Search Results - "Kartsev, V."

Functionally substituted 2-aminothiazoles as antimicrobial agents: in vitro and in silico evaluation by Petrou, A., Kartsev, V., Geronikaki, A., Glamočlija, J., Ciric, A., Sokovic, M.

“…Nine new functionally substituted derivatives of 2-aminothiazole were evaluated for antimicrobial activity using microdilution method against the panel of…”
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Appendix A. dithioloquinolinethiones as new potential multitargeted antibacterial and antifungal agents: Synthesis, biological evaluation and molecular docking studies by Kartsev, V., Shikhaliev, Khidmet S., Geronikaki, A., Medvedeva, Svetlana M., Ledenyova, Irina V., Krysin, Mikhail Yu, Petrou, A., Ciric, A., Glamoclija, J., Sokovic, M.

“…Herein we report the design, synthesis, molecular docking study and evaluation of antimicrobial activity of ten new dithioloquinolinethiones. The structures of…”
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Antibacterial activity of griseofulvin analogues as an example of drug repurposing by Geronikaki, A., Kartsev, V., Petrou, A., Akrivou, M.G., Vizirianakis, I.S., Chatzopoulou, F.M., Lichitsky, B., Sirakanyan, S., Kostic, M., Smiljkovic, M., Soković, M., Druzhilovskiy, D., Poroikov, V.

“…•Computational prediction of antibacterial activity.•Similarity assessment.•Antibacterial activity evaluation.•Docking to antibacterial targets. Griseofulvin…”
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Anti-inflammatory action of new hybrid N-acyl-[1,2]dithiolo-[3,4-c]quinoline-1-thione by Medvedeva, S.M., Petrou, A., Fesatidou, M., Gavalas, A., Geronikaki, A.A., Savosina, P.I., Druzhilovskiy, D.S., Poroikov, V.V., Shikhaliev, K.S., Kartsev, V.G.

“…Most of pharmaceutical agents display a number of biological activities. It is obvious that testing even one compound for thousands of biological activities is…”
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One-Pot Synthesis of 3-Oxocycloalka[c]pyridines by Sirakanyan, S. N., Geronikaki, A., Kartsev, V. G., Hakobyan, E. K., Hovakimyan, A. A.

“…A new efficient one-pot procedure has been developed for the synthesis of 1-substituted partially hydrogenated 3-oxocycloalka[ c ]pyridine-4-carbonitriles by…”
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Phenoptosis in arthropods and immortality of social insects by Kartsev, V. M.

“…In general, there are no drastic differences in phenoptosis patterns in plant and animal organisms. However, there are some specific features characteristic…”
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New Structural Modifications of Cotarnine Alkaloid Derivatives: Cotarnone and Dihydrocotarnine by Kartsev, V. G., Zubenko, A. A., Divaeva, L. N., Morkovnik, A. S., Baryshnikova, T. K., Shirinian, V. Z.

“…Simplest derivatives of the cotarnine alkaloid, like cotarnone and 1,2-dihydrocotarnine, undergo electrophilic Einhorn acylamidomethylation (with 60–95% yield)…”
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Effect of Plasma Deposition Production Parameters on Protective and Functional Coating Formation by Kravchenko, I. N., Zhachkin, S. Yu, Timashov, E. P., Trifonov, G. I., Kartsev, S. V., Kuznetsov, S. N.

“…Improvement of plasma deposition wear-resistant coatings technology is demonstrated. At the same time, special attention is paid to one of the most important…”
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Molecular docking, design, synthesis and biological evaluation of novel 2,3-aryl-thiazolidin-4-ones as potent NNRTIs by Geronikaki, A., Petrou, A., Kartsev, V., Eleftheriou, P., Boga, R., Bartolo, B., Crespan, E., Franco, G., Maga, G.

