Search Results - "Kadowaki, Chie"

Syntheses of the AB and EFGH ring segments of gambierol by Kadota, Isao, Kadowaki, Chie, Park, Choul-Hong, Takamura, Hiroyoshi, Sato, Kumi, Chan, Philip W.H, Thorand, Stephan, Yamamoto, Yoshinori

“…Stereocontrolled syntheses of the AB and EFGH ring systems of gambierol ( 1 ) are described. The two key intermediates 3 and 55 , representing the AB and EFGH…”
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A novel convergent approach to trans-fused polyether frameworks based on the reaction of vinylstannanes and triflates and its application to a synthetic study of the EFGH ring system of gambierol by Kadowaki, Chie, Chan, Philip W.H, Kadota, Isao, Yamamoto, Yoshinori

“…A new strategy for the convergent assembly of six-membered polycyclic ether ring fragments has been developed based upon the novel reaction between…”
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Synthetic studies towards gambierol. Part 2: Synthesis of the EFGH ring segment by Kadota, Isao, Kadowaki, Chie, Takamura, Hiroyoshi, Yamamoto, Yoshinori

“…The EFGH ring segment of gambierol was synthesized from 2-deoxy- d-ribose in 40 steps. The present synthesis includes a SmI 2-mediated reductive cyclization…”
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Imidazopyridine derivatives as potent and selective Polo-like kinase (PLK) inhibitors by Sato, Yoshiyuki, Onozaki, Yu, Sugimoto, Tetsuya, Kurihara, Hideki, Kamijo, Kaori, Kadowaki, Chie, Tsujino, Toshiaki, Watanabe, Akiko, Otsuki, Sachie, Mitsuya, Morihiro, Iida, Masato, Haze, Kyosuke, Machida, Takumitsu, Nakatsuru, Yoko, Komatani, Hideya, Kotani, Hidehito, Iwasawa, Yoshikazu

“…Design and optimization of novel imidazopyridine derivatives led to the identification of a potent and selective PLK inhibitor 36. A novel class of…”
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Practical Synthesis of a HIV Integrase Inhibitor by Zhong, Yong-Li, Pipik, Brenda, Lee, Jaemoon, Kohmura, Yoshinori, Okada, Shigemitsu, Igawa, Kazunobu, Kadowaki, Chie, Takezawa, Akihiro, Kato, Shinji, Conlon, David A, Zhou, Hua, King, Anthony O, Reamer, Robert A, Gauthier, Jr, Donald R, Askin, David

“…A practical and efficient synthesis of the potent HIV integrase inhibitor 1 is described. Starting from readily available 3,4-dihydro-2H-pyran, the six-step…”
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Practical Synthesis of a Neuropeptide Y Antagonist via Stereoselective Addition to a Ketene by Iida, Takehiko, Satoh, Hiroki, Maeda, Kenji, Yamamoto, Yuhei, Asakawa, Ken-ichi, Sawada, Naotaka, Wada, Toshihiro, Kadowaki, Chie, Itoh, Takahiro, Mase, Toshiaki, Weissman, Steven A, Tschaen, Dave, Krska, Shane, Volante, R. P

“…The synthesis of neuropeptide Y antagonist 1, currently under clinical investigation for the treatment of obesity, is described. The convergent synthesis from…”
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Synthesis of the E ring of gambierol by Kadota, Isao, Kadowaki, Chie, Yoshida, Noriko, Yamamoto, Yoshinori

“…The synthesis of the E ring of gambierol was achieved from D-ribose via the intramolecular reaction of allylstannane with an aldehyde as a key step. The…”
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Why are benzimidazoles efficiently acylated with esters? Identification of a tetrahedral hemiacetal alkoxide intermediate by Asakawa, Ken-ichi, Dannenberg, J.J., Fitch, Kenneth J., Hall, Stan S., Kadowaki, Chie, Karady, Sandor, Kii, Satoshi, Maeda, Kenji, Marcune, Benjamin F., Mase, Toshiaki, Miller, Ross A., Reamer, Robert A., Tschaen, David M.

“…[Display omitted] 2-Lithio benzimidazoles were acylated with esters, lactones, and lactams. The tetrahedral hemiacetal intermediates responsible for the…”
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Palladium catalyzed addition of carbon pronucleophiles to conjugated enynes by Gevorgyan, Vladimir, Kadowaki, Chie, Salter, Matthew M., Kadota, Isao, Saito, Shinichi, Yamamoto, Yoshinori

“…Palladium catalyzed addition of certain carbon pronucleophiles 2 to conjugated enynes 1 afforded the corresponding allenes 3 in good to excellent yields. The…”
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