Search Results - "Kasaplar, Pınar"

A multi-substrate screening approach for the identification of a broadly applicable Diels–Alder catalyst by Kim, Hyejin, Gerosa, Gabriela, Aronow, Jonas, Kasaplar, Pinar, Ouyang, Jie, Lingnau, Julia B., Guerry, Paul, Farès, Christophe, List, Benjamin

“…When developing a synthetic methodology, chemists generally optimize a single substrate and then explore the substrate scope of their method. This approach has…”
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Approaching sub-ppm-level asymmetric organocatalysis of a highly challenging and scalable carbon–carbon bond forming reaction by Bae, Han Yong, Höfler, Denis, Kaib, Philip S. J., Kasaplar, Pinar, De, Chandra Kanta, Döhring, Arno, Lee, Sunggi, Kaupmees, Karl, Leito, Ivo, List, Benjamin

“…The chemical synthesis of organic molecules involves, at its very essence, the creation of carbon–carbon bonds. In this context, the aldol reaction is among…”
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Continuous Flow, Highly Enantioselective Michael Additions Catalyzed by a PS-Supported Squaramide by Kasaplar, Pinar, Rodríguez-Escrich, Carles, Pericàs, Miquel A

“…A polystyrene (PS) supported bifunctional squaramide organocatalyst promotes fast Michael addition of 2-hydroxy-1,4-naphthoquinone to nitroalkenes with very…”
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Polystyrene-Supported Diarylprolinol Ethers as Highly Efficient Organocatalysts for Michael-Type Reactions by Alza, Esther, Sayalero, Sonia, Kasaplar, Pinar, Almaşi, Diana, Pericàs , Miquel A.

“…α,α‐Diphenylprolinol methyl‐ and trimethylsilyl ethers anchored onto a polystyrene resin have been prepared by a copper‐catalyzed azide–alkyne cycloadditions…”
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Practical Silyl Protection of Ribonucleosides by Blaisdell, Thomas P, Lee, Sunggi, Kasaplar, Pinar, Sun, Xixi, Tan, Kian L

“…Herein we report the site-selective silylation of the ribonucelosides. The method enables a simple and efficient procedure for accessing suitably protected…”
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Synthesis and Topoisomerase I inhibitory properties of klavuzon derivatives by Akçok, İsmail, Mete, Derya, Şen, Ayhan, Kasaplar, Pınar, Korkmaz, Kemal S., Çağır, Ali

“…Asymmetric and racemic syntheses of heteroatom-substituted klavuzon derivatives are reported. Anti-proliferative activity of seven novel racemic klavuzon…”
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6-Bicycloaryl substituted ( S)- and ( R)-5,6-dihydro-2 H-pyran-2-ones: Asymmetric synthesis, and anti-proliferative properties by Kasaplar, Pınar, Yılmazer, Özgür, Çağır, Ali

“…( R)-Goniothalamin, is a member of styryl lactones, possesses selective cytotoxicity against cancer cell lines. In this work, replacement of styryl substituent…”
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A Polystyrene-Supported, Highly Recyclable Squaramide Organocatalyst for the Enantioselective Michael Addition of 1,3-Dicarbonyl Compounds to β-Nitrostyrenes by Kasaplar, Pinar, Riente, Paola, Hartmann, Caroline, Pericàs, Miquel A.

“…A chiral squaramide has been supported onto a polystyrene (PS) resin through a copper‐catalyzed azide–alkyne cycloaddition (CuAAC) reaction and used as a very…”
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Michael acceptor properties of 6-bicycloaryl substituted (R)-5,6-dihydro-2H-pyran-2-ones by Kasaplar, Pınar, Çakmak, Özgür Yılmazer, Çağır, Ali

“…Michael acceptor property of 5,6-dihydro-2H-pyran-2-ones is crucial for biological activity, and potency depends upon the Log P values and 3D structure of the…”
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Asymmetric Synthesis and Anti-Tumor Properties of Conformationally Constrained Analogues of (S)-And (R)-Goniothalamin by Kasaplar, Pınar

“…Naturally isolated 5-substituted-a,B-unsaturated-.-lactones gained great attention of researchers due to their cytotoxic and anti-tumor properties. Styryl…”
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A Polystyrene-Supported, Highly Recyclable Squaramide Organocatalyst for the Enantioselective Michael Addition of 1,3-Dicarbonyl Compounds to [beta]-Nitrostyrenes by Kasaplar, Pinar, Riente, Paola, Hartmann, Caroline, Pericas, Miquel A

“…A chiral squaramide has been supported onto a polystyrene (PS) resin through a copper-catalyzed azide-alkyne cycloaddition (CuAAC) reaction and used as a very…”
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6-Bicycloaryl substituted (S)-and (R)-5,6-dihydro-2H-pyran-2-ones : Asymmetric synthesis, and anti-proliferative properties by KASAPLAR, Pinar, YILMAZER, Ozgür, CAGIR, Ali

“…(R)-Goniothalamin, is a member of styryl lactones, possesses selective cytotoxicity against cancer cell lines. In this work, replacement of styryl substituent…”
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Synthesis of 5'-O-DMT-2'-O-TBS Mononucleosides Using an Organic Catalyst by Lee, Sunggi, Blaisdell, Thomas P, Kasaplar, Pinar, Sun, Xixi, Tan, Kian L

“…This unit describes a highly effective method to produce 5'-O-DMT-2'-O-TBS mononucleosides selectively using a small organic catalyst. This methodology avoids…”
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