Search Results - "Katti, S.B"

Design, synthesis, and evaluation of 2-aryl-3-heteroaryl-1,3-thiazolidin-4-ones as anti-HIV agents by Rawal, Ravindra K., Tripathi, Rajkamal, Katti, S.B., Pannecouque, Christophe, De Clercq, Erik

“…In the present study, 2-aryl-3-heteroaryl-1,3-thiazolidin-4-ones have been assembled by reflux protocol three component reaction of amine, aldehyde and…”
Get full text

Sixteen-years of clinically relevant dipeptidyl peptidase-IV (DPP-IV) inhibitors for treatment of type-2 diabetes: a perspective by Kushwaha, R N, Haq, W, Katti, S B

“…Inhibition of DPP-IV enzyme has taken centre stage as a validated drug target for type 2 diabetes therapy and as a result of research efforts done towards…”
Get more information

Design and synthesis of 2-(2,6-dibromophenyl)-3-heteroaryl-1,3-thiazolidin-4-ones as anti-HIV agents by Rawal, Ravindra K., Tripathi, Rajkamal, Katti, S.B., Pannecouque, Christophe, De Clercq, Erik

“…A series of 2-(2,6-dibromophenyl)-3-heteroaryl-1,3-thiazolidin-4-ones were designed, synthesized and evaluated as selective human immunodeficiency virus type-1…”
Get full text

Thiazolidin-4-one and thiazinan-4-one derivatives analogous to rosiglitazone as potential antihyperglycemic and antidyslipidemic agents by Raza, Saman, Srivastava, Swayam P., Srivastava, Daya S., Srivastava, Arvind K., Haq, W., Katti, S.B.

“…A number of thiazolidin-4-one and thiazinan-4-one derivatives were prepared by three component condensation in one pot reaction method. These compounds were…”
Get full text

Structure-activity relationship studies on clinically relevant HIV-1 NNRTIs by Rawal, R K, Murugesan, V, Katti, S B

“…In addition to the nucleoside reverse transcriptase inhibitors (NRTIs), protease inhibitors (PIs) and integrase inhibitors (INIs), nonnucleoside reverse…”
Get more information

Design, synthesis and antiplasmodial activity of novel imidazole derivatives based on 7-chloro-4-aminoquinoline by Kondaparla, Srinivasarao, Manhas, Ashan, Dola, Vasantha Rao, Srivastava, Kumkum, Puri, Sunil K., Katti, S.B.

“…[Display omitted] •Novel series of short chain 4-aminoquinoline-imidazole derivatives were designed and synthesized.•Assessment of 4-aminoquinolines for in…”
Get full text

Synthesis and evaluation of 2-(2,6-dihalophenyl)-3-pyrimidinyl-1,3-thiazolidin-4-one analogues as anti-HIV-1 agents by Rawal, Ravindra K., Tripathi, Rajkamal, Katti, S.B., Pannecouque, Christophe, De Clercq, Erik

“…In the present study, a series of 2-(2,6-dihalophenyl)-3-pyrimidinyl-1,3-thiazolidin-4-ones were designed on the prediction of quantitative structure–activity…”
Get full text

2-(Aryl)-3-furan-2-ylmethyl-thiazolidin-4-ones as selective HIV-RT Inhibitors by Rawal, Ravindra K., Prabhakar, Yenamandra S., Katti, S.B., De Clercq, E.

“…In the present study, 4-thiazolidinones have been assembled by DCC-mediated three-component reaction of amine, aldehyde and mercapto acetic acid and tested as…”
Get full text

Antimalarial activity of novel 4-aminoquinolines active against drug resistant strains by Kondaparla, Srinivasarao, Soni, Awakash, Manhas, Ashan, Srivastava, Kumkum, Puri, Sunil K., Katti, S.B.

