Search Results - "Kalampaliki, Amalia D."
-
1
Synthesis and Biological Evaluation of Resveratrol Methoxy Derivatives
Published in Molecules (Basel, Switzerland) (01-07-2023)“…Resveratrol, a naturally occurring stilbene, exhibits numerous beneficial health effects. Various studies have demonstrated its diverse biological actions,…”
Get full text
Journal Article -
2
Synthesis and Biological Evaluation of 2-Substituted Quinazolin-4(3 H )-Ones with Antiproliferative Activities
Published in Molecules (Basel, Switzerland) (01-12-2023)“…Sixteen new 2-substituted quinazolines were synthesized using a straightforward methodology starting from 2-methoxybezoic acid or 3-methoxy-2-naphthoic acid…”
Get full text
Journal Article -
3
A Three-Step, Gram-Scale Synthesis of Hydroxytyrosol, Hydroxytyrosol Acetate, and 3,4-Dihydroxyphenylglycol
Published in Molecules (Basel, Switzerland) (05-09-2019)“…Hydroxytyrosol and two other polyphenols of olive tree, hydroxytyrosol acetate and 3,4-dihydroxyphenylglycol, are known for a wide range of beneficial…”
Get full text
Journal Article -
4
Chemometrically Assisted Optimization of Pregabalin Fluorescent Derivatization Reaction with a Novel Xanthone Analogue and Validation of the Method for the Determination of Pregabalin in Bulk via a Plate Reader
Published in Molecules (Basel, Switzerland) (17-03-2022)“…Quantitation of chromophore-free analytes is always a challenge. To this purpose, derivatization of the analyte constitutes a common strategy, leading to a…”
Get full text
Journal Article -
5
3,6-Dihydro-5H-pyrazolo [4′,3′:5,6]pyrano[3,4-b]indol-5-one
Published in MolBank (01-09-2022)“…Pyrano [3,4-b]indol-1(9H)-ones and indolo [2,3-c]coumarins are important classes of heterocyclic compounds with versatile biological activities. Herein, we…”
Get full text
Journal Article -
6
Design and Synthesis of Pyrazole-Based Macrocyclic Kinase Inhibitors Targeting BMPR2
Published in ACS medicinal chemistry letters (08-06-2023)“…Bone morphogenetic protein (BMP) signaling is mediated by transmembrane protein kinases that form heterotetramers consisting of type-I and type-II receptors…”
Get full text
Journal Article -
7
The pyrazolo[4,3-c]pyrazole core as a novel and versatile scaffold for developing dual DYRK1A-CLK1 inhibitors targeting key processes of Alzheimer's disease pathology
Published in European journal of medicinal chemistry reports (01-12-2024)“…In the current study, we designed, synthesized, and characterized a series of substituted pyrazolo[4,3-c]pyrazoles. These novel compounds were evaluated in…”
Get full text
Journal Article -
8
Synthesis of novel xanthone and acridone carboxamides with potent antiproliferative activities
Published in Arabian journal of chemistry (01-11-2020)“…[Display omitted] Several new amino-substituted acridone and xanthone derivatives have been designed and synthesized, using an efficient methodology from…”
Get full text
Journal Article -
9
3,6-Dihydro-5IH/I-pyrazolo [4′,3′:5,6]pyrano[3,4-Ib/I]indol-5-one
Published in MolBank (01-07-2022)“…Pyrano [3,4-b]indol-1(9H)-ones and indolo [2,3-c]coumarins are important classes of heterocyclic compounds with versatile biological activities. Herein, we…”
Get full text
Journal Article -
10
Synthesis, spectroscopic and computational evaluation of a xanthene-based fluorogenic derivatization reagent for the determination of primary amines
Published in Dyes and pigments (01-12-2021)“…To detect an analyte, typically at the sub-nanomolar scale, extremely sensitive analytical tools are required. Fluorescence is the spectroscopy of choice to…”
Get full text
Journal Article -
11
Corrigendum to “The pyrazolo[4,3-c]pyrazole core as a novel and versatile scaffold for developing dual DYRK1A-CLK1 inhibitors targeting key processes of Alzheimer's disease pathology” [Europ. J. Med. Chem. Rep. 12 (2024) 100193]
Published in European journal of medicinal chemistry reports (01-10-2024)Get full text
Journal Article