Search Results - "Jones, Eric D"

Small molecule inhibitors of the LEDGF site of human immunodeficiency virus integrase identified by fragment screening and structure based design by Peat, Thomas S, Rhodes, David I, Vandegraaff, Nick, Le, Giang, Smith, Jessica A, Clark, Lisa J, Jones, Eric D, Coates, Jonathan A V, Thienthong, Neeranat, Newman, Janet, Dolezal, Olan, Mulder, Roger, Ryan, John H, Savage, G Paul, Francis, Craig L, Deadman, John J

“…A fragment-based screen against human immunodeficiency virus type 1 (HIV) integrase led to a number of compounds that bound to the lens epithelium derived…”
Get full text

Design of a series of bicyclic HIV-1 integrase inhibitors. Part 2: Azoles: Effective metal chelators by Le, Giang, Vandegraaff, Nick, Rhodes, David I., Jones, Eric D., Coates, Jonathan A.V., Thienthong, Neeranat, Winfield, Lisa J., Lu, Long, Li, Xinming, Yu, Changjiang, Feng, Xiao, Deadman, John J.

“…Synthesis of a diverse set of azoles and their utilizations as an amide isostere in the design of HIV integrase inhibitors is described. The Letter identified…”
Get full text

Antiviral agents 3. Discovery of a novel small molecule non-nucleoside inhibitor of Hepatitis B Virus (HBV) by Crosby, Ian T., Bourke, David G., Jones, Eric D., Jeynes, Tyrone P., Cox, Susan, Coates, Jonathan A.V., Robertson, Alan D.

“…The discovery of a small molecule non-nucleoside inhibitor of Hepatitis B Virus is described. During our work on conocurvone derived naphthoquinone ‘trimers’…”
Get full text

Correction: Small Molecule Inhibitors of the LEDGF Site of Human Immunodeficiency Virus Integrase Identified by Fragment Screening and Structure Based Design by Peat, Thomas S., Rhodes, David I., Vandegraaff, Nick, Le, Giang, Smith, Jessica A., Clark, Lisa J., Jones, Eric D., Coates, Jonathan A. V., Thienthong, Neeranat, Newman, Janet, Dolezal, Olan, Mulder, Roger, Ryan, John H., Savage, G. Paul, Francis, Craig L., Deadman, John J.

Get full text

The Effect of Preoperative Education Prior to Hip or Knee Arthroplasty on Immediate Postoperative Outcomes by Jones, Eric D., Davidson, Lynda J., Cline, Thomas W.

“…There is ample research demonstrating improved patient outcomes when using an enhanced recovery program. However, the literature reporting the impact of…”
Get full text

Condensed-Phase and Oxidation Reaction Behavior of Ti/2B Foils in Varied Gaseous Environments by Reeves, Robert V, Rodriguez, Mark A, Jones, Eric D, Adams, David P

“…The effect of gaseous environment on self-propagating reactions in Ti/2B multilayer foils was studied. Multilayers with reactant layer periodicities from 50 to…”
Get full text

Rare-earth transition-metal intermetallic compounds produced via self-propagating, high-temperature synthesis by McDonald, Joel P., Rodriguez, Mark A., Jones, Eric D., Adams, David P.

“…Several binary intermetallic compounds—each containing a rare-earth (RE) element paired with a transition metal (TM)—were prepared by self-propagating,…”
Get full text

Design of a series of bicyclic HIV-1 integrase inhibitors. Part 1: Selection of the scaffold by Jones, Eric D., Vandegraaff, Nick, Le, Giang, Choi, Neil, Issa, William, Macfarlane, Katherine, Thienthong, Neeranat, Winfield, Lisa J., Coates, Jonathan A.V., Lu, Long, Li, Xinming, Feng, Xiao, Yu, Changjiang, Rhodes, David I., Deadman, John J.

“…HIV integrase inhibitors based on a novel bicyclic pyrimidinone core is presented. Nine variations of the core scaffold are evaluated leading to optimization…”
Get full text

Antiviral agents 2. Synthesis of trimeric naphthoquinone analogues of conocurvone and their antiviral evaluation against HIV by Crosby, Ian T., Bourke, David G., Jones, Eric D., de Bruyn, Paula J., Rhodes, David, Vandegraaff, Nick, Cox, Susan, Coates, Jonathan A.V., Robertson, Alan D.

“…The synthesis of a new series of conocurvone analogues is presented that explores the importance of the pyran rings of conocurvone, their degree of…”
Get full text

Structural basis for a new mechanism of inhibition of HIV-1 integrase identified by fragment screening and structure-based design by Rhodes, David I, Peat, Thomas S, Vandegraaff, Nick, Jeevarajah, Dharshini, Le, Giang, Jones, Eric D, Smith, Jessica A, Coates, Jonathan A V, Winfield, Lisa J, Thienthong, Neeranat, Newman, Janet, Lucent, Del, Ryan, John H, Savage, G Paul, Francis, Craig L, Deadman, John J

“…HIV-1 integrase is a clinically validated therapeutic target for the treatment of HIV-1 infection, with one approved therapeutic currently on the market. This…”
Get full text

Discovery of potent HIV integrase inhibitors active against raltegravir resistant viruses by Le, Giang, Vandegraaff, Nick, Rhodes, David I., Jones, Eric D., Coates, Jonathan A.V., Lu, Long, Li, Xinming, Yu, Changjiang, Feng, Xiao, Deadman, John J.

“…A series of novel HIV integrase inhibitors active against rategravir resistant strains are reported. Initial SAR studies revealed that activities against…”
Get full text

Microwave-promoted synthesis of 3-amino-substituted 1,2-benzisoxazoles by Smith, Jessica A, Le, Giang, Jones, Eric D, Deadman, John

“…1,2-benzisoxazole derivatives have been the focus of numerous studies, due to their biological and chemical interest. We demonstrate an efficient synthesis of…”
Get more information

Letter to the Editor by Liu, Jinjin, Zhong Mingjin, Jones, Eric D, Davidson, Lynda J, Cline, Thomas W

Get full text

Letter to the Editor by Liu, Jinjin, Zhong, Mingjin, Jones, Eric D., Davidson, Lynda J., Cline, Thomas W.

Get full text

Letter to the Editor by Liu, Jinjin, Zhong, Mingjin, Jones, Eric D., Davidson, Lynda J., Cline, Thomas W.

Get full text

Letter to the Editor by Liu, Jinjin, Zhong, Mingjin, Jones, Eric D, Davidson, Lynda J, Cline, Thomas W

Get full text

Mathematics Instruction for Secondary Students with Learning Disabilities by Jones, Eric D

“…The poor achievement of secondary students with learning disabilities in mathematics is often affected by prior low achievement, low expectations for success,…”
Get more information

Mathematics: Educational Tools for Diverse Learners by Carnine, Doug, Jones, Eric D, Dixon, Robert

“…Discusses emerging tools implied by recent reform efforts in mathematics education. Critiques current textbooks based on three factors (rate content is…”
Get more information

Direct observation of spinlike reaction fronts in planar energetic multilayer foils by McDonald, Joel P., Hodges, V. Carter, Jones, Eric D., Adams, David P.

“…Propagating reactions in initially planar cobalt/aluminum exothermic multilayer foils have been investigated using high-speed digital photography. Real-time…”
Get full text

Curriculum-Based Assessment: Testing What Is Taught and Teaching What Is Tested by Jones, Eric D., Southern, W. Thomas, Brigham, Frederick J.

“…Over the last 15 years empirical studies have documented positive effects resulting from the use of curriculum-based assessment (CBA) procedures on the…”
Get full text