“…Nonnucleoside reverse transcriptase inhibitors (NNRTIs) remain the most promising anti-AIDS agents that target the HIV-1 reverse transcriptase enzyme (RT)…”
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Imidazole Derivative As a Novel Translation Inhibitor by Lukianov, D A, Buev, V S, Ivanenkov, Y A, Kartsev, V G, Skvortsov, D A, Osterman, I A, Sergiev, P V

“…Searching for novel compounds with antibiotic activity and understanding their mechanism of action is extremely important. The ribosome is one of the main…”
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Synthesis of Benzoannelated Canthin-6-One Analogs by Sen’ko, O. A., Dybenko, A. G., Garazd, M. M., Kartsev, V. G.

“…Benzoannelated structural analogs of the natural alkaloid canthin-6-one were synthesized…”
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Synthesis of New Heterocyclic Systems on the Basis of 7-Benzyl-3-chloro-1-(morpholin-4-yl)-5,6,7,8-tetrahydro-2,7-naphthiridine-4-carbonitrile by Sirakanyan, S. N., Kartsev, V. G., Hakobyan, E. K., Hovakimyan, A. A.

“…Methods have been developed for the synthesis of new 8-amino-3-benzyl-5-(morpholin-4-yl)-1,2,3,4-tetrahydropyrimido[4′,5′: 4,5]thieno[2,3- c…”
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To evaluation of the state of the own macroscopic force field of liquids by Kartsev, V. N., Shtykov, S. N., Pankin, K. E.

“…The work analyzes both literature data on the dependence of the internal liquid pressure on thermodynamic parameters of state and theoretical ideas of the…”
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Optimization of Plasma Deposition and Coating Plasma Fusion Parameters and Regimes by Kravchenko, I. N., Kartsev, S. V., Kuznetsov, Yu. A., Velichko, S. A.

“…Results are provided for studies concerning the choice of parameters and optimization of plasma spraying regimes (plasmatron arc current strength is 170 – 175…”
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Method for Protecting Plasma-Jet Hard-Facing by Gas Powder Flow by Kravchenko, I. N., Kartsev, S. V., Kuznetsov, Yu. A.

“…The results of investigation of the rate of gas flow and powder particles flying at plasma-jet hard-facing by a constricted arc in gas powder protective media…”
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Synthesis of N-Acylamino-Acid Derivatives of Cytisine by Yazlovitskii, A. V., Garazd, M. M., Kartsev, V. G.

“…N -acylamino-acid derivatives of cytisine were prepared by reacting cytisine with methyl esters of aminoacid isocyanates…”
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Pyridine—Azepine Structural Modification of 3,4-Dihydro-nor-isoharmine by Zubenko, A. A., Morkovnik, A. S., Divaeva, L. N., Kartsev, V. G., Anisimov, A. A., Suponitsky, K. Yu

“…Structural modification of 3,4-dihydro-nor-isoharmine through expansion of the dihydropyridine ring to dihydroazepine was accomplished in two stages including…”
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Chemical Modification of Plant Alkaloids. 8. Stereocontrolled T-Reactions of (1R,5S,12S)-Tetrahydrocytisine Derivatives by Krasnov, K. A., Kartsev, V. G., Dobrokhotova, E. V., Kultyshkina, E. K., Chernikova, N. Yu, Dorovatovskii, P. V., Zubavichus, Ya. V., Khrustalev, V. N.

“…New heterocyclic quinolizidine systems were prepared from (1 R ,5 S ,12 S )-tetrahydrocytisine. The synthetic scheme included arylation of tetrahydrocytisine…”
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Effect of Component Surface Preparation on Coating Adhesive Strength during Plasma Spraying by Kravchenko, I. N., Kartsev, S. V., Velichko, S. A., Kuznetsov, Yu. A., Pastukhov, A. G.

“…Results of studying the effect of component surface preparation on coating adhesive strength with a substrate are presented. A new method of surface…”
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Evaluation of the Thermal Stability of Composite Powder Materials in a Plasma Jet by Kravchenko, I. N., Kuznetsov, Yu. A., Galinovskii, A. L., Velichko, S. A., Ionov, P. A., Kartsev, S. V.

“…The paper presents the results of studying thermal stability of materials operating in a plasma jet under high temperature and rapid thermal load variation…”
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