N, Motyakin, Mikhail V, Pokrovsky, Vadim S, Kovarski, Alexander L, Gorobets, Maria G, Retivov, Vasily M, Khachatryan, Derenik S

“…Magnetic nanosystems (MNSs) consisting of magnetic iron oxide nanoparticles (IONPs) coated by human serum albumin (HSA), commonly used as a component of hybrid…”
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Biologically active quinazoline-based hydroxamic acids by Osipov, Vasily N., Khachatryan, Derenik S., Balaev, Alexandr N.

“…Molecular hybridization has become a new promising way to treat multifactorial diseases with a single compound that acts on multiple targets. The combination…”
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Labeling and receptor affinity of an ultra‐short somatostatin analogue Thz‐Phe‐D‐Trp‐Lys‐Thr‐DOTA by Fedotova, Anzhelika O., Egorova, Bayirta V., Posypanova, Galina A., Titchenko, Nikolay A., Khachatryan, Derenik S., Kolotaev, Anton V., Osipov, Vasiliy N., Kalmykov, Stepan N.

“…Somatostatin analogues play an important role in the therapy of neuroendocrine tumors by binding to somatostatin receptors on the surface of cancer cells. In…”
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Nonmetallic Wurtz coupling reaction of perfluorohexyl iodide by Kolotaev, Anton V., Khachatryan, Derenik S.

“…[Display omitted] •A new pathway of dimerization of perfluoroalkyl halides to perfluoroalkanes was found.•Perfluoroalkyl halides under the action of…”
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Synthesis of new quinazoline-containing hydroxamic acids as potential HDAC/VEGFR inhibitors. Unusual rearrangements with pyrrolidone ring opening and dehydration of 3-N-hydroxyquinazoline fragment containing tetracycles by Kolotaev, Anton V., Matevosyan, Karine R., Osipov, Vasiliy N., Khachatryan, Derenik S.

“…[Display omitted] Synthesis pathways were developed and new hydroxamic acids were obtained as potential inhibitors of HDAC/VEGFR2, including tetracycles…”
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[161Tb]Tb-Thz-Phe-D-Trp-Lys-Thr-DOTA: A potential radiopharmaceutical for the treatment of neuroendocrine tumors by Fedotova, Anzhelika O., Egorova, Bayirta V., Yu. Aleshin, Gleb, Zamurueva, Lyubov S., Alieva, Ramiz A., Posypanova, Galina A., Priselkova, Anna B., Kolotaev, Anton V., Khachatryan, Derenik S., Osipov, Vasily N., Kalmykov, Stepan N.

“…[Display omitted] Thz-Phe-D-Trp-Lys-Thr-DOTA, a conjugate of the DOTA chelator and the Thz-Phe-D-Trp-Lys-Thr pentapeptide, was labeled with 152Eu and 161Tb…”
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