Search Results - "Kapdi, Anant"

Transition-Metal-Catalyzed Direct Arylation of (Hetero)Arenes by C----H Bond Cleavage by Ackermann, Lutz, Vicente, Rubén, Kapdi, Anant R

“…The area of transition-metal-catalyzed direct arylation through cleavage of C---H bonds has undergone rapid development in recent years, and is becoming an…”
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Late‐Stage Peptide Diversification by Position‐Selective C−H Activation by Wang, Wei, Lorion, Mélanie M., Shah, Jagrut, Kapdi, Anant R., Ackermann, Lutz

“…The late‐stage modification of structurally complex peptides bears great potential for drug discovery, crop protection, and the pharmaceutical industry, among…”
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Anti-cancer palladium complexes: a focus on PdX2L2, palladacycles and related complexes by Kapdi, Anant R, Fairlamb, Ian J S

“…Much success has been achieved with platinum-based chemotherapeutic agents, i.e. through interactions with DNA. The long-term application of Pt complexes is…”
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DMSO‐Assisted K3PO4‐Catalyzed Cooperative Metal‐Free, Base‐Free Etherification of Chloroheteroarenes at Low Temperature by Khandagale, Deepali, Kori, Santosh, Kapdi, Anant R.

“…Etherification of chloroheteroarenes was performed at low temperatures under metal‐free, ligand‐free and base‐free conditions, that is, the reaction is…”
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DMSO-Assisted K 3 PO 4 -Catalyzed Cooperative Metal-Free, Base-Free Etherification of Chloroheteroarenes at Low Temperature by Khandagale, Deepali, Kori, Santosh, Kapdi, Anant R

“…Etherification of chloroheteroarenes was performed at low temperatures under metal-free, ligand-free and base-free conditions, that is, the reaction is…”
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DNA-encoded libraries via late-stage functionalization strategies: a review by Sahu, Rajesh, Yadav, Saurav, Nath, Suvadeep, Banerjee, Joydeep, Kapdi, Anant R

“…The hit finding strategy in drug discovery has undergone a tremendous change in the past decade with the advent of DNA-encoded libraries with diverse chemical…”
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Phenothiazine-Based Cu(II)-Selective Fluorescent Sensor: GHK-Cu Sensing Applications by Sahu, Rajesh, Yadav, Saurav, Gunturu, Krishna Chaitanya, Kapdi, Anant R.

“…Sensing important metals in different environments is an important area and involves the development of a wide variety of metal-sensing materials. The…”
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Diverse meta-C–H Functionalization of Amides by Gholap, Aniket, Bag, Sukdev, Pradhan, Sukumar, Kapdi, Anant R, Maiti, Debabrata

“…Overriding the preference for favorable proximal metalation by ortho-directing amide group, a pyrimidine-based directing group (DG) has been demonstrated for…”
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Cobalt(II)/N‑Hydroxyphthalimide-Catalyzed Cross-Dehydrogenative Coupling Reaction at Room Temperature under Aerobic Condition by Patil, Mahendra R, Dedhia, Noopur P, Kapdi, Anant R, Kumar, A.Vijay

“…This work reports a cobalt­(II)/N-hydroxyphthalimide (NHPI)-catalyzed cross-dehydrogenative oxidative coupling of N-aryl tetrahydroisoquinolines with various…”
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Cu(II)/PTABS-Promoted, Chemoselective Amination of HaloPyrimidines by Phulwale, Vikram, Shet, Harshita, Gunturu, Krishna Chaitanya, Rout, Smruti Rekha, Dandela, Rambabu, Adhav, Suyog, Kapdi, Anant R.

“…Chemoselective amination is a highly desired synthetic methodology, given its importance as a possible strategy to synthesize various drug molecules and…”
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Ambient‐Temperature, Metal‐Free, CDI‐Mediated Ex‐Situ Conversion of Acids to Amides: A Useful Late‐Stage Strategy by Patel, Manisha A., Kapdi, Anant R.

