Search Results - "Katalin Szalai, Krisztina"

Harnessing dual-mode RIPK1 ligands for cross-species anti-necroptosis inhibitor compounds by Levente Petró, József, Bana, Péter, Linke, Nikolett, Eszter Szabó, Judit, Katalin Szalai, Krisztina, Kálomista, Ildikó, Gábor Vass, Csaba, Hornyánszky, Gábor, Greiner, István, Éles, János

“…[Display omitted] •Synthesis and biological evaluation of novel mixed type RIPK1 inhibitors.•Installation of a rigid acetylene moiety enhanced the…”
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hERG Optimization of Benzofuro−Pyridine and Pyrazino−Indole Derivatives as MCHR1 Antagonists by Huszár, József, Bozó, Éva, Beke, Gyula, Katalin Szalai, Krisztina, Kardos, Péter, Boros, András, Greiner, István, Éles, János

“…Obesity is a global epidemic associated with multiple severe diseases. Several pharmacotherapies have been investigated including the antagonists of melanin…”
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Design, synthesis and biological evaluation of novel cyclic malonamide derivatives as selective RIPK1 inhibitors by Petró, József Levente, Bényei, Gyula, Bana, Péter, Linke, Nikolett, Horti, Ferenc, Szabó, Judit Eszter, Szalai, Krisztina Katalin, Hornyánszky, Gábor, Greiner, István, Éles, János

“…[Display omitted] Receptor-interacting serine/threonine-protein kinase 1 (RIPK1) plays a key role in cell death and inflammation. RIPK1 is a well-established…”
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Novel bradykinin-1 antagonists containing a (1,2,3,4-tetrahydro-isoquinolin-1-yl)acetic acid scaffold by Huszár, József, Timár, Zoltán, Szalai, Krisztina Katalin, Keserű, György, Fülöp, Ferenc, Penke, Botond

“…A novel B 1 antagonist core was utilized and the effects of modification of its amide side chain on the biological activity were tested. The imino functional…”
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Aspartic acid scaffold in bradykinin B1 antagonists by Huszár, József, Timár, Zoltán, Bogár, Ferenc, Penke, Botond, Kiss, Róbert, Szalai, Krisztina Katalin, Schmidt, Éva, Papp, Andrea, Keserű, György

“…Several novel bradykinin B1 receptor (B1R) antagonists were synthesized utilizing a new aspartic acid scaffold. This core is derived from the highly potent…”
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