Search Results - "Kadry, Asmaa M."
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Green synthesis, biological and molecular docking of some novel sulfonamide thiadiazole derivatives as potential insecticidal against Spodoptera littoralis
Published in Scientific reports (06-11-2023)“…Although crop plants provide the majority of human food, pests and insects frequently cause huge economic losses. In order to develop innovative insecticidal…”
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Synthesis and antidiabetic activity of novel triazole derivatives containing amino acids
Published in Journal of heterocyclic chemistry (01-06-2020)“…New series of triazole derivatives coupled with amino acids 1a‐h were obtained via multicomponent reaction of 2‐hydroxy benzaldehyde or 2‐hydroxy acetophenone…”
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Ultrasound-assisted green synthesis of triazole-based azomethine/thiazolidin-4-one hybrid inhibitors for cancer therapy through targeting dysregulation signatures of some Rab proteins
Published in Green chemistry letters and reviews (02-01-2023)“…The overexpression of Rab proteins was linked to cancer development, making this family of proteins an attractive drug target for the identification of novel…”
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Spiro heterocycles bearing piperidine moiety as potential scaffold for antileishmanial activity: synthesis, biological evaluation, and in silico studies
Published in Journal of enzyme inhibition and medicinal chemistry (01-12-2023)“…New spiro-piperidine derivatives were synthesised via the eco-friendly ionic liquids in a one-pot fashion. The in vitro antileishmanial activity against…”
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Efficient and Recoverable Bio-Organic Catalyst Cysteine for Synthesis, Docking Study, and Antifungal Activity of New Bio-Active 3,4-Dihydropyrimidin-2(1H)‑ones/thiones Under Microwave Irradiation
Published in ACS omega (05-07-2022)“…An eco-friendly green bio-organic catalyst and low-cost 3,4-dihydropyrimidin-2(1H)-ones/thione derivatives 4–7 have been synthesized using a high-yield,…”
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Synthesis, docking and characterization of some novel 5-(S-alkyl)-1.3.4-thiadiazole-2-carboxamide derivatives as anti-inflammatory and antibacterial agents
Published in BMC chemistry (27-07-2024)“…Because of the great pharmacological and industrial significance of 1,3,4-thiadiazole and its related compounds, researchers are still very interested in them…”
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Synthesis, docking and biological evaluation of purine-5- N -isosteresas anti-inflammatory agents
Published in RSC advances (28-05-2024)“…An operationally simple one-pot three-component and convenient synthesis method for a series of diverse purine analogues of 5-amino-7-(substituted)-…”
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Correction: Synthesis, docking and biological evaluation of purine-5- N -isosteres as anti-inflammatory agents
Published in RSC advances (12-07-2024)“…[This corrects the article DOI: 10.1039/D4RA02970D.]…”
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An efficient eco-friendly, simple, and green synthesis of some new spiro-N-(4-sulfamoyl-phenyl)-1,3,4-thiadiazole-2-carboxamide derivatives as potential inhibitors of SARS-CoV-2 proteases: drug-likeness, pharmacophore, molecular docking, and DFT exploration
Published in Molecular diversity (01-02-2024)“…Introduction The coronavirus disease 2019 (COVID-19) pandemic has caused a global health crisis. The severe acute respiratory syndrome coronavirus 2…”
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An operationally simple, one‐pot, convenient synthesis, and in vitro anti‐inflammatory activity of some new spirotriazolotriazine derivatives
Published in Journal of heterocyclic chemistry (01-01-2024)“…The wide biological actions of triazolotriazine hybrids, benzene‐sulfonamide derivatives, exhibit a good chance of displaying in vitro anti‐inflammatory…”
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Thiadiazole/Thiadiazine Derivatives as Insecticidal Agent: Design, Synthesis, and Biological Assessment of 1,3,4-(Thiadiazine/Thiadiazole)-Benzenesulfonamide Derivatives as IGRs Analogues against Spodoptera littoralis
Published in Journal of agricultural and food chemistry (22-05-2024)“…In keeping with our investigation, a simple and practical synthesis of novel heterocyclic compounds with a sulfamoyl moiety that can be employed as…”
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Novel 2‑Acetamido-2-ylidene-4-imidazole Derivatives (El-Saghier Reaction): Green Synthesis, Biological Assessment, and Molecular Docking
Published in ACS omega (22-08-2023)“…El-Saghier reaction is the novel, general, and green reaction of various amines with ethyl cyanoacetate and ethyl glycinate hydrochloride. A new series of…”
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Green synthesis, antileishmanial activity evaluation, and in silico studies of new amino acid-coupled 1,2,4-triazoles
Published in Medicinal chemistry research (15-02-2019)“…Candidates of triazole-containing amino acid derivatives 5a−k were prepared under green chemistry conditions via multicomponent reaction using lemon juice as…”
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Synthesis and antimicrobial activity of some novel 1,2-dihydro-[1,2,4]triazolo[1,5-]pyrimidines bearing amino acid moiety
Published in RSC advances (13-01-2021)“…A new series of [1,2,4]-triazole bearing amino acid derivatives 2a-d - 9a-d were synthesized under green chemistry conditions via multicomponent reaction using…”
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Synthesis, Structural Stability Calculation, and Antibacterial Evaluation of Novel 3,5-Diphenylcyclohex-2-en-1-one Derivatives
Published in Synthetic communications (01-01-2015)“…Starting with 3,5-diphenylcyclohex-2-en-1-one, 3,5-diphenylcyclohex-2-en-1-semicarbazone, 1-chloro-3,5-diphenylcyclohex-2-en-2-carbaldehyde, and…”
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Utility of amino acid coupled 1,2,4-triazoles in organic synthesis: synthesis of some new antileishmainal agents
Published in Bulletin of the Chemical Society of Ethiopia (01-01-2018)“…Starting from 3-amino-5-(2-hydroxyphenyl) amino acid coupled triazoles 1a-e, new 3-(2-hydroxyphenyl)-3H-imidazo[2,1-c][1,2,4]triazol-6(5/f)-one 2a,b, 3b,d, 6a…”
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Correction: Synthesis, docking and biological evaluation of purine-5--isosteres as anti-inflammatory agents
Published in RSC advances (12-07-2024)“…Correction for 'Synthesis, docking and biological evaluation of purine-5- N -isosteres as anti-inflammatory agents' by Ahmed M. El-Saghier et al. , RSC Adv. ,…”
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18
Synthesis, docking and biological evaluation of purine-5--isosteresas anti-inflammatory agents
Published in RSC advances (03-06-2024)“…An operationally simple one-pot three-component and convenient synthesis method for a series of diverse purine analogues of 5-amino-7-(substituted)- N…”
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