“…An efficient ex‐situ method for the amidation of carboxylic acids mediated by CDI has been disclosed herewith. This metal‐free strategy is performed at ambient…”
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Ubiquitous Role of Phosphine‐Based Water‐Soluble Ligand in Promoting Catalytic Reactions in Water by Patel, Manisha A., Kapdi, Anant R.

“…Catalysis has been at the forefront of the developments that has revolutionised synthesis and provided the impetus in the discovery of platform technologies…”
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Strategies for the Synthesis of Fluorinated Nucleosides, Nucleotides and Oligonucleotides by Shet, Harshita, Sahu, Rajesh, Sanghvi, Yogesh S., Kapdi, Anant R.

“…Fluorinated nucleosides and oligonucleotides are of specific interest as probes for studying nucleic acids interaction, structures, biological transformations,…”
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Phosphine ligands based on the ferrocenyl platform: Advances in catalytic cross-couplings by Bandaru, Siva Sankar Murthy, Shah, Jagrut, Bhilare, Shatrughn, Schulzke, Carola, Kapdi, Anant R., Roger, Julien, Hierso, Jean-Cyrille

“…•Ferrocenyl monophosphine ligands in non-chiral carbon–carbon bond formation.•P,N–, P,O–and P,S–ferrocenyl monophosphine ligands for cross-coupling…”
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Ambient Temperature Metal‐Free Thiomethylation of Chloroheteroarenes and Chloropurines by Patel, Manisha A., Vora, Raj K., Sanghvi, Yogesh S., Kapdi, Anant R.

“…Herein, we report an in‐situ mild and metal‐free protocol for thiomethylation of heteroarenes in high yields. The thiomethylation of various chloropurines,…”
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Pd/PTABS: Catalyst for Room Temperature Amination of Heteroarenes by Murthy Bandaru, Siva Sankar, Bhilare, Shatrughn, Chrysochos, Nicolas, Gayakhe, Vijay, Trentin, Ivan, Schulzke, Carola, Kapdi, Anant R

“…A mild and highly efficient catalytic amination procedure for chloroheteroarenes at ambient temperature using the Pd/PTABS catalytic system is reported. The…”
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Discovery, Synthesis, and Scale-up of Efficient Palladium Catalysts Useful for the Modification of Nucleosides and Heteroarenes by Bhilare, Shatrughn, Shet, Harshita, Sanghvi, Yogesh S, Kapdi, Anant R

“…Nucleic acid derivatives are imperative biomolecules and are involved in life governing processes. The chemical modification of nucleic acid is a fascinating…”
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Room-Temperature Amination of Chloroheteroarenes in Water by a Recyclable Copper(II)-Phosphaadamantanium Sulfonate System by Parmar, Udaysinh, Somvanshi, Dipesh, Kori, Santosh, Desai, Aman A, Dandela, Rambabu, Maity, Dilip K, Kapdi, Anant R

“…Buchwald–Hartwig amination of chloroheteroarenes has been a challenging synthetic process, with very few protocols promoting this important transformation at…”
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Pd/PTABS: Low-Temperature Thioetherification of Chloro(hetero)arenes by Bandaru, Siva Sankar Murthy, Bhilare, Shatrughn, Cardozo, Jesvita, Chrysochos, Nicolas, Schulzke, Carola, Sanghvi, Yogesh S, Gunturu, Krishna Chaitanya, Kapdi, Anant R

“…The thioetherification of heteroaryl chlorides is an essential synthetic methodology that provides access to bioactive drugs and agrochemicals. Due to their…”
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Nucleoside/Nucleotide or Nucleic Acid Modification & Applications by Kapdi, Anant R., Arseniyadis, Stellios, Lakshman, Mahesh K.

“…“The field of nucleosides, nucleotides, and nucleic acids has been in existence for some decades, leading to a notion that the area is well‐explored and/or…”
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