Search Results - "Katti, S B"

2-(Aryl)-3-furan-2-ylmethyl-thiazolidin-4-ones as selective HIV-RT Inhibitors by Rawal, Ravindra K., Prabhakar, Yenamandra S., Katti, S.B., De Clercq, E.

“…In the present study, 4-thiazolidinones have been assembled by DCC-mediated three-component reaction of amine, aldehyde and mercapto acetic acid and tested as…”
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Synthesis and Antimalarial Activity of Side Chain Modified 4-Aminoquinoline Derivatives by Solomon, V. Raja, Haq, W., Srivastava, Kumkum, Puri, Sunil K., Katti, S. B.

“…A new series of side-chain modified 4-aminoquinolines have been synthesized and found active against P. falciparum in vitro and P. yoelli in vivo. Compounds 6,…”
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Design, synthesis, and evaluation of 2-aryl-3-heteroaryl-1,3-thiazolidin-4-ones as anti-HIV agents by Rawal, Ravindra K., Tripathi, Rajkamal, Katti, S.B., Pannecouque, Christophe, De Clercq, Erik

“…In the present study, 2-aryl-3-heteroaryl-1,3-thiazolidin-4-ones have been assembled by reflux protocol three component reaction of amine, aldehyde and…”
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Synthesis and evaluation of 2-(2,6-dihalophenyl)-3-pyrimidinyl-1,3-thiazolidin-4-one analogues as anti-HIV-1 agents by Rawal, Ravindra K., Tripathi, Rajkamal, Katti, S.B., Pannecouque, Christophe, De Clercq, Erik

“…In the present study, a series of 2-(2,6-dihalophenyl)-3-pyrimidinyl-1,3-thiazolidin-4-ones were designed on the prediction of quantitative structure–activity…”
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Design and synthesis of 2-(2,6-dibromophenyl)-3-heteroaryl-1,3-thiazolidin-4-ones as anti-HIV agents by Rawal, Ravindra K., Tripathi, Rajkamal, Katti, S.B., Pannecouque, Christophe, De Clercq, Erik

“…A series of 2-(2,6-dibromophenyl)-3-heteroaryl-1,3-thiazolidin-4-ones were designed, synthesized and evaluated as selective human immunodeficiency virus type-1…”
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Synthesis and Evaluation of Chirally Defined Side Chain Variants of 7-Chloro-4-Aminoquinoline To Overcome Drug Resistance in Malaria Chemotherapy by Dola, Vasantha Rao, Soni, Awakash, Agarwal, Pooja, Ahmad, Hafsa, Raju, Kanumuri Siva Rama, Rashid, Mamunur, Wahajuddin, Muhammad, Srivastava, Kumkum, Haq, W, Dwivedi, A K, Puri, S K, Katti, S B

“…A novel 4-aminoquinoline derivative [( )-7-chloro- -(4-methyl-1-(4-methylpiperazin-1-yl)pentan-2-yl)-quinolin-4-amine triphosphate] exhibiting curative…”
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Structure-activity relationship studies on clinically relevant HIV-1 NNRTIs by Rawal, R K, Murugesan, V, Katti, S B

“…In addition to the nucleoside reverse transcriptase inhibitors (NRTIs), protease inhibitors (PIs) and integrase inhibitors (INIs), nonnucleoside reverse…”
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4-Aminoquinoline derived antimalarials: Synthesis, antiplasmodial activity and heme polymerization inhibition studies by Solomon, V.R., Haq, W., Smilkstein, M., Srivastava, Kumkum, Puri, Sunil K., Katti, S.B.

“…A new series of 4-aminoquinoline derivatives have been synthesized and found to be active against both susceptible and resistant strains of Plasmodium…”
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Non-nucleoside inhibitors of the hepatitis C virus NS5B RNA-dependant RNA polymerase : 2-Aryl-3-heteroaryl-1,3-thiazolidin-4-one derivatives by RAWAL, Ravindra K, KATTI, S. B, KAUSHIK-BASU, Neerja, ARORA, Payal, ZHENHUA PAN

“…Hepatitis C virus (HCV) NS5B RNA polymerase is crucial for replicating the HCV RNA genome and is an attractive target for developing anti-HCV drugs. A novel…”
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Human beta casein fragment (54-59) modulates M. bovis BCG survival and basic transcription factor 3 (BTF3) expression in THP-1 cell line by Thakur, Dharamsheela, Saxena, Reshu, Singh, Vandana, Haq, Wahajul, Katti, S B, Singh, Bhupendra Narain, Tripathi, Raj Kamal

“…Immunostimulatory peptides potentiate the immune system of the host and are being used as a viable adjunct to established therapeutic modalities in treatment…”
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Design and synthesis of new antimalarial agents from 4-aminoquinoline by Solomon, V. Raja, Puri, Sunil K., Srivastava, Kumkum, Katti, S.B.