“…[Display omitted] •Novel side chain modified 4-aminoquinolines were designed and synthesized.•Assessment of 4-aminoquinolines for in vitro and in vivo…”
Get full text

Carbodiimide mediated synthesis of 4-thiazolidinones by one-pot three-component condensation by Srivastava, Tumul, Haq, W, Katti, S.B

“…In the present study, 4-thiazolidinones have been assembled by DCC mediated three-component reaction of amine, aldehyde and mercaptoacetic acid. The final…”
Get full text

4-Aminoquinoline derived antimalarials: Synthesis, antiplasmodial activity and heme polymerization inhibition studies by Solomon, V.R., Haq, W., Smilkstein, M., Srivastava, Kumkum, Puri, Sunil K., Katti, S.B.

“…A new series of 4-aminoquinoline derivatives have been synthesized and found to be active against both susceptible and resistant strains of Plasmodium…”
Get full text

Non-nucleoside inhibitors of the hepatitis C virus NS5B RNA-dependant RNA polymerase : 2-Aryl-3-heteroaryl-1,3-thiazolidin-4-one derivatives by RAWAL, Ravindra K, KATTI, S. B, KAUSHIK-BASU, Neerja, ARORA, Payal, ZHENHUA PAN

“…Hepatitis C virus (HCV) NS5B RNA polymerase is crucial for replicating the HCV RNA genome and is an attractive target for developing anti-HCV drugs. A novel…”
Get full text

Design, synthesis of 4-aminoquinoline-derived thiazolidines and their antimalarial activity and heme polymerization inhibition studies by Solomon, V Raja, Haq, W, Srivastava, Kumkum, Puri, Sunil K, Katti, S B

“…The present study describes the synthesis of a series of new 4-aminoquinoline-derived thiazolidines and evaluation of their antimalarial activity against a…”
Get more information

Design and synthesis of new antimalarial agents from 4-aminoquinoline by Solomon, V. Raja, Puri, Sunil K., Srivastava, Kumkum, Katti, S.B.

“…In the present study, synthesis of a new series of 4-aminoquinoline derivatives and evaluation of their activity against a chloroquine sensitive strain of P…”
Get full text

2-(2,6-Dihalo-phenyl)-3-heteroaryl-2-ylmethyl-1, 3-thiazolidin-4-ones: Anti-HIV agents by Rawal, Ravindra K, Tripathi, Rajkamal, Kulkarni, Smitha, Paranjape, R, Katti, S.B, Pannecouque, Christophe, De Clercq, Erik

“…A diversity of novel 2-aryl-3-heteroaryl-2-ylmethyl-1,3-thiazolidin-4-ones were designed and synthesized by reacting heteroaryl-2-ylmethyl amine with various…”
Get full text

CoMFA and CoMSIA analysis of tetrahydroquinolines as potential antimalarial agents by Deshpande, S., Jaiswal, S., Katti, S.B., Prabhakar, Y.S.

“…Comparative molecular field analysis (CoMFA) and comparative molecular similarity indices analysis (CoMSIA) were used on a dataset of compounds, some of them…”
Get full text

Synthesis and biological evaluation of 2,3-diaryl substituted-1,3-thiazolidin-4-ones as anti-HIV agents by Rawal, Ravindra K, Tripathi, Raj Kamal, Katti, S B, Pannecouque, Christophe, De Clercq, Erik

“…A series of 1,3-thiazolidin-4-ones and metathiazanones were synthesized and evaluated as anti-HIV agents. The results of the in vitro assays showed that some…”
Get more information

Synthesis and antimicrobial activity of erythromycin-A oxime analogs by Pandey, Deepa, Katti, S.B, Haq, W, Tripathi, C.K.M

“…A few amino alcohol as well as ester derivatives of erythromycin-9-oxime have been synthesized in moderate yield. These compounds have shown antibacterial…”
Get full text

A diagnostically relevant epitope of A. fumigatus by Sarma, P.U., Gupta, T.M., Priyadarsiny, P., Shah, A., Haq, W., Katti, S.B.

Get full text

3′-Deoxyribonucleosides and their derivatives as anti-amoebic agents by Ghosal, S, KrishnaPrasad, B.N, Khanna, M, Dwivedi, A.K, Singh, S, Kumar, A, Katti, S.B

“…In general nucleoside analogues were found to possess in vitro amoebicidal property against trophozoites of Entamoeba histolytica. The acid-labile nature of…”
Get full text