“…In the present study, synthesis of a new series of 4-aminoquinoline derivatives and evaluation of their activity against a chloroquine sensitive strain of P…”
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Design, synthesis and antiplasmodial activity of novel imidazole derivatives based on 7-chloro-4-aminoquinoline by Kondaparla, Srinivasarao, Manhas, Ashan, Dola, Vasantha Rao, Srivastava, Kumkum, Puri, Sunil K., Katti, S.B.

“…[Display omitted] •Novel series of short chain 4-aminoquinoline-imidazole derivatives were designed and synthesized.•Assessment of 4-aminoquinolines for in…”
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Isolation, characterization and antifungal docking studies of wortmannin isolated from Penicillium radicum by Singh, Vineeta, Praveen, Vandana, Tripathi, Divya, Haque, Shafiul, Somvanshi, Pallavi, Katti, S. B., Tripathi, C. K. M.

“…During the search for a potent antifungal drug, a cell-permeable metabolite was isolated from a soil isolate taxonomically identified as Penicillium radicum…”
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Synthesis and biological evaluation of 4-thiazolidinone derivatives as potential antimycobacterial agents by Srivastava, Tumul, Gaikwad, A., Haq, W., Sinha, S., Katti, S. B.

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Sixteen-years of clinically relevant dipeptidyl peptidase-IV (DPP-IV) inhibitors for treatment of type-2 diabetes: a perspective by Kushwaha, R N, Haq, W, Katti, S B

“…Inhibition of DPP-IV enzyme has taken centre stage as a validated drug target for type 2 diabetes therapy and as a result of research efforts done towards…”
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Synthesis and antimicrobial activity of erythromycin-A oxime analogs by Pandey, Deepa, Katti, S.B, Haq, W, Tripathi, C.K.M

“…A few amino alcohol as well as ester derivatives of erythromycin-9-oxime have been synthesized in moderate yield. These compounds have shown antibacterial…”
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Thiazolidin-4-one and thiazinan-4-one derivatives analogous to rosiglitazone as potential antihyperglycemic and antidyslipidemic agents by Raza, Saman, Srivastava, Swayam P., Srivastava, Daya S., Srivastava, Arvind K., Haq, W., Katti, S.B.

“…A number of thiazolidin-4-one and thiazinan-4-one derivatives were prepared by three component condensation in one pot reaction method. These compounds were…”
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Antimalarial activity of novel 4-aminoquinolines active against drug resistant strains by Kondaparla, Srinivasarao, Soni, Awakash, Manhas, Ashan, Srivastava, Kumkum, Puri, Sunil K., Katti, S.B.

“…[Display omitted] •Novel side chain modified 4-aminoquinolines were designed and synthesized.•Assessment of 4-aminoquinolines for in vitro and in vivo…”
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Chiral Separation of Ormeloxifene Hydrochloride, a Non-steroidal Contraceptive Agent by Ahmad, Hafsa, Gupta, Varsha, Dwivedi, Atma Prakash, Katti, S. B., Dwivedi, Anil Kumar

“…Ormeloxifene hydrochloride (Centchroman) is once-a-week non-steroidal oral contraceptive agent marketed in India and other countries. In this study, we report…”
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Topological descriptors in modeling the HIV inhibitory activity of 2-aryl-3-pyridyl-thiazolidin-4-ones by Prabhakar, Y S, Rawal, R K, Gupta, M K, Solomon, V Raja, Katti, S B

“…The HIV-1 RT inhibitory activity of 2-(2,6-dihalophenyl)-3-(substituted pyridin-2-yl)-thiazolidin-4-ones has been analyzed with different topological…